
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| SK-BR-3 | Homo sapiens | = 0.03 nM | NPASS | ||||
| Reverse transcriptase | Human immunodeficiency virus 1 | >288000 nM | BindingDB | ||||
| OVCAR-3 | Homo sapiens | = 0.1 nM | NPASS | ||||
| KB | Homo sapiens | = 0.034 nM | NPASS | ||||
| Human immunodeficiency virus type 1 reverse transcriptase | Human immunodeficiency virus 1 | Q72547 | > 200.0 ug.mL-1 | NPASS | |||
| SW-620 | Homo sapiens | > 0.1 nM | NPASS | ||||
| HCT-15 | Homo sapiens | = 0.75 nM | NPASS | ||||
| A549 | Homo sapiens | = 0.16 nM|= 0.59 nM | NPASS | ||||
| A2780 | Homo sapiens | = 0.74 nM | NPASS | ||||
| A-431 | Homo sapiens | = 0.04 nM | NPASS | ||||
| A-375 | Homo sapiens | = 0.037 nM | NPASS | ||||
| HeLa | Homo sapiens | = 0.33 nM|= 1.1 nM | NPASS | ||||
| MCF7 | Homo sapiens | = 0.044 nM | NPASS |