IMPPAT Phytochemical information: 
Camptothecin

Camptothecin
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
NCI-H1993Homo sapiens= 9621.56 nMNPASS
NCI-H2009Homo sapiens= 68.13 nMNPASS
NCI-H2029Homo sapiens= 491.21 nMNPASS
NCI-H2030Homo sapiens= 48.53 nMNPASS
NCI-H2052Homo sapiens= 28.34 nMNPASS
NCI-H2087Homo sapiens= 5.074 nMNPASS
NCI-H209Homo sapiens= 0.04843 nMNPASS
NCI-H2122Homo sapiens= 12.98 nMNPASS
NCI-H2126Homo sapiens= 178.42 nMNPASS
NCI-H2170Homo sapiens= 13.71 nMNPASS
NCI-H2228Homo sapiens= 49.0 nMNPASS
NCI-H2291Homo sapiens= 975.25 nMNPASS
NCI-H23Homo sapiens= 40.69 nM|= 70.0 nMNPASS
NCI-H2342Homo sapiens= 618.33 nMNPASS
NCI-H2347Homo sapiens= 185.61 nMNPASS
NCI-H2405Homo sapiens= 58.48 nMNPASS
NCI-H2452Homo sapiens= 90.89 nMNPASS
NCI-H28Homo sapiens= 38.68 nMNPASS
NCI-H292= 2.24 nMNPASS
NCI-H226Homo sapiens= 22.49 nMNPASS
NCI-H1975Homo sapiens= 334.48 nM|= 1200.0 nMNPASS
NCI-H1623Homo sapiens= 0.7479 nMNPASS
NCI-H1793Homo sapiens= 27.23 nMNPASS
NCI-H128Homo sapiens= 18.0 nMNPASS
NCI-H1299Homo sapiens= 9.425 nM|= 3140.0 nM|= 800.0 nMNPASS
NCI-H1304Homo sapiens= 59.28 nMNPASS
NCI-H1355Homo sapiens= 66.1 nMNPASS
NCI-H1395Homo sapiens= 110.1 nMNPASS
NCI-H1437Homo sapiens= 34.93 nMNPASS
NCI-H1563Homo sapiens= 150.37 nMNPASS
NCI-H1573Homo sapiens= 173.4 nMNPASS
NCI-H1581Homo sapiens= 33.5 nMNPASS
NCI-H358Homo sapiens= 105.42 nMNPASS
NCI-H1648Homo sapiens= 38.07 nMNPASS
NCI-H1650Homo sapiens= 149.39 nMNPASS
NCI-H1651Homo sapiens= 14.95 nMNPASS
NCI-H1666Homo sapiens= 18.71 nMNPASS
NCI-H1693Homo sapiens= 26.69 nMNPASS
NCI-H1703Homo sapiens= 6.515 nMNPASS
NCI-H1755Homo sapiens= 208.78 nMNPASS
NCI-H1770Homo sapiens= 157.32 nMNPASS
NCI-H1792Homo sapiens= 40.12 nMNPASS
NCI-H1838Homo sapiens= 253.14 nMNPASS
NCI-H441Homo sapiens= 28.46 nMNPASS
NCI-H720Homo sapiens= 44.69 nMNPASS
NCI-H460Homo sapiens= 6.9 nM= 330.0 nM|= 180.0 nM|= 6.2 nM|> 25000.0 nM|> 1000.0 nM|= 13.0 nM|< 40.0 nM|= 30.0 nM|= 5.0 nM|= 2.0 nM|= 3.0 nM|= 24.12 nM|= 190.0 nM|= 110.0 nM|= 5370.0 nM|= 120.0 nM|= 790.0 nMNPASS
NOS-1Homo sapiens= 91.86 nMNPASS
NTERA-2-cl-D1Homo sapiens= 0.2738 nMNPASS
NUGC-3Homo sapiens= 3.136 nMNPASS
NYHomo sapiens= 4356.62 nMNPASS
OAW-28Homo sapiens= 7.263 nMNPASS
OAW-42Homo sapiens= 8.99 nMNPASS
OC-314Homo sapiens= 2.506 nMNPASS
OCI-AML2Homo sapiens= 0.8868 nMNPASS
OCUB-MHomo sapiens= 38.13 nMNPASS
OE19Homo sapiens= 3273.33 nMNPASS
OE33Homo sapiens= 25.55 nMNPASS
OMC-1Homo sapiens= 78.21 nMNPASS
ONS-76Homo sapiens= 2.406 nMNPASS
OS-RC-2Homo sapiens= 9.968 nMNPASS
OVCAR-3Homo sapiens= 956.65 nMNPASS
OVCAR-4Homo sapiens= 188.55 nMNPASS
OVCAR-5Homo sapiens= 43.33 nMNPASS
OVCAR-8Homo sapiens= 7.272 nMNPASS
P12-IchikawaHomo sapiens= 0.1016 nMNPASS
NON-PROTEIN TARGET= 330.0 nM|= 8.5 nM|= 61000.0 nM|= 33.0 nM|= 5.6 nM|> 10000.0 nM|= 5385.0 nM|= 500.0 nM|= 24.0 nM|= 0.004 nM|> 10.0 nM|= 5.0 nM|= 15.0 nM|= 25.0 nM|= 26.0 nM|= 0.08 ug.mL-1|= 4.0 nM|= 28.7 nM|= 3280.0 nM|= 6.0 nM|= 1700.0 nM|= 60.0 nM|= 30.0 nM|> 25000.0 nM|= 52.0 nM|= 57.0 nM|= 260.0 nM|= 15200.0 nM|< 100.0 nM|= 10.0 nM|< 1000.0 nM|= 6.8 nM|= 423.0 nM|= 37.1 nM|< 10.0 nM|= 300.0 nM|= 2780.0 nM|= 10070.0 nM|= 1980.0 nM|= 474.0 nM|= 786.0 nM|= 131.0 nM|= 120.0 nM|= 3600.0 nM|= 6300.0 nM|= 40.0 nM|= 0.15 nM|= 70.0 nM|= 220.0 nM|= 710.0 nM|= 960.0 nM|< 3.0 nM|= 140.0 nM|= 100.0 nM|= 190.0 nM|<= 100.0 nM|= 1290.0 nM|= 20.0 nM|= 2820.0 nM|= 7000.0 nM|= 7100.0 nM|= 5.5 nM|= 3.0 nM|= 35.0 nM|= 9520.0 nM|= 11360.0 nM|= 17650.0 nM|= 59130.0 nM|= 29810.0 nM|> 100000.0 nM|= 1410.0 nM|= 1270.0 nM|= 460.0 nM|= 1520.0 nM|= 80.0 nM|= 1.4 nM|= 130.0 nM|= 600.0 nM|= 1120.0 nM|= 310.0 nM|= 13700.0 nM|= 110.0 nM|= 400.0 nM|= 830.0 nM|= 1060.0 nM|= 590.0 nM|= 380.0 nM|= 350.0 nM|= 4540.0 nM|= 890.0 nM|= 1240.0 nM|= 6700.0 nM|= 3040.0 nM|= 1840.0 nM|= 5930.0 nMNPASS
NCI-H446Homo sapiens= 56.63 nM|> 200000.0 nMNPASS
NOMO-1Homo sapiens= 1.557 nMNPASS
NKM-1Homo sapiens= 0.441 nMNPASS
NCI-H510AHomo sapiens= 1.699 nMNPASS
NCI-H520Homo sapiens= 25.01 nMNPASS
NCI-H520= 162.01 nMNPASS
NCI-H526Homo sapiens= 1.028 nMNPASS
NCI-H596= 2968.73 nMNPASS
NCI-H630Homo sapiens= 282.32 nMNPASS
NCI-H650Homo sapiens= 54.96 nMNPASS
NCI-H661Homo sapiens= 13.55 nMNPASS
NCI-H69Homo sapiens= 1.0 nM|= 311.44 nMNPASS
NCI-H1155Homo sapiens= 1.188 nMNPASS
NCI-H727Homo sapiens= 1009.34 nMNPASS
NCI-H747Homo sapiens= 296.49 nMNPASS
NCI-H810Homo sapiens= 50.3 nMNPASS
NCI-H82Homo sapiens= 588.29 nMNPASS
NCI-H928= 7.8 nMNPASS
NCI-N87Homo sapiens= 8.743 nM|= 2320.0 nMNPASS
NEC8Homo sapiens= 3.108 nMNPASS
NH-12Homo sapiens= 3.793 nMNPASS
NHDFHomo sapiens= 5380.0 nMNPASS
NMC-G1Homo sapiens= 19.82 nMNPASS
NCI-H1092Homo sapiens= 43.18 nMNPASS
MC-IXCHomo sapiens= 0.513 nMNPASS
