IMPPAT Phytochemical information: 
Isoxanthohumol

Isoxanthohumol
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
PC-3Homo sapiens= 71320.0 nMNPASS
Protein kinase C thetaHomo sapiensQ04759= 31600.0 nMNPASS
Protein kinase C alphaHomo sapiensP17252= 45300.0 nMNPASS
MCF7Homo sapiens= 26540.0 nM|= 15300.0 nM|= 4690.0 nMNPASS
NON-PROTEIN TARGET= 35420.0 nMNPASS
HT-29Homo sapiens= 88820.0 nMNPASS
Estrogen receptor alphaHomo sapiensP03372= 1400.0 nMNPASS
Beta-secretase 1Homo sapiensP56817= 27700.0 nMNPASS
3-phosphoinositide dependent protein kinase-1Homo sapiensO15530= 58700.0 nMNPASS
IshikawaHomo sapiens= 24900.0 nMNPASS