| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Muscarinic acetylcholine receptor M5 | Homo sapiens | P08912 | 55.0 nM | 8000 nM | | | BindingDB |
| Muscarinic acetylcholine receptor M4 | Homo sapiens | P08173 | 33 nM|14 nM|9.0 nM | 5000 nM | | 1.5 nM|160 nM | BindingDB |
| Muscarinic acetylcholine receptor M3 | Rattus norvegicus | P08483 | | | | 398 nM | BindingDB |
| Muscarinic acetylcholine receptor M3 | Homo sapiens | P20309 | 210 nM | 17000 nM | | | BindingDB |
| Muscarinic acetylcholine receptor M2 | Rattus norvegicus | P10980 | | 2000 nM|860 nM|858 nM|84 nM | | 480 nM|500 nM|290 nM|84.0 nM|0.500000 nM|60 nM|160 nM|199 nM | BindingDB |
| Muscarinic acetylcholine receptor M2 | Mus musculus | Q9ERZ4 | | | | 1.7 nM|1500 nM | BindingDB |
| Muscarinic acetylcholine receptor M2 | Homo sapiens | P08172 | 19 nM | 400 nM | | 235 nM|660 nM|148 nM|10000 nM|324 nM|851 nM|1023 nM|1778 nM | BindingDB |
| Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 | Homo sapiens | P08172|P08173|P08912|P11229|P20309 | | | 930 nM | | BindingDB |
| Muscarinic acetylcholine receptor M1 | Rattus norvegicus | P08482 | | 113 nM|360 nM|100 nM | | 490 nM|196 nM|120 nM|630 nM | BindingDB |
| Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 | Rattus norvegicus | P08482|P08483|P08485|P08911|P10980 | | 660 nM|2700 nM|2 nM|407 nM|1.5 nM|3300 nM|17 nM|2.8 nM | | 60 nM|0.500000 nM|4.0 nM|140 nM|830 nM|193 nM|230 nM | BindingDB |
| Muscarinic acetylcholine receptor M1 | Homo sapiens | P11229 | 390 nM|1.6 nM | 2.3 nM|27100 nM|9000 nM|364 nM | | 1.1 nM|17 nM | BindingDB |
| Muscarinic acetylcholine receptor DM1 | Drosophila melanogaster | P16395 | | | | 21500 nM|19400 nM | BindingDB |
| Muscarinic acetylcholine receptor | Cavia porcellus | | 50 nM | | 1200 nM | | BindingDB |
| Mucolipin-3 | Homo sapiens | Q8TDD5 | >29900 nM | | | | BindingDB |
| Ion channel NompC | Danio rerio | | 29900 nM | | | | BindingDB |
| Beta-arrestin-1 | Oryctolagus cuniculus | Q95223 | | | | 214 nM|1564 nM | BindingDB |
| Acetylcholinesterase | Mus musculus | P21836 | | | | 1500 nM|1.7 nM | BindingDB |
| 5-hydroxytryptamine receptor 7 | Rattus norvegicus | P32305 | | | | >10000 nM | BindingDB |
| Muscarinic acetylcholine receptor M1 | Mus musculus | P12657 | 270 nM | | | | BindingDB |