NBsusSRHomo sapiens= 0.1936 nMNPASS
MCF-10AHomo sapiens= 2190.0 nM|= 2580.0 nMNPASS
MCF-12AHomo sapiens< 10.0 nMNPASS
MCF10Homo sapiens= 24770.0 nMNPASS
MCF7Homo sapiens= 72.0 nM= 3.1 nM|= 0.02 ug.mL-1|= 320.0 nM|= 40.0 nM|= 10000.0 nM|= 200.0 nM|= 1100.0 nM|= 3.0 nM|= 10.0 nM|= 7420.0 nM|= 60.0 nM|= 1220.0 nM|= 20.0 nM|= 14200.0 nM|= 2430.0 nM|= 650.0 nM|= 70.0 nM|= 11120.0 nM|= 1.6 nM|= 56.0 nM|= 2600.0 nM|= 1800.0 nM|= 3910.0 nM|< 100.0 nM|= 80.0 nM|< 1000.0 nM|< 10.0 nM|= 6.427 nM|= 26.0 nM|= 3.3 nM|< 0.024 ug.mL-1|= 65.1 nM|= 0.5 nM|= 0.6 nM|<= 100.0 nM|= 6000.0 nM|< 1.8 nM|= 71300.0 nM|= 30.0 nM|= 87.5 nM|= 28660.0 nM|= 73.0 nM|= 13620.0 nM|= 340.0 nM|= 160.0 nM|= 420.0 nM|= 680.0 nM|= 84.0 nM|= 1670.0 nM|= 2500.0 nM|= 18600.0 nM|= 560.0 nM|= 2800.0 nM|= 21.0 nM|= 350.0 nMNPASS
MDA-MB-157Homo sapiens= 20.0 nM|= 7.569 nMNPASS
MDA-MB-175-VIIHomo sapiens= 83.02 nMNPASS
MDA-MB-231Homo sapiens= 291.0 nM|= 4160.0 nM|= 1100.0 nM|= 920.0 nM|= 680.0 nM|= 300.0 nM|= 4200.0 nM|= 330.0 nM|= 970.0 nM|= 2700.0 nM|< 10.0 nM|= 229.98 nM|= 162.0 nM|= 342.0 nM|= 2110.0 nM|= 5770.0 nM|= 307.0 nM|= 540.0 nM|= 16440.0 nM|= 0.32 nM|= 28.4 nM|= 23980.0 nM|= 8830.0 nM|= 264.0 nM|> 6400.0 nM|= 420.0 nM|= 1060.0 nM|= 490.0 nM|= 241.0 nM|> 100000.0 nM|= 170.0 nMNPASS
MDA-MB-361Homo sapiens= 170.0 nM|= 34.43 nMNPASS
MDA-MB-415Homo sapiens= 134.42 nMNPASS
MDA-MB-435Homo sapiens= 15.0 nM|= 375.0 nM|= 710.0 nM|= 43.6 nM|< 1.0 nM|= 1000.0 nM|= 2700.0 nM|= 310.0 nMNPASS
MDA-MB-436Homo sapiens= 31860.0 nMNPASS
MDA-MB-453Homo sapiens< 10.0 nM|= 6.965 nMNPASS
MDA-MB-468Homo sapiens= 14760.0 nM|= 1710.0 nMNPASS
ME-180Homo sapiens= 2.692 nMNPASS
MEFMus musculus= 5.87 ug.mL-1NPASS
MEG-01Homo sapiens= 39.51 nMNPASS
MEL-HOHomo sapiens= 7.628 nMNPASS
MEL-JUSOHomo sapiens= 35.62 nMNPASS
MFE-280Homo sapiens= 21.56 nMNPASS
MC116Homo sapiens= 15.86 nMNPASS
MFE-296Homo sapiens< 1000.0 nMNPASS
P30-OHKHomo sapiens= 2.792 nMNPASS
M059JHomo sapiens= 4.095 nM|= 5500.0 nMNPASS
LNCaP-Clone-FGCHomo sapiens= 31.03 nMNPASS
LOX IMVIHomo sapiens= 48.0 nM|= 3.72 nMNPASS
LS-1034Homo sapiens= 9492.4 nMNPASS
LS-123Homo sapiens= 7325.59 nMNPASS
LS-411NHomo sapiens= 58.08 nMNPASS
LS-513Homo sapiens= 19.37 nMNPASS
LU-134-AHomo sapiens= 0.5865 nMNPASS
LU-135Homo sapiens= 28.16 nMNPASS
LU-139Homo sapiens= 16.44 nMNPASS
LU-99AHomo sapiens= 3.854 nMNPASS
LX-1Homo sapiens= 120.0 nMNPASS
LXF-289 cell line= 7.054 nMNPASS
Leishmania donovaniLeishmadonovani= 7840.0 nM|= 3794.0 nM|= 12820.0 nM|= 6582.0 nMNPASS
Leishmania infantumLeishmaitum= 34400.0 nM|= 1120.0 nMNPASS
Lewis lung carcinoma cell line= 33.0 nMNPASS
LoVoHomo sapiens= 3100.0 nM|= 14.93 nM|= 0.32 nM|= 1540.0 nMNPASS
Lu-65Homo sapiens= 276.33 nMNPASS
Lu-99 cell line= 0.001 ug.mL-1NPASS
Lu1Homo sapiens= 28.7 nMNPASS
M14Homo sapiens= 9.948 nMNPASS
NCI-H1048Homo sapiens= 0.5292 nMNPASS
MFH-inoHomo sapiens= 27.08 nMNPASS
MG-63Homo sapiens= 7.654 nMNPASS
MX1Homo sapiens= 1700.0 nMNPASS
MZ1-PCHomo sapiens= 20.33 nMNPASS
MZ2-MELHomo sapiens= 14.11 nMNPASS
MZ7-melHomo sapiens= 8.612 nMNPASS
MacrophageMus musculus= 18320.0 nMNPASS
MeWoHomo sapiens= 46.97 nMNPASS
Melanoma-associated antigen E1Q9HCI5>55182 nMBindingDB
MoHomo sapiens= 111.97 nMNPASS
Multidrug resistance-associated protein 4Homo sapiensO15439= 7400.0 nMNPASS
NB-4Homo sapiens= 2010.0 nMNPASS
NB10Homo sapiens= 0.6143 nMNPASS
NB12Homo sapiens= 44.02 nMNPASS
NB13Homo sapiens= 28.8 nMNPASS
NB14Homo sapiens= 0.9071 nMNPASS
NB17Homo sapiens= 2.175 nMNPASS
NB5Homo sapiens= 1.925 nMNPASS
NB6Homo sapiens= 182.71 nMNPASS
NB69Homo sapiens= 0.5694 nMNPASS
NB7Homo sapiens= 16.8 nMNPASS
MV4-11Homo sapiens= 0.7058 nMNPASS
MFM-223Homo sapiens= 5270.72 nMNPASS
MT4Homo sapiens= 4.0 nMNPASS
MS-1Homo sapiens= 2.774 nMNPASS
MGC-803Homo sapiens= 9450.0 nM|= 2960.0 nM|= 4270.0 nM|> 150000.0 nM|= 17760.0 nMNPASS
MHCC97HHomo sapiens= 0.32 nMNPASS
MHH-ES-1Homo sapiens= 0.1293 nMNPASS
MHH-NB-11Homo sapiens= 0.8418 nMNPASS
MHH-PREB-1Homo sapiens= 2.733 nMNPASS
MIA PaCa-2Homo sapiens= 400.0 nM|= 2.759 nM|= 190.0 nM|= 180.0 nMNPASS
MKN-1Homo sapiens= 37.91 nMNPASS
MKN-28Homo sapiens= 51.21 nMNPASS
MKN-45Homo sapiens= 17.0 nM|= 27.5 nMNPASS
MKN-7Homo sapiens= 144.23 nMNPASS
ML-2Homo sapiens= 2.165 nMNPASS
MLMAHomo sapiens= 8.145 nMNPASS
MMAC-SFHomo sapiens= 38.4 nMNPASS
MN-60Homo sapiens= 5.083 nMNPASS
MOLT-13Homo sapiens= 1.787 nMNPASS
MOLT-16Homo sapiens= 0.7318 nMNPASS
MOLT-4Homo sapiens= 1.616 nM|= 0.04 nMNPASS
MPP-89Homo sapiens= 27.24 nMNPASS
MRC5Homo sapiens= 890.0 nM|= 1700.0 nM|= 800.0 nM|= 1.7 10^-5 uM|= 9020.0 nMNPASS
MSTO-211HHomo sapiens= 8.238 nMNPASS
