| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| NCI-H1993 | Homo sapiens | | | = 9621.56 nM | | | NPASS |
| NCI-H2009 | Homo sapiens | | | = 68.13 nM | | | NPASS |
| NCI-H2029 | Homo sapiens | | | = 491.21 nM | | | NPASS |
| NCI-H2030 | Homo sapiens | | | = 48.53 nM | | | NPASS |
| NCI-H2052 | Homo sapiens | | | = 28.34 nM | | | NPASS |
| NCI-H2087 | Homo sapiens | | | = 5.074 nM | | | NPASS |
| NCI-H209 | Homo sapiens | | | = 0.04843 nM | | | NPASS |
| NCI-H2122 | Homo sapiens | | | = 12.98 nM | | | NPASS |
| NCI-H2126 | Homo sapiens | | | = 178.42 nM | | | NPASS |
| NCI-H2170 | Homo sapiens | | | = 13.71 nM | | | NPASS |
| NCI-H2228 | Homo sapiens | | | = 49.0 nM | | | NPASS |
| NCI-H2291 | Homo sapiens | | | = 975.25 nM | | | NPASS |
| NCI-H23 | Homo sapiens | | | = 40.69 nM|= 70.0 nM | | | NPASS |
| NCI-H2342 | Homo sapiens | | | = 618.33 nM | | | NPASS |
| NCI-H2347 | Homo sapiens | | | = 185.61 nM | | | NPASS |
| NCI-H2405 | Homo sapiens | | | = 58.48 nM | | | NPASS |
| NCI-H2452 | Homo sapiens | | | = 90.89 nM | | | NPASS |
| NCI-H28 | Homo sapiens | | | = 38.68 nM | | | NPASS |
| NCI-H292 | | | | = 2.24 nM | | | NPASS |
| NCI-H226 | Homo sapiens | | | = 22.49 nM | | | NPASS |
| NCI-H1975 | Homo sapiens | | | = 334.48 nM|= 1200.0 nM | | | NPASS |
| NCI-H1623 | Homo sapiens | | | = 0.7479 nM | | | NPASS |
| NCI-H1793 | Homo sapiens | | | = 27.23 nM | | | NPASS |
| NCI-H128 | Homo sapiens | | | = 18.0 nM | | | NPASS |
| NCI-H1299 | Homo sapiens | | | = 9.425 nM|= 3140.0 nM|= 800.0 nM | | | NPASS |
| NCI-H1304 | Homo sapiens | | | = 59.28 nM | | | NPASS |
| NCI-H1355 | Homo sapiens | | | = 66.1 nM | | | NPASS |
| NCI-H1395 | Homo sapiens | | | = 110.1 nM | | | NPASS |
| NCI-H1437 | Homo sapiens | | | = 34.93 nM | | | NPASS |
| NCI-H1563 | Homo sapiens | | | = 150.37 nM | | | NPASS |
| NCI-H1573 | Homo sapiens | | | = 173.4 nM | | | NPASS |
| NCI-H1581 | Homo sapiens | | | = 33.5 nM | | | NPASS |
| NCI-H358 | Homo sapiens | | | = 105.