| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| NPC1-like intracellular cholesterol transporter 1 | Homo sapiens | Q9UHC9 | >10000 nM | | | | BindingDB |
| LNCaP | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | > 200000.0 nM|> 50000.0 nM|> 20000.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | > 50000.0 nM | | | NPASS |
| Niemann-Pick C1-like protein 1 | Homo sapiens | Q9UHC9 | > 10000.0 nM | | | | NPASS |
| T47D | Homo sapiens | | | = 2550.0 nM | | | NPASS |
| SMMC-7721 | Homo sapiens | | | > 20000.0 nM | | | NPASS |
| SW480 | Homo sapiens | | | > 20000.0 nM | | | NPASS |
| Sex hormone-binding globulin | Homo sapiens | P04278 | | | 14 nM | | BindingDB |
| Solute carrier organic anion transporter family member [3-691] | Zebrafish | | | | | 6.8e+2 nM | BindingDB |
| Trypanosoma cruzi | Trypanosoma cruzi | | | > 300000.0 nM|= 62000.0 nM|= 13840.0 nM | | | NPASS |
| Testis-specific androgen-binding protein | Homo sapiens | P04278 | | | = 14.45 nM | | NPASS |
| PC-12 | Rattus norvegicus | | | = 0.29 nM | | | NPASS |
| J774.A1 | Mus musculus | | | = 141.0 nM | | | NPASS |
| Jurkat | Homo sapiens | | | = 46500.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 47800.0 nM|> 20000.0 nM | | | NPASS |
| Androgen receptor | Rattus norvegicus | P15207 | | 29512.09 nM | | | BindingDB |
| Beta-glucuronidase | Escherichia coli (strain K12) | P05804 | | 7.79e+4 nM | | | BindingDB |
| Beta-glucuronidase | Homo sapiens | P08236 | | 77900 nM|= 77900.0 nM | | | BindingDB, NPASS |
| Corticosteroid binding globulin | Homo sapiens | P08185 | | | | = 10000.0 nM | NPASS |
| Corticosteroid-binding globulin | Homo sapiens | P08185 | | | | 10000 nM | BindingDB |
| A-431 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| Glucose-6-phosphate 1-dehydrogenase | Homo sapiens | P11413 | | 24900 nM|11300 nM|12460 nM|= 11300.0 nM|= 24900.0 nM|= 12460.0 nM | | 8900 nM|6200 nM|= 8900.0 nM|= 6200.0 nM | BindingDB, NPASS |
| G-protein coupled bile acid receptor 1 | Homo sapiens | Q8TDU6 | 3330 nM|= 3330.0 nM | | | | BindingDB, NPASS |
| HT-29 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| Glucose-6-phosphate 1-dehydrogenase | Trypanosoma brucei | Q9GRG7 | | | | = 1700.0 nM|= 1100.0 nM | NPASS |
| Glucose-6-phosphate 1-dehydrogenase | Trypanosoma brucei | | | | | 1700 nM|1100 nM | BindingDB |
| HL-60 | Homo sapiens | | | > 20000.0 nM | | | NPASS |