P388Mus musculus= 32.0 nM|= 0.005 ug.mL-1|= 0.00474 ug.mL-1|= 7.0 nM|= 13.0 nM|= 10.0 nM|= 32.1 nM|= 0.004 nM|= 9.0 nM|> 10000.0 nM|= 4.0 nM|= 14.0 nMNPASS
SK-MEL-30Homo sapiens= 2281.97 nMNPASS
PA-1Homo sapiens= 0.981 nMNPASS
SiHaHomo sapiens= 86.88 nMNPASS
Somatostatin receptorHomo sapiensP32745= 2.21 nMNPASS
Somatostatin receptor type 1/2/3/4/5Homo sapiensP30872|P30874|P31391|P32745|P353462.2 nMBindingDB
T-24Homo sapiens= 88.0 nM|= 6.0 nM|= 1.614 nM|= 6800.0 nM|= 3090.0 nMNPASS
T47DHomo sapiens= 207.0 nM|= 9170.0 nM|< 1000.0 nM|< 10.0 nM|= 1530.0 nM|= 13.52 nM|= 70.0 nM|= 300.0 nM|= 280.0 nM|= 750.0 nM|= 1840.0 nM|= 310.0 nM|= 80.0 nM|= 1620.0 nM|= 11170.0 nM|= 4100.0 nM|= 2100.0 nM|= 2310.0 nM|= 490.0 nM|= 250.0 nM|= 3670.0 nM|= 90.0 nMNPASS
T84Homo sapiens= 4602.33 nMNPASS
T98GHomo sapiens= 27.15 nMNPASS
TCC-SUPHomo sapiens= 39.04 nMNPASS
TE-1Homo sapiens= 35.11 nMNPASS
TE-10Homo sapiens= 147.61 nMNPASS
TE-11Homo sapiens= 16.33 nMNPASS
TE-12Homo sapiens= 265.25 nMNPASS
TE-5Homo sapiens= 7.38 nMNPASS
TE-6Homo sapiens= 178.5 nMNPASS
TE-8Homo sapiens= 4.17 nMNPASS
TE-9Homo sapiens= 23.65 nMNPASS
TERT-RPE1Homo sapiens> 40000.0 nM|= 27200.0 nMNPASS
TGBC11TKBHomo sapiens= 12.24 nMNPASS
TGBC1TKBHomo sapiens= 109.97 nMNPASS
Serotonin 2b (5-HT2b) receptorHomo sapiensP41595= 970.0 nM= 617.0 nMNPASS
TGBC24TKBHomo sapiens= 53.71 nMNPASS
Serine/threonine-protein kinase Chk1Homo sapiensO147572.1 nM|= 2.1 nMBindingDB, NPASS
SW982Homo sapiens= 4.062 nMNPASS
SW-620Homo sapiens= 1.2 nM|= 0.15 nM= 4.082 nMNPASS
SW1088Homo sapiens= 27.77 nMNPASS
SW13Homo sapiens= 2.993 nMNPASS
SW1417Homo sapiens= 52.7 nMNPASS
SW1463Homo sapiens= 51.69 nMNPASS
SW1573Homo sapiens= 2.348 nMNPASS
SW1710Homo sapiens= 33.57 nMNPASS
SW1783Homo sapiens= 24.57 nMNPASS
SW1990Homo sapiens= 37.88 nM|= 200.0 nMNPASS
SW48Homo sapiens= 3.017 nMNPASS
SW480Homo sapiens= 0.01 ug.mL-1|= 290.0 nM|= 210.0 nMNPASS
SW626Homo sapiens= 28.7 nM|= 76.9 nMNPASS
SW684Homo sapiens= 711.49 nMNPASS
SW756Homo sapiens= 4.211 nMNPASS
SW780Homo sapiens= 25.78 nMNPASS
SW837Homo sapiens= 48.92 nMNPASS
SW872Homo sapiens= 24.16 nMNPASS
SW900Homo sapiens= 31.84 nMNPASS
SW948Homo sapiens= 160.0 nM|= 260.2 nMNPASS
Saccharomyces cerevisiaeSaccharomyces cerevisiae> 200000.0 nM|= 0.16 ug.mL-1|= 0.014 ug.mL-1|> 100.0 ug.mL-1|= 0.18 ug.mL-1|= 0.06 ug.mL-1NPASS
SW 962Homo sapiens= 20.51 nMNPASS
THP-1Homo sapiens= 160.0 nM= 600.0 nM|= 71.0 nM|= 1890.0 nMNPASS
TK-10Homo sapiens= 55.79 nMNPASS
UACC-893Homo sapiens= 383.65 nMNPASS
UMC-11Homo sapiens= 2511.11 nMNPASS
UMUC3Homo sapiens= 3.093 nMNPASS
UO-31Homo sapiens= 34.07 nMNPASS
VA-ES-BJHomo sapiens= 3.469 nMNPASS
VM-CUB-1Homo sapiens= 2.21 nMNPASS
VMRC-RCZHomo sapiens= 47.35 nMNPASS
VeroChlorocebus aethiops= 0.054 ug.mL-1|= 0.02 ug.mL-1|= 0.6 ug.mL-1|= 58.0 ug.mL-1NPASS
WI-38Homo sapiens= 0.4 ug.mL-1|= 0.03 ug.mL-1|= 30.0 nM|= 8370.0 nMNPASS
WIL2-NSHomo sapiens= 5.0 nMNPASS
WM-115Homo sapiens= 102.32 nMNPASS
WiDrHomo sapiens= 17.0 nM|= 0.07 ug.mL-1NPASS
YAPCHomo sapiens= 29.6 nMNPASS
YH-13Homo sapiens= 11.65 nMNPASS
YKG-1Homo sapiens= 5.453 nMNPASS
ZR-75-1Homo sapiens< 10.0 nMNPASS
ZR-75-30Homo sapiens= 261.0 nM|= 240.0 nMNPASS
no-10Homo sapiens= 174.04 nMNPASS
no-11Homo sapiens= 113.08 nMNPASS
UACC-62Homo sapiens= 31.03 nMNPASS
TI-73Homo sapiens= 14.55 nMNPASS
UACC-257Homo sapiens= 115.96 nMNPASS
U-937Homo sapiens= 680.0 nM|= 32.0 nM|= 15.0 nM|= 300.0 nM|= 1980.0 nM|= 18240.0 nM|= 1810.0 nMNPASS
TYK-nuHomo sapiens= 4.94 nMNPASS
Telomerase reverse transcriptaseHomo sapiensO14746>300000 nM|> 300000.0 nMBindingDB, NPASS
Topoisomerase I subunit BLeishmamajor670 nMBindingDB
Type II restriction enzyme BamHIBacillus amyloliquefaciensP23940>300000 nMBindingDB
Type II restriction enzyme EcoRIEscherichia coliP00642>300000 nMBindingDB
Type II restriction enzyme HindIIIHaemophilus influe (strain ATCC 51907 / DSM 11121 / KW20 / Rd)P43870>300000 nMBindingDB
Type II restriction enzyme PstIProvidencia stuartiiP00640>300000 nMBindingDB
Type II restriction enzyme ScaIStreptomyces caespitosusO52691>300000 nMBindingDB
Type-2 restriction enzyme BamHIBacillus amyloliquefaciensP23940> 300000.0 nMNPASS
Type-2 restriction enzyme EcoRIEscherichia coliP00642> 300000.0 nMNPASS
Type-2 restriction enzyme HindIIIHaemophilus influe (strain ATCC 51907 / DSM 11121 / KW20 / Rd)P43870> 300000.0 nMNPASS
Type-2 restriction enzyme PstIProvidencia stuartiiP00640> 300000.0 nMNPASS
Type-2 restriction enzyme ScaIStreptomyces caespitosusO52691> 300000.0 nMNPASS
Tyrosyl-DNA phosphodiesterase 1Homo sapiensQ9NUW8>111000 nM|> 111000.0 nM|= 0.0 nMBindingDB, NPASS
Tyrosyl-DNA phosphodiesterase 2Homo sapiensO95551>111000 nM|> 111000.0 nM|= 0.0 nMBindingDB, NPASS
U-118-MGHomo sapiens= 19.0 nMNPASS
