IMPPAT Phytochemical information: 
Hyperforin

Hyperforin
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
SMMC-7721Homo sapiens> 40000.0 nMNPASS
Pregnane X receptorHomo sapiensO75469= 27.0 nMNPASS
NON-PROTEIN TARGET= 2100.0 nMNPASS
MCF7Homo sapiens> 40000.0 nMNPASS
SW480Homo sapiens> 40000.0 nMNPASS
Dihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, mitochondrialHomo sapiensP10515= 578.0 nMNPASS
Cytochrome P450 3A4Homo sapiensP08684= 2300.0 nMNPASS
A549Homo sapiens> 40000.0 nMNPASS
HL-60Homo sapiens> 40000.0 nMNPASS
Serotonin transporterRattus norvegicusP31652= 1.1 ug.mL-1NPASS