| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Plasmodium falciparum | Plasmodium falciparum | | = 1080.0 nM|> 1065.0 nM | | | | NPASS |
| Metabotropic glutamate receptor 8 | Rattus norvegicus | P70579 | | | | 1200 nM | BindingDB |
| Metabotropic glutamate receptor 7 | Homo sapiens | Q14831 | < 200000.0 nM | | | >10000 nM | BindingDB, NPASS |
| Metabotropic glutamate receptor 6 | Rattus norvegicus | P35349 | 2700 nM|= 2700.0 nM | | | | BindingDB, NPASS |
| Metabotropic glutamate receptor 6 | Homo sapiens | O15303 | | | | 2700 nM | BindingDB |
| Metabotropic glutamate receptor 4 | Rattus norvegicus | P31423 | 4000 nM|= 4000.0 nM|< 100000.0 nM | | | 2300 nM | BindingDB, NPASS |
| Metabotropic glutamate receptor 7 | Rattus norvegicus | P35400 | 160000 nM|= 160000.0 nM | | | | BindingDB, NPASS |
| Glutamate carboxypeptidase II | Homo sapiens | Q04609 | | = 523000.0 nM | | | NPASS |
| Glutamate carboxypeptidase 2 [44-750] | Homo sapiens | Q04609 | | 523000 nM | | | BindingDB |
| Carbonic anhydrase VA | Homo sapiens | P35218 | | | | = 360000.0 nM | NPASS |
| Carbonic anhydrase IX | Homo sapiens | Q16790 | | | | = 920000.0 nM | NPASS |
| Carbonic anhydrase IV | Homo sapiens | P22748 | | | | = 4260000.0 nM | NPASS |
| Carbonic anhydrase II | Homo sapiens | P00918 | | | | = 420000.0 nM | NPASS |
| Metabotropic glutamate receptor 4 | Homo sapiens | Q14833 | 1000 nM|1300 nM|= 1000.0 nM|= 1300.0 nM | | | 2000 nM | BindingDB, NPASS |