U-251Homo sapiens= 1.869 nMNPASS
U-266Homo sapiens= 69.51 nMNPASS
U-87 MGHomo sapiens= 6.632 nM|< 1850.0 nMNPASS
U2OSHomo sapiens= 13.54 nMNPASS
P388CPT5Mus musculus= 2800.0 nMNPASS
SW 954Homo sapiens= 20.35 nMNPASS
SU-DHL-2Homo sapiens= 940.0 nMNPASS
RPMI 8402Homo sapiens= 5.0 nM|= 6.0 nM|> 10000.0 nMNPASS
RPMI-2650Homo sapiens= 2.217 nMNPASS
RPMI-7951Homo sapiens= 4.753 nM|= 220.0 nMNPASS
RPMI-8226Homo sapiens= 6.0 nM|= 29.49 nM|= 2.05 ug.mL-1NPASS
RPMI-8866Homo sapiens= 1.725 nMNPASS
RS4-11Homo sapiens= 0.9022 nMNPASS
RT-112Homo sapiens= 14.88 nMNPASS
RVH-421Homo sapiens= 71.47 nMNPASS
RXF 393Homo sapiens= 4.662 nMNPASS
RajiHomo sapiens= 1000.0 nM|= 3270.0 nMNPASS
Ramos-2G6-4C10Homo sapiens= 10.51 nMNPASS
RencaMus musculus= 304.0 nMNPASS
Reverse transcriptaseHuman immunodeficiency virus 1>574000 nMBindingDB
Ribonuclease pancreaticBos taurusP61823>300000 nM|> 300000.0 nMBindingDB, NPASS
S-117Homo sapiens= 78.15 nMNPASS
SAOS-2Homo sapiens= 17.77 nMNPASS
SARS-CoV-2Severe acute respiratory syndrome coronavirus 2> 20000.0 nM|> 19952.62 nMNPASS
SASHomo sapiens= 1.241 nM|= 6000.0 nMNPASS
SBC-1Homo sapiens= 27.79 nMNPASS
RO82-W-1Homo sapiens= 14.91 nMNPASS
SBC-5Homo sapiens= 32.15 nMNPASS
RMG-IHomo sapiens= 244.5 nMNPASS
RH-18Homo sapiens= 389.64 nMNPASS
PANC-03-27Homo sapiens= 7.103 nMNPASS
PANC-08-13Homo sapiens= 44.89 nMNPASS
PANC-1Homo sapiens= 180.0 nM|= 90.0 nMNPASS
PBMCHomo sapiens> 10000.0 nMNPASS
PC-14Homo sapiens= 13.58 nMNPASS
PC-3Homo sapiens= 57.0 nM|= 310.0 nM|= 1414.4 nM|= 52.0 nM|= 1400.0 nM|= 16240.0 nM|= 30.0 nM|= 12.0 nM|= 9.753 nM|= 78.0 nM|= 1200.0 nM|= 10.0 nM|= 2500.0 nM|= 100.0 nM|= 6960.0 nM|= 400.0 nM|> 40000.0 nM|= 18240.0 nM|= 2400.0 nMNPASS
PC-3MHomo sapiens= 480.0 nM|= 190.0 nMNPASS
PFSK-1Homo sapiens= 26.03 nMNPASS
PSN1Homo sapiens= 3.069 nMNPASS
Panc1005Homo sapiens= 19.68 nMNPASS
Panel (56 tumour cell lines)= 40.0 nMNPASS
Plasmodium falciparumPlasmodium falciparum= 0.83 nM|= 1.41 nM|= 1.12 nM|= 1.32 nM|= 0.89 nM|= 0.56 nM|= 794.33 nM|= 1258.93 nM|= 1000.0 nM|= 501.19 nMNPASS
QG-56= 0.00463 ug.mL-1NPASS
QIMR-WILHomo sapiens= 0.7753 nMNPASS
RCC10RGBHomo sapiens= 113.62 nMNPASS
RCM-1Homo sapiens= 28.66 nMNPASS
RDHomo sapiens= 15.74 nM|= 4490.0 nM|= 1240.0 nM|= 1720.0 nMNPASS
RERF-LC-MSHomo sapiens= 22.87 nMNPASS
RH-1Homo sapiens= 3.86 nMNPASS
RKOHomo sapiens= 4.23 nM|< 1850.0 nM|= 61.7 nMNPASS
SW 1116Homo sapiens= 190.35 nMNPASS
SCC-15Homo sapiens= 18.57 nMNPASS
SCC-4Homo sapiens= 19.26 nMNPASS
SK-N-ASHomo sapiens= 5.377 nMNPASS
SK-N-DZHomo sapiens= 21.69 nMNPASS
SK-N-FIHomo sapiens= 106.62 nMNPASS
SK-NEP-1Homo sapiens= 1.227 nMNPASS
SK-OV-3Homo sapiens= 37.0 nM|= 20.0 nM|= 51.0 nM|= 14.0 nM|= 1.54 ug.mL-1|= 2544.0 nM|= 7210.91 nM|= 5.5 nM|= 5500.0 nM|= 3820.0 nM|= 2560.0 nM|= 4860.0 nMNPASS
SK-PN-DWHomo sapiens= 1.16 nMNPASS
SK-UT-1Homo sapiens= 3.067 nMNPASS
SK-VLBHomo sapiens= 41.0 nM|= 53.0 nMNPASS
SKG-IIIaHomo sapiens= 4.582 nMNPASS
SMMC-7721Homo sapiens= 20.0 nM|= 3.0 nM|= 1080.0 nM|= 450.0 nM|> 10000.0 nM|= 3950.0 nMNPASS
SN12CHomo sapiens= 4.503 nMNPASS
SNB-75Homo sapiens= 17.34 nMNPASS
SNU-387Homo sapiens= 256.33 nMNPASS
SNU-423Homo sapiens= 128.79 nMNPASS
SNU-449Homo sapiens= 194.29 nMNPASS
SNU-5Homo sapiens= 42.71 nMNPASS
SNU-638Homo sapiens= 98.0 nM|= 280.0 nMNPASS
SNU-C2BHomo sapiens= 35.38 nMNPASS
SNU1Homo sapiens= 1.088 nMNPASS
SK-MES-1Homo sapiens= 10.0 nM|= 10.78 nMNPASS
SCC-25Homo sapiens= 56.73 nMNPASS
SK-MEL3Homo sapiens= 329.41 nMNPASS
SK-MEL-28Homo sapiens= 40.0 nM|= 17.13 nM|< 10.0 nM|= 2260.0 nMNPASS
SCC-9Homo sapiens= 33.19 nMNPASS
SCHHomo sapiens= 628.09 nMNPASS
SF-126Homo sapiens= 2.835 nMNPASS
SF-268Homo sapiens= 59.0 nM= 40.0 nM|= 190.0 nM|= 70.0 nM|= 3.379 nMNPASS
SF-295Homo sapiens= 7.909 nMNPASS
SF-539Homo sapiens= 9.009 nMNPASS
SGC-7901Homo sapiens< 1850.0 nM|= 5800.0 nMNPASS
SH-4Homo sapiens= 59.8 nMNPASS
SH-SY5YHomo sapiens= 610.0 nMNPASS
SHP77Homo sapiens= 1543.63 nMNPASS
SJRH30Homo sapiens= 298.06 nMNPASS
SJSA-1Homo sapiens= 18.0 nMNPASS
SK-BR-3Homo sapiens= 20.0 nM|< 10.0 nM|= 210.0 nMNPASS
SK-HEP1Homo sapiens= 7.253 nM|= 900.0 nMNPASS
SK-LMS-1Homo sapiens= 180.87 nMNPASS
SK-LU-1Homo sapiens= 4.713 nMNPASS
SK-MEL-1Homo sapiens= 51.29 nMNPASS
SK-MEL-2Homo sapiens= 75.0 nM|= 165.0 nM|= 6.88 ug.mL-1|= 7860.0 nM|= 54.75 nMNPASS
SK-MEL-24Homo sapiens= 38.51 nM|= 460.0 nMNPASS
LNCaPHomo sapiens= 86.1 nMNPASS
LN-405Homo sapiens= 517.64 nMNPASS
LB2518-MELHomo sapiens= 87.25 nMNPASS
LK-2Homo sapiens= 35.53 nMNPASS
CWR22RHomo sapiens= 9.314 nMNPASS
Ca-SkiHomo sapiens= 4.97 nM|= 1800.0 nMNPASS
Ca9-22Homo sapiens= 2.211 nMNPASS
CaR-1Homo sapiens= 6.427 nMNPASS
Caco-2Homo sapiens= 9550.0 nMNPASS
Calu-3Homo sapiens= 32.8 nMNPASS
