| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| cGMP-dependent 3',5'-cyclic phosphodiesterase | Rattus norvegicus | Q01062 | | 96000 nM | | | BindingDB |
| Phosphodiesterase 2A | Rattus norvegicus | Q01062 | | = 96000.0 nM | | | NPASS |
| Phosphodiesterase 1 | Rattus norvegicus | Q01066 | | > 1000000.0 nM | | | NPASS |
| No relevant target | | | | = 620000.0 nM | | | NPASS |
| P-glycoprotein 1 | Homo sapiens | P08183 | | = 23400.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 2042.0 nM | | | NPASS |
| Multidrug resistance-associated protein 1 | Homo sapiens | P33527 | | 26350 nM|= 26350.0 nM | | | BindingDB, NPASS |
| L929 | Mus musculus | | | > 100000.0 nM | | | NPASS |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens | Q9UNQ0 | | 1880 nM|822 nM | | | BindingDB |
| ATP-binding cassette sub-family G member 2 | Homo sapiens | Q9UNQ0 | | = 1880.0 nM|= 822.0 nM | | | NPASS |