| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| MCF7 | Homo sapiens | | | = 5.0 ug.mL-1|= 35000.0 nM|= 41800.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 44890.0 nM | | | NPASS |
| Mitochondrial import inner membrane translocase subunit TIM10 | Saccharomyces cerevisiae (strain ATCC 204508 / S288c) | P87108 | | 48800 nM | | | BindingDB |
| Mitochondrial import inner membrane translocase subunit TIM10 | Saccharomyces cerevisiae S288c | P87108 | | = 48800.0 nM | | | NPASS |
| NAD-dependent deacetylase sirtuin 3 | Homo sapiens | Q9NTG7 | = 170.0 nM | | = 290.0 nM|= 2990.0 nM|= 1010.0 nM|= 970.0 nM|= 40000.0 nM | | NPASS |
| NAD-dependent protein deacetylase sirtuin-3, mitochondrial | Homo sapiens | Q9NTG7 | 170 nM | | | | BindingDB |
| NCI-H1650 | Homo sapiens | | | = 37350.0 nM | | | NPASS |
| NCI-H1975 | Homo sapiens | | | = 30200.0 nM | | | NPASS |
| NCI-H358 | Homo sapiens | | | = 31570.0 nM | | | NPASS |
| NCI-H441 | Homo sapiens | | | = 33320.0 nM | | | NPASS |
| NCI-H460 | Homo sapiens | | | = 38460.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 36100.0 nM|= 65400.0 nM | | | NPASS |
| Neuraminidase | InflueA virus | B4URF0 | | = 1390.0 nM|= 30100.0 nM | | | NPASS |
| Neuraminidase | InflueA virus (A/WSN/1933(H1N1)) | P03470 | | 30100 nM|1390 nM | | | BindingDB |
| Vero | Chlorocebus aethiops | | | = 22500.0 nM | | | NPASS |
| PANC-1 | Homo sapiens | | | = 31240.0 nM | | | NPASS |
| PC-9 | | | | = 36720.0 nM | | | NPASS |
| Platelet glycoprotein VI | Homo sapiens | Q9HCN6 | | | 289000 nM | | BindingDB |
| Platelet glycoprotein VI (GPVI) | Homo sapiens | Q9HCN6 | | | = 289000.0 nM | | NPASS |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens | P09917 | | 4200 nM | | | BindingDB |
| Prostaglandin G/H synthase 1 | Ovis aries | P05979 | | 1800 nM | | | BindingDB |
| Prostaglandin G/H synthase 2 | Ovis aries | P79208 | | 2100 nM | | | BindingDB |
| RKO | Homo sapiens | | | = 11420.0 nM | | | NPASS |
| Retinoic acid receptor RXR-alpha | Homo sapiens | P19793 | 11800 nM | | | | BindingDB |
| Retinoid X receptor alpha | Homo sapiens | P19793 | = 11800.0 nM | | | | NPASS |
| SARS coronavirus | SARS coronavirus | | = 6500.0 nM | | | | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 50000.0 nM | | | NPASS |
| SW480 | Homo sapiens | | | = 15140.0 nM | | | NPASS |
| Spike glycoprotein | Severe acute respiratory syndrome coronavirus 2 | P0DTC2 | | | 25010 nM|= 25010.0 nM | | BindingDB, NPASS |
| UACC-903 | Homo sapiens | | | = 7450.0 nM|= 5100.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 29030.0 nM | | | NPASS |
| L02 | Homo sapiens | | | = 25490.0 nM | | | NPASS |
| Gamma-aminobutyric acid receptor subunit alpha-1/ beta-1 | Homo sapiens | | = 57000.0 nM | | | | NPASS |
| I10 | Mus musculus | | | = 31110.0 nM | | | NPASS |