Calu-6Homo sapiens= 178.95 nMNPASS
LN-229Homo sapiens= 0.32 nMNPASS
Canalicular multispecific organic anion transporter 2Homo sapiensO15438> 133000.0 nMNPASS
Caov-3 cell line= 2900000.0 nM|= 30.0 nMNPASS
Capan-2Homo sapiens= 452.29 nMNPASS
ChaGo-K-1Homo sapiens= 304.67 nMNPASS
Col2Homo sapiens= 45.0 nMNPASS
Cystic fibrosis transmembrane conductance regulatorHumanP13569>50000 nMBindingDB
D-247MGHomo sapiens= 39.54 nMNPASS
D-263MGHomo sapiens= 9.114 nMNPASS
D-336MGHomo sapiens= 5.205 nMNPASS
D-392MGHomo sapiens= 17.73 nMNPASS
D-423MGHomo sapiens= 2.551 nMNPASS
CW-2Homo sapiens= 35.45 nMNPASS
D-502MGHomo sapiens= 22.59 nMNPASS
CTV-1Homo sapiens= 0.9054 nMNPASS
CT26.WTMus musculus= 430.0 nMNPASS
CNE-2Homo sapiens= 100.0 nM|= 980.0 nMNPASS
COLO 205Homo sapiens= 5.4 nM|= 50.0 nMNPASS
COLO-320-HSRHomo sapiens= 62.09 nMNPASS
COLO-668Homo sapiens= 22.32 nMNPASS
COLO-678Homo sapiens= 3682.73 nMNPASS
COLO-679Homo sapiens= 4791.52 nMNPASS
COLO-680NHomo sapiens= 72.45 nMNPASS
COLO-684Homo sapiens= 13.82 nMNPASS
COLO-741Homo sapiens= 109.27 nMNPASS
COLO-792Homo sapiens= 169.17 nMNPASS
COLO-800Homo sapiens= 0.4281 nMNPASS
COLO-824Homo sapiens= 269.5 nMNPASS
COLO-829Homo sapiens= 11.67 nMNPASS
COR-L105Homo sapiens= 184.93 nMNPASS
COR-L23Homo sapiens= 6.849 nMNPASS
COR-L88Homo sapiens= 40.93 nMNPASS
CP50-MEL-BHomo sapiens= 72.08 nMNPASS
CP66-MELHomo sapiens= 208.15 nMNPASS
CT26Mus musculus= 34.0 nMNPASS
CTB-1Homo sapiens= 0.4292 nMNPASS
CNEHomo sapiens= 340.0 nMNPASS
D-542MGHomo sapiens= 291.41 nMNPASS
D283 Med= 3.198 nMNPASS
DNA topoisomerase type IB small subunitLeishmamajorQ95Z89= 670.0 nMNPASS
DOHH-2Homo sapiens= 0.6022 nMNPASS
DOKHomo sapiens= 18.92 nMNPASS
DSH1Homo sapiens= 15.75 nMNPASS
DU-145Homo sapiens= 10.0 nM|= 3200.0 nM|= 1460.0 nM|= 3570.0 nM|= 940.0 nM|= 660.0 nM|= 1000.0 nM|= 400.0 nM|= 20.0 nM|= 610.0 nM|= 310.0 nM|= 2370.0 nM|= 15.0 nM|= 9290.0 nM|= 1060.0 nM|= 28.7 nM|= 2281.94 nM|= 390.0 nM|= 800.0 nM|= 4010.0 nM|= 110.0 nM|= 950.0 nM|= 29.0 nM|= 100.0 nM|= 50.0 nM|= 16.0 nM|= 1990.0 nM|= 70.0 nM|= 33.45 nM|= 210.0 nMNPASS
DU-4475Homo sapiens= 3.067 nMNPASS
DaoyHomo sapiens= 0.4809 nMNPASS
Deoxyribonuclease-1Bos taurusP00639>300000 nM|> 300000.0 nMBindingDB, NPASS
Deoxyribonuclease-2-alphaSus scrofaO62855>300000 nM|> 300000.0 nMBindingDB, NPASS
Detroit 551Homo sapiens= 990.0 nMNPASS
Detroit562Homo sapiens= 13.34 nMNPASS
DoTc2-4510Homo sapiens= 4.032 nMNPASS
EC-GI-10Homo sapiens= 7.904 nMNPASS
ECC10Homo sapiens= 3.853 nMNPASS
EFM-19Homo sapiens= 126.89 nMNPASS
EFO-21Homo sapiens= 20.32 nMNPASS
EFO-27Homo sapiens= 80.99 nMNPASS
EGI-1Homo sapiens= 25.07 nMNPASS
EKVXHomo sapiens= 436.37 nMNPASS
DNA topoisomerase II alphaHomo sapiensP11388> 300000.0 nMNPASS
D-566MGHomo sapiens= 0.1315 nMNPASS
DNA topoisomerase IMus musculusQ04750= 40000.0 nM|= 12000.0 nMNPASS
DNA topoisomerase IHomo sapiensP11387= 350.0 nM= 700.0 nM|= 679.0 nM|= 127000.0 nM|= 680.0 nM|= 300.0 nM|= 4000.0 nM|= 17000.0 nM|= 9000.0 nM|= 20000.0 nM|= 2200.0 nM|= 3750.0 nM|= 4950.0 nM|= 4750.0 nM|= 25.0 nM|= 2500.0 nM|= 27000.0 nM|= 62900.0 nM|= 62000.0 nM|= 224.0 nM|= 2430.0 nMNPASS
DBHomo sapiens= 1.161 nMNPASS
DBTRG-05MGHomo sapiens= 40.86 nMNPASS
DC3FCricetulus griseus= 6.0 nMNPASS
DELHomo sapiens= 0.8157 nMNPASS
DJM-1Homo sapiens= 436.47 nMNPASS
DK-MGHomo sapiens= 84.75 nMNPASS
DLD-1Homo sapiens= 14000000.0 nM|= 210.0 nMNPASS
DMS-114Homo sapiens= 81.1 nMNPASS
DMS-273Homo sapiens= 6.072 nMNPASS
DMS-79Homo sapiens= 31.85 nMNPASS
DNA ligaseEnterobacteria phage T4P00970>300000 nM|> 300000.0 nMBindingDB, NPASS
DNA topoisomeraseBos taurus17000 nMBindingDB
DNA topoisomeraseBos taurusA0JN73= 17000.0 nMNPASS
DNA topoisomerase 1Chlorocebus aethiopsQ7YR2627000 nM|= 27000.0 nMBindingDB, NPASS
DNA topoisomerase 1Homo sapiensP11387350 nM127000 nM|679 nM|1400 nM|4000 nM|17000 nM|9000 nM|700 nM|1600 nM|680 nM|300 nM|20000 nM|2200 nM|224 nM|4950 nM|4750 nM|3750 nM|2500 nM|25 nM|27000 nM|62900 nM|62 nMBindingDB
DNA topoisomerase 1HumanP113872.0e+4 nMBindingDB
DNA topoisomerase 1Mus musculusQ0475040000 nM|12000 nMBindingDB
DNA topoisomerase 2-alphaHomo sapiensP11388>300000 nMBindingDB
DNA topoisomerase 2-alphaHumanP11388>3.50e+5 nMBindingDB
DNA topoisomerase ILeishmadonovani (strain BPK282A1)E9BRC0= 21920.0 nM|= 9200.0 nMNPASS
EM-2Homo sapiens= 4.08 nMNPASS
CHP-212Homo sapiens= 1.026 nMNPASS
CGTH-W-1Homo sapiens= 3.275 nMNPASS
A498Homo sapiens= 7.077 nMNPASS
