| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Nuclear factor NF-kappa-B complex | Homo sapiens | Q04206 | | = 41000.0 nM | | | NPASS |
| Pancreatic triacylglycerol lipase | Sus scrofa | P00591 | | 50400 nM|= 50400.0 nM | | | BindingDB, NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 15848.93 nM|= 12589.25 nM|= 10000.0 nM | | | NPASS |
| Vero | Chlorocebus aethiops | | | = 125.0 ug.mL-1 | | | NPASS |
| Serine/threonine-protein kinase 33 | Homo sapiens | Q9BYT3 | 21410 nM | | | | BindingDB |
| Sodium/glucose cotransporter 1 | Homo sapiens | P13866 | | 12400 nM|= 12400.0 nM | | 86000 nM|= 86000.0 nM | BindingDB, NPASS |
| Solute carrier family 28 member 3 | Homo sapiens | Q9HAS3 | | | | 32280 nM|= 32280.0 nM | BindingDB, NPASS |
| Sodium/hydrogen exchanger 9B2 | Homo sapiens | Q86UD5 | | = 90000.0 nM | | | NPASS |
| Solute carrier family 2, facilitated glucose transporter member 1 | Homo sapiens | P11166 | | 21400 nM | | | BindingDB |
| NON-PROTEIN TARGET | | | | = 54000.0 nM | | | NPASS |
| Sortase B | Staphylococcus aureus | Q2FZE3 | | = 9.74 ug.mL-1 | | | NPASS |
| Transthyretin | Homo sapiens | P02766 | | | 8100 nM|= 8100.0 nM | | BindingDB, NPASS |
| Sodium/glucose cotransporter 2 | Homo sapiens | P31639 | | 18300 nM|= 18300.0 nM | | | BindingDB, NPASS |
| Monocarboxylate transporter 4 | Homo sapiens | O15427 | | 41000 nM|= 41000.0 nM | | | BindingDB, NPASS |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | P0DTD1 | | 335000 nM | | | BindingDB |
| Monocarboxylate transporter 1 | Rattus norvegicus | P53987 | | 28000 nM|= 28000.0 nM | | | BindingDB, NPASS |
| Alpha-chymotrypsin | Bos taurus | P00766 | | > 300000.0 nM | | | NPASS |
| Beta-lactamase | Enterobacter cloacae | P05364 | | 496000 nM|= 496000.0 nM | | | BindingDB, NPASS |
| Chymotrypsinogen A | Bos taurus | P00766 | | >300000 nM | | | BindingDB |
| Cytochrome P450 19A1 | Homo sapiens | P11511 | | = 2600.16 nM | | | NPASS |
| DNA topoisomerase 2-alpha | Homo sapiens | P11388 | | 167000 nM | | | BindingDB |
| DNA topoisomerase II alpha | Homo sapiens | P11388 | | = 46.1 ug.mL-1 | | | NPASS |
| Monocarboxylate transporter 2 | Rattus norvegicus | Q66HS9 | | 14000 nM|= 14000.0 nM | | | BindingDB, NPASS |
| Epidermal growth factor receptor erbB1 | Homo sapiens | P00533 | | = 25000000.0 nM | | | NPASS |
| Estrogen receptor alpha | Homo sapiens | P03372 | | = 300.0 nM | | | NPASS |
| Glucose transporter | Homo sapiens | P11166 | | = 21400.0 nM | | | NPASS |
| Glucose-6-phosphate translocase | Homo sapiens | O43826 | | = 340000.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | > 10000.0 nM|= 7000.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Epidermal growth factor receptor | Homo sapiens | P00533 | | 25000000 nM | | | BindingDB |