| A2780 | Homo sapiens | | | = 30500.0 nM|= 41200.0 nM|= 31580.0 nM | | | NPASS |
| A549 | Homo sapiens | | | > 5.0 ug.mL-1|= 35000.0 nM|= 12510.0 nM|= 7750.0 nM|= 35310.0 nM|= 35410.0 nM|= 34100.0 nM|= 29700.0 nM|= 38040.0 nM | | | NPASS |
| Angiotensin-converting enzyme 2 | Homo sapiens | Q9BYF1 | | | 16980 nM|= 16980.0 nM | | BindingDB, NPASS |
| Arachidonate 5-lipoxygenase | Homo sapiens | P09917 | | = 4200.0 nM | | | NPASS |
| K562 | Homo sapiens | | | > 5.0 ug.mL-1|= 21100.0 nM|= 23910.0 nM|= 22100.0 nM|= 28400.0 nM | | | NPASS |
| CCRF-CEM | Homo sapiens | | | = 10900.0 nM | | | NPASS |
| CNE2Z | Homo sapiens | | | = 31270.0 nM | | | NPASS |
| Cannabinoid CB1 receptor | Homo sapiens | P21554 | > 10000.0 nM | | | = 6460.0 nM|= 6.46 nM | NPASS |
| Cannabinoid CB2 receptor | Homo sapiens | P34972 | | | | = 5610.0 nM|= 5.61 nM | NPASS |
| Cannabinoid receptor 1 | Homo sapiens | P21554 | >10000 nM | | | 6.5 nM|6460 nM | BindingDB |
| Cannabinoid receptor 2 | Homo sapiens | P34972 | | | | 1763 nM|5.6 nM|5610 nM | BindingDB |
| Cyclooxygenase-1 | Ovis aries | P05979 | | = 1800.0 nM | | | NPASS |
| Cyclooxygenase-2 | Ovis aries | P79208 | | = 2100.0 nM | | | NPASS |
| GABA-A receptor alpha-1/beta-3 | Homo sapiens | | = 59600.0 nM | | | | NPASS |
| GABA-A receptor; GABA-A site (alpha1/beta2 interface) | Homo sapiens | P47870 | = 39300.0 nM | | | | NPASS |
| BV-2 | Mus musculus | | | = 17000.0 nM | | | NPASS |
| Gamma-aminobutyric acid receptor subunit alpha-1/beta-2 | Homo sapiens | P14867|P47870 | 39300 nM | | | | BindingDB |
| GABA-A receptor; alpha-1/beta-2/gamma-2 | Homo sapiens | P18507 | = 76200.0 nM | | | | NPASS |
| Human immunodeficiency virus 1 | Human immunodeficiency virus 1 | | = 3300.0 nM | | | | NPASS |
| Hepatitis C virus | Hepatitis C virus | | = 9400.0 nM | | | | NPASS |
| HeLa | Homo sapiens | | | > 5.0 ug.mL-1|= 62000.0 nM | | | NPASS |
| HUVEC | Homo sapiens | | | = 52600.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | = 23050.0 nM|= 13240.0 nM|= 6.1 ug.mL-1|= 25000.0 nM|= 31580.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 16500.0 nM|= 34300.0 nM|= 33880.0 nM|= 32900.0 nM|= 23850.0 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | = 19050.0 nM|= 47650.0 nM | | | NPASS |
| HCC827 | Homo sapiens | | | = 33880.0 nM | | | NPASS |
| Gamma-aminobutyric acid receptor subunit alpha-5/beta-2 | Homo sapiens | | = 23400.0 nM | | | | NPASS |
| Gamma-aminobutyric acid receptor subunit alpha-3/ beta-2 | Homo sapiens | | = 52400.0 nM | | | | NPASS |
| Gamma-aminobutyric acid receptor subunit alpha-2/beta-2 | Homo sapiens | | = 46400.0 nM | | | | NPASS |
| Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2 | Homo sapiens | P14867|P18507|P47870 | 76200 nM | | | | BindingDB |
| HEK293 | Homo sapiens | | | = 9.3 ug.mL-1|= 40000.0 nM | | | NPASS |