A549Homo sapiens= 2530.0 nM|= 8.0 nM|= 330000.0 nM|= 14.0 nM|= 67.0 nM|= 69.0 nM|= 3120.0 nM|= 4.0 nM|= 10.0 nM|= 58.0 nM|= 3100.0 nM|= 47.0 nM|= 40.0 nM|= 5.379 nM|= 57.0 nM|= 30.0 nM|= 3600.0 nM|= 0.072 ug.mL-1|= 91.0 nM|= 260.0 nM|= 33.8 nM|= 2610.0 nM|= 15.8 nM|= 14.09 nM|= 99.0 nM|= 37050.0 nM|= 650.0 nM|< 10.0 nM|= 16.0 nM|= 1300.0 nM|= 1.0 nM|= 26450.0 nM|= 100.0 nM|= 1600.0 nM|= 350.0 nM|= 9.0 nM|= 240.0 nM|= 6.0 nM|= 8.63 nM|= 700.0 nM|= 13640.0 nM|< 1000.0 nM|= 5500.0 nM|= 8870.0 nM|= 5930.0 nM|= 2210.0 nM|= 1310.0 nM|= 4430.0 nM|= 0.32 nM|= 90.0 nM|= 2800.0 nM|= 3320.0 nM|= 39.0 nM|= 32110.0 nM|= 50880.0 nM|= 1560.0 nM|= 1000.0 nM|= 170.0 nM|= 8900.0 nM|= 470.0 nM|= 32100.0 nM|= 74.0 nM|= 370.0 nM|< 1850.0 nMNPASS
A673Homo sapiens= 0.8149 nMNPASS
A704Homo sapiens= 15.35 nMNPASS
ABC-1Homo sapiens= 3.468 nMNPASS
ACHNHomo sapiens= 6.663 nMNPASS
ACNHomo sapiens= 85.66 nMNPASS
AGSHomo sapiens= 20.0 nM|= 16.13 nM|= 23760.0 nMNPASS
ALL-POHomo sapiens= 1.534 nMNPASS
AM-38Homo sapiens= 4.408 nMNPASS
AN3-CAHomo sapiens= 33.98 nMNPASS
ASPC1Homo sapiens= 168.37 nMNPASS
ATN-1Homo sapiens= 2.043 nMNPASS
ATP-binding cassette sub-family C member 2Homo sapiensQ92887>133000 nMBindingDB
ATP-binding cassette sub-family C member 3Homo sapiensO15438>133000 nMBindingDB
ATP-binding cassette sub-family C member 4Homo sapiensO154397400 nMBindingDB
AU565Homo sapiens= 3.68 nMNPASS
BALL-1Homo sapiens= 108.94 nMNPASS
BB30-HNCHomo sapiens= 21.55 nMNPASS
A4-FukHomo sapiens= 1.749 nMNPASS
BB49-HNCHomo sapiens= 120.28 nMNPASS
A388Homo sapiens= 10.12 nMNPASS
A2780Homo sapiens= 7.0 nM|= 280.0 nM|= 4.0 nM|= 200.0 nM|= 0.07 ug.mL-1|= 300.0 nM|= 260.0 nM|= 2.902 nM|= 13.0 nM|= 900.0 nM|= 29.0 nMNPASS
23132-87Homo sapiens= 19.46 nMNPASS
4T1Mus musculus= 170.0 nMNPASS
5637Homo sapiens= 4.183 nMNPASS
639-VHomo sapiens= 0.1714 nMNPASS
647-VHomo sapiens= 0.8964 nMNPASS
697Homo sapiens= 2.029 nMNPASS
769-PHomo sapiens= 25.34 nMNPASS
786-0Homo sapiens= 5.021 nMNPASS
8-MG-BAHomo sapiens= 1.502 nMNPASS
8305CHomo sapiens= 93.98 nMNPASS
833K= 10.0 nMNPASS
8505CHomo sapiens= 3.301 nMNPASS
A-375Homo sapiens= 3.688 nM|= 187.0 nM|= 13.0 nM|= 660.0 nMNPASS
A-427Homo sapiens= 24.0 nM|= 4.251 nMNPASS
A-431Homo sapiens= 11.0 nM|= 1552.36 nMNPASS
A101DHomo sapiens= 257.84 nMNPASS
A172Homo sapiens= 140.0 nM|= 12.76 nMNPASS
A204Homo sapiens= 4.525 nMNPASS
A2058Homo sapiens= 3.599 nMNPASS
A3-KAWHomo sapiens= 1.669 nMNPASS
CHL-1Homo sapiens= 6.091 nMNPASS
BB65-RCCHomo sapiens= 1.853 nMNPASS
BE-13Homo sapiens= 4.564 nMNPASS
CAKI-1Homo sapiens= 5.354 nMNPASS
CAKI-2Homo sapiens= 3960.0 nMNPASS
CAL-120Homo sapiens= 594.73 nMNPASS
CAL-12THomo sapiens= 262.05 nMNPASS
CAL-27Homo sapiens= 2.018 nMNPASS
CAL-33Homo sapiens= 5.997 nMNPASS
CAL-39Homo sapiens= 19.16 nMNPASS
CAL-51Homo sapiens= 29.74 nMNPASS
CAL-54Homo sapiens= 4.758 nMNPASS
CAL-62Homo sapiens= 0.9836 nMNPASS
CAL-72Homo sapiens= 150.57 nMNPASS
CAL-85-1Homo sapiens= 7923.68 nMNPASS
CAMA-1Homo sapiens= 70.0 nM|= 87.43 nMNPASS
CAPAN-1Homo sapiens= 14.95 nM|= 210.0 nMNPASS
CAS-1Homo sapiens= 121.91 nMNPASS
CCD 19LuHomo sapiens= 2.0 ug.mL-1NPASS
CCRF-CEMHomo sapiens= 0.005 ug.mL-1|= 5300.0 nM|= 0.84 nM|= 3.0 nM|= 40.0 nM|= 5.0 nM|= 5.547 nM|= 80.0 nM|= 2.0 nMNPASS
CCRF-SBHomo sapiens= 3.0 nMNPASS
CFPAC-1Homo sapiens= 14.75 nMNPASS
CA46Homo sapiens= 520.0 nMNPASS
BCPAPHomo sapiens= 3.041 nMNPASS
C8166Homo sapiens= 41.48 nMNPASS
C3AHomo sapiens= 56.87 nMNPASS
BENHomo sapiens= 107.08 nMNPASS
BFTC-905Homo sapiens= 0.1398 nMNPASS
BFTC-909Homo sapiens= 6.925 nMNPASS
BGC-823Homo sapiens= 9670.0 nM|= 9700.0 nM|= 210.0 nM|= 57.0 nMNPASS
BHT-101Homo sapiens= 1.822 nMNPASS
BHYHomo sapiens= 5.31 nMNPASS
BJHomo sapiens= 7.67 nM> 40000.0 nMNPASS
BPH-1Homo sapiens= 2.082 nMNPASS
BT-20Homo sapiens= 70.0 nM|< 10.0 nM|= 25.99 nMNPASS
BT-474Homo sapiens= 12750.0 nM|= 1985.76 nMNPASS
BT-549Homo sapiens= 17.64 nMNPASS
BV-173Homo sapiens= 2.381 nMNPASS
BXPC-3Homo sapiens= 240.0 nM|= 116.78 nM|= 62.5 nMNPASS
BeckerHomo sapiens= 23.34 nMNPASS
Bel-7402Homo sapiens= 7.0 nM|= 2.72 ug.mL-1|= 12500.0 nM|= 170.0 nM|= 260.0 nM|= 14.0 nMNPASS
Bile salt export pumpHomo sapiensO95342>135000 nM|>133000 nM|> 135000.0 nM|> 133000.0 nMBindingDB, NPASS
C-33-AHomo sapiens= 6.477 nMNPASS
C2BBe1Homo sapiens= 2.438 nMNPASS
C32Homo sapiens= 13.37 nMNPASS
C6Rattus norvegicus< 1850.0 nMNPASS
EOL1Homo sapiens= 0.2708 nMNPASS
Canalicular multispecific organic anion transporter 1Homo sapiensQ92887> 133000.0 nMNPASS
ES1Homo sapiens= 0.09574 nMNPASS
IST-SL1Homo sapiens= 34.38 nMNPASS
IntegraseHuman immunodeficiency virus 1>100000 nMBindingDB
J-RT3-T3-5Homo sapiens= 2.579 nMNPASS
J82Homo sapiens= 4.722 nMNPASS
JARHomo sapiens= 14.54 nMNPASS
JEG-3Homo sapiens= 13.12 nMNPASS
JVM-2Homo sapiens= 3029.5 nMNPASS
JVM-3Homo sapiens= 2.504 nMNPASS
IST-MES1Homo sapiens= 10.56 nMNPASS
JurkatHomo sapiens= 5.6 nM|= 1.4 nM|= 26.0 nM|= 110.0 nM|= 85.0 nM|= 22000.0 nM|= 51500.0 nM|= 100.0 nMNPASS
