| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| SF-268 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 51900.0 nM|= 99900.0 nM|> 100000.0 nM | | | NPASS |
| Proteasome subunit beta type-5 | Homo sapiens | P28074 | | 5210 nM | | | BindingDB |
| Proteasome Macropain subunit MB1 | Homo sapiens | P28074 | | = 5210.0 nM | | | NPASS |
| NCI-H460 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| A549 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| HT-1080 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Aromatase | Homo sapiens | P11511 | | 3800 nM | | | BindingDB |
| MCF7 | Homo sapiens | | | > 50000.0 nM | | | NPASS |