
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| HL-60 | Homo sapiens | = 5500.0 nM | NPASS | ||||
| NACHT, LRR and PYD domains-containing protein 3 | Homo sapiens | Q96P20 | 5900 nM|= 5900.0 nM | BindingDB, NPASS | |||
| NACHT, LRR and PYD domains-containing protein 3 | Mus musculus | Q8R4B8 | 2300 nM|= 2300.0 nM | BindingDB, NPASS | |||
| NON-PROTEIN TARGET | = 6200.0 nM | NPASS | |||||
| Pyruvate kinase PKM | Homo sapiens | P14618 | 6.0 nM | BindingDB | |||
| Pyruvate kinase isozymes M1/M2 | Homo sapiens | P14618 | = 6.0 nM | NPASS |