K562Homo sapiens= 57.0 nM|= 40.0 nM|= 1400.0 nM|= 80.0 nM|= 2.0 nM|= 590.0 nM|= 1180.0 nM|= 1077.74 nM|= 31.0 nM|= 400.0 nM|= 130.0 nM|= 5370.0 nM|< 3.0 nM|= 90.0 nM|= 711.0 nM|= 70.0 nM|= 320.0 nM|= 2690.0 nM|= 580.0 nMNPASS
KALS-1Homo sapiens= 69.89 nMNPASS
KARPAS-299Homo sapiens= 2892.53 nMNPASS
KARPAS-45Homo sapiens= 134.47 nMNPASS
KATO III stomach cancer cell lines= 46000000.0 nM|= 1170.0 nMNPASS
KBHomo sapiens= 3.6 nM|= 0.01 ug.mL-1= 9.0 nM|= 40.0 nM|= 70.0 nM|= 30.0 nM|= 35.0 nM|= 1040.0 nM|= 0.01 ug.mL-1|= 0.04 ug.mL-1|= 8.0 nM|< 0.005 ug.mL-1|= 20.0 nM|= 28.7 nM|= 3.0 nM|= 38.0 nM|= 1220.0 nM|< 13.0 nM|= 8.8 nM|= 121.0 nM|= 37.0 nM|= 50.0 nMNPASS
KB 3-1Homo sapiens= 10.0 nM|= 20.0 nMNPASS
KB VCR R= 9.0 nM|= 0.03 ug.mL-1NPASS
K5Homo sapiens= 3.201 nMNPASS
IST-MEL1Homo sapiens= 3.81 nMNPASS
IMR-90Homo sapiens= 430.0 nMNPASS
IMR-32Homo sapiens= 80.0 nMNPASS
HeLaHomo sapiens= 117.2 nM|= 500.0 nM|= 1080.0 nM|= 0.19 ug.mL-1|= 72.0 nM|= 200.0 nM|= 1850.0 nM|= 860.0 nM|= 630.0 nM|= 1220.0 nM|= 580.0 nM|= 940.0 nM|= 400.0 nM|= 1100.0 nM|= 8.9 nM|= 1500.0 nM|= 8930.0 nM|= 1010.0 nM|= 1570.0 nM|= 0.28 ug.mL-1|= 24.0 nM|= 130.0 nM|= 420.0 nM|= 11620.0 nM|= 180.0 nM|= 410.0 nM|= 14000.0 nM|= 1590.0 nM|= 6130.0 nM|= 19800.0 nM|= 590.0 nM|= 60010.0 nM|= 90.0 nM|= 60.0 nM|= 10100.0 nM|= 3800.0 nM|= 2620.0 nM|= 120.0 nM|= 1370.0 nM|= 80.0 nM|= 1300.0 nM|> 50000.0 nM|= 660.0 nM|= 6510.0 nM|= 1660.0 nM|= 8280.0 nM|= 6000.0 nM|= 230.0 nMNPASS
Hep 3B2Homo sapiens= 434.29 nMNPASS
HepG2Homo sapiens= 6.3 nM|= 0.09 ug.mL-1|= 30.0 nM|= 300.0 nM|= 130.0 nM|= 200.0 nM|= 455.0 nM|= 60.0 nM|= 6400.0 nM|= 20.0 nM|< 100.0 nM|= 10.0 nM|= 32300.0 nM|= 600.0 nM|= 50.0 nM|< 1000.0 nM|= 4920.0 nM|= 13200.0 nM|= 500.0 nM|= 430.0 nM|= 4370.0 nM|= 370.0 nM|= 6080.0 nM|= 1360.0 nM|= 4790.0 nM|= 660.0 nM|= 5690.0 nM|= 400.0 nM|= 40.0 nM|= 110.0 nM|= 33.16 nM|< 1850.0 nM|= 3500.0 nMNPASS
Heterogeneous nuclear ribonucleoprotein A1Homo sapiensP0965182.7 nM|= 82.7 nMBindingDB, NPASS
Histone deacetylaseHomo sapiensO15379|P56524|Q13547|Q8WUI4|Q92769|Q969S8|Q96DB2|Q9BY41|Q9UBN7|Q9UKV0|Q9UQL650 nMBindingDB
Histone deacetylaseHomo sapiensQ13547|O15379|Q9UBN7|Q92769|Q9UQL6|Q8WUI4|Q9BY41|Q96DB2|P56524|Q9UKV0|Q969S8= 50.0 nMNPASS
Hs-578THomo sapiens= 144.69 nMNPASS
HuCCT-1Homo sapiens= 73.21 nMNPASS
HuO-3N1Homo sapiens= 12.65 nMNPASS
HuO9Homo sapiens= 2.881 nMNPASS
HuP-T3Homo sapiens= 36.35 nMNPASS
HuP-T4Homo sapiens= 0.8814 nMNPASS
HuTu80Homo sapiens= 3.382 nMNPASS
Huh-7Homo sapiens< 100.0 nM|= 150.0 nM|= 60.0 nM|= 115.84 nM|= 0.32 nM|= 2.3 nM|< 1850.0 nMNPASS
Human immunodeficiency virus type 1 integraseHuman immunodeficiency virus 1Q7ZJM1> 100000.0 nMNPASS
Human immunodeficiency virus type 1 reverse transcriptaseHuman immunodeficiency virus 1Q72547> 200.0 ug.mL-1NPASS
IA-LMHomo sapiens= 12.0 nMNPASS
IGR-1Homo sapiens= 151.26 nMNPASS
IGROV-1Homo sapiens= 1650.0 nM|= 12.0 nM|= 36.34 nMNPASS
KE-37Homo sapiens= 1.535 nMNPASS
KG-1Homo sapiens= 2310.0 nMNPASS
KG-1= 1.11 nM|= 1600.0 nMNPASS
KGNHomo sapiens= 10.59 nMNPASS
KYSE-510Homo sapiens= 6.754 nMNPASS
KYSE-520 cell line= 82.56 nMNPASS
KYSE-70 cell line= 92.14 nMNPASS
Kasumi 1= 4.066 nMNPASS
L-363Homo sapiens= 1.869 nMNPASS
L-428Homo sapiens= 148.3 nMNPASS
L02Homo sapiens= 2150.0 nM|> 150000.0 nM|= 140.0 nMNPASS
L1210Mus musculus= 30.0 nM|= 23.0 nM|= 330.0 nM|= 15.0 nM|= 126.0 nM|= 14.0 nM|= 180.0 nM|= 60.0 nM|= 510.0 nMNPASS
L2987Homo sapiens= 400.0 nMNPASS
LAMA-84Homo sapiens= 7.02 nMNPASS
LAN-6Homo sapiens= 124.47 nMNPASS
LB1047-RCCHomo sapiens= 7.897 nMNPASS
LB2241-RCCHomo sapiens= 2.076 nMNPASS
LB373-MEL-DHomo sapiens= 91.19 nMNPASS
LB771-HNCHomo sapiens= 196.84 nMNPASS
LB831-BLCHomo sapiens= 18.37 nMNPASS
LC-2-adHomo sapiens= 2.806 nMNPASS
LCLC-103H cell line= 20.49 nMNPASS
LCLC-97TM1Homo sapiens= 8.136 nMNPASS
KYSE-450Homo sapiens= 23.73 nMNPASS
HUVECHomo sapiens= 200.0 nM|= 10.0 nM|= 60.0 nM|= 12.0 nMNPASS
KYSE-410Homo sapiens= 78.11 nMNPASS
KYSE-180Homo sapiens= 13.18 nMNPASS
KINGS-1Homo sapiens= 332.9 nMNPASS
KLEHomo sapiens= 411.5 nMNPASS
KM-H2Homo sapiens= 55.67 nMNPASS
KM12Homo sapiens= 74.99 nMNPASS
KMOE-2Homo sapiens= 11.26 nMNPASS
KNS-42Homo sapiens= 33.14 nMNPASS
KNS-62Homo sapiens= 7.701 nMNPASS
KNS-81-FDHomo sapiens= 19.42 nMNPASS
KOSC-2Homo sapiens= 4.393 nMNPASS
KP-4Homo sapiens= 3.162 nMNPASS
KP-N-YNHomo sapiens= 102.97 nMNPASS
KP-N-YSHomo sapiens= 736.29 nMNPASS
EPLC-272HHomo sapiens= 72.8 nMNPASS
KU-19-19Homo sapiens= 22.03 nMNPASS
KU812 cell line= 8.365 nMNPASS
KURAMOCHIHomo sapiens= 3634.01 nMNPASS
KY821Homo sapiens= 8.123 nMNPASS
KYSE-140Homo sapiens= 69.74 nMNPASS
KYSE-150 cell line= 245.96 nMNPASS
