
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| Histamine H1 receptor | Homo sapiens | P35367 | >10000 nM | BindingDB | |||
| Histamine H2 receptor | Homo sapiens | P25021 | >10000 nM | BindingDB | |||
| Histamine H3 receptor | Homo sapiens | Q9Y5N1 | 5.37 nM | BindingDB | |||
| Histamine H3 receptor | Rattus norvegicus | Q9QYN8 | 24.5 nM|25 nM|66 nM | BindingDB | |||
| Histamine H4 receptor | Homo sapiens | Q9H3N8 | >10000 nM | BindingDB |