KYSE-270Homo sapiens= 5.223 nMNPASS
HTC-C3Homo sapiens= 31.47 nMNPASS
KS-1Homo sapiens= 57.87 nMNPASS
HT1197Homo sapiens= 1093.19 nMNPASS
G-402Homo sapiens= 24.5 nMNPASS
GAKHomo sapiens= 218.07 nMNPASS
GAMGHomo sapiens= 1.527 nMNPASS
GB-1Homo sapiens= 4.677 nMNPASS
GCIYHomo sapiens= 66.15 nMNPASS
GCTHomo sapiens= 5.023 nMNPASS
GI-1Homo sapiens= 3.365 nMNPASS
GI-ME-NHomo sapiens= 33.89 nMNPASS
GMS-10Homo sapiens= 7.311 nMNPASS
GOTOHomo sapiens= 0.7058 nMNPASS
GP5dHomo sapiens= 12.49 nMNPASS
GR-STHomo sapiens= 0.701 nMNPASS
HT55Homo sapiens= 192.44 nMNPASS
H-EMC-SSHomo sapiens= 95.58 nMNPASS
H22Mus musculus= 540.0 nMNPASS
H4Homo sapiens= 0.6154 nMNPASS
H9Homo sapiens= 0.3582 nMNPASS
HAL-01Homo sapiens= 2.551 nMNPASS
HC-1Homo sapiens= 3.344 nMNPASS
G-401Homo sapiens= 19.16 nMNPASS
HCC 2998Homo sapiens= 150.28 nMNPASS
G-361Homo sapiens= 2544.45 nMNPASS
FTC-133Homo sapiens= 4.567 nMNPASS
ES3Homo sapiens= 0.9311 nMNPASS
ES4Homo sapiens= 1.474 nMNPASS
ES5Homo sapiens= 0.7735 nMNPASS
ES6Homo sapiens= 88.05 nMNPASS
ES7Homo sapiens= 0.02543 nMNPASS
ES8Homo sapiens= 0.7956 nMNPASS
ESS-1Homo sapiens= 7.079 nMNPASS
ETK-1Homo sapiens= 34.89 nMNPASS
EW-1Homo sapiens= 1.777 nMNPASS
EW-11Homo sapiens= 2.659 nMNPASS
EW-13Homo sapiens= 3.267 nMNPASS
EW-16Homo sapiens= 0.1214 nMNPASS
EW-18Homo sapiens= 150.08 nMNPASS
EW-22Homo sapiens= 0.5566 nMNPASS
EW-24Homo sapiens= 4.033 nMNPASS
EW-3Homo sapiens= 0.3192 nMNPASS
Erythrocyte= 429.9 ug.mL-1NPASS
Eukaryotic translation initiation factor 2-alpha kinase 3Homo sapiensQ9NZJ5> 55700.0 nMNPASS
Eukaryotic translation initiation factor 2-alpha kinase 3HumanQ9NZJ5>55700 nMBindingDB
FaDuHomo sapiens= 0.5392 nMNPASS
HCC1187Homo sapiens= 314.07 nMNPASS
GT3TKBHomo sapiens= 1.759 nMNPASS
HCC1419Homo sapiens= 4155.69 nMNPASS
HL-60Homo sapiens= 66.0 nM|= 5.0 nM|= 18.0 nM|= 13.0 nM|= 130000.0 nM|= 89.0 nM|= 800.0 nM|= 6.0 nM|= 65.0 nM|= 67.0 nM|= 590.0 nM|= 100.0 nM|= 17.0 nM|= 600.0 nM|= 3.734 nM|= 60.0 nM|= 15.0 nM|= 920.0 nM|= 19.0 nM|= 6.7 nM|= 20.0 nM|= 70.0 nM|= 420.0 nM|< 64.0 nM|= 1700.0 nM|= 910.0 nMNPASS
HLEHomo sapiens= 5.753 nMNPASS
HMV-2 cell line= 8.887 nMNPASS
HNHomo sapiens= 1.399 nMNPASS
HO-1-N-1Homo sapiens= 0.8385 nMNPASS
HOC-21 cell line= 0.0147 ug.mL-1NPASS
HCC1395Homo sapiens= 1367.35 nMNPASS
HOP-92Homo sapiens= 8.787 nMNPASS
HOSHomo sapiens= 1.398 nMNPASS
HPAF-IIHomo sapiens= 55.12 nMNPASS
HSC-2Homo sapiens= 11.7 nMNPASS
HSC-3Homo sapiens= 3.015 nMNPASS
HSC-4Homo sapiens= 0.1816 nMNPASS
HTHomo sapiens= 29.71 nMNPASS
HT-1080Homo sapiens= 80.0 nM|= 0.3944 nMNPASS
HT-1376Homo sapiens= 1780.55 nMNPASS
HT-144Homo sapiens= 17.86 nMNPASS
HT-29Homo sapiens= 60.0 nM= 46.0 nM|= 1400.0 nM|= 80.0 nM|= 87.8 nM|= 30.0 nM|= 14.0 nM|= 3160.0 nM|= 8810.0 nM|= 2000.0 nM|= 90.0 nM|= 120.0 nM|= 400.0 nM|= 850.0 nM|= 1220.0 nM|= 1070.0 nM|= 260.0 nM|= 10000.0 nM|= 85.52 nM|= 0.7 nM|= 60.0 nM|> 100000.0 nM|= 70.0 nM|> 150000.0 nM|= 1370.0 nMNPASS
HT-3Homo sapiens= 0.2119 nMNPASS
HHHomo sapiens= 13.52 nMNPASS
HGC-27Homo sapiens= 4.073 nM|> 150000.0 nM|= 166.0 nMNPASS
HOP-62Homo sapiens= 3293.6 nMNPASS
HELHomo sapiens= 6.311 nMNPASS
HCC1569Homo sapiens= 267.54 nMNPASS
HCC1806Homo sapiens= 3.143 nMNPASS
HEp-2Homo sapiens= 0.02 ug.mL-1|= 700.0 nM|= 3040.0 nM|= 3010.0 nMNPASS
HCC1954Homo sapiens= 266.61 nMNPASS
HCC2218Homo sapiens= 55.5 nMNPASS
HCC38Homo sapiens= 12.86 nMNPASS
HCC70Homo sapiens= 45.46 nM|= 44.0 nMNPASS
HCCLM9Homo sapiens> 150000.0 nMNPASS
HCE-4Homo sapiens= 1.814 nMNPASS
HCC1937Homo sapiens= 349.21 nMNPASS
HCT-116Homo sapiens= 1000.0 nM|= 9.0 nM|= 2.0 nM|= 2770.0 nM|= 130.0 nM|= 2300.0 nM|= 3970.0 nM|= 22.9 nM|< 100.0 nM|< 1000.0 nM|= 110.0 nM|< 10.0 nM|= 5.051 nM|= 16.0 nM|= 70.0 nM|= 90.0 nM|= 120.0 nM|= 11.5 nM|= 159.0 nM|= 1880.0 nM|= 30.0 nM|= 8.5 nM|= 20.0 nM|= 13.0 nM|= 400.0 nM|= 50.0 nM|= 250.0 nM|= 40.0 nM|< 1850.0 nM|= 600.0 nM|= 17.0 nM|= 2.01 nMNPASS
HCT-15Homo sapiens= 18.0 nM|= 80.0 nM|= 83.0 nM|= 3.0 nM|= 640.0 nM|= 760.0 nM|= 500.0 nM|= 67.0 nM|= 800.0 nM|= 0.096 ug.mL-1|= 166.0 nM|= 260.0 nM|= 9920.0 nM|= 1380.0 nM|= 776.97 nM|= 420.0 nM|= 2820.0 nM|= 520.0 nM|= 300.0 nM|= 6080.0 nM|= 600.0 nM|= 50.0 nM|= 20.0 nM|= 49.0 nM|= 1590.0 nMNPASS
HCT-8Homo sapiens= 7.0 nM|< 0.005 ug.mL-1|= 3150.0 nM|= 3200.0 nM|< 13.0 nM|= 260.0 nM|= 24.0 nMNPASS
HCE-THomo sapiens= 5.469 nMNPASS
HD-MY-ZHomo sapiens= 1.634 nMNPASS
HDLM-2Homo sapiens= 486.07 nMNPASS
HEC-1Homo sapiens= 18.13 nMNPASS
HEC-1B cell line= 8640.0 nM|= 60.0 nMNPASS
HEK-293THomo sapiens= 5650.0 nM|= 30.0 nM|= 690.0 nMNPASS
HEK293Homo sapiens= 7940.0 nM|= 1010.0 nM|= 780.0 nM|= 280.0 nM|= 10.0 nM|= 54690.0 nM|= 0.56 nM|= 1610.0 nM|= 600.0 nM|= 8750.0 nM|= 5.6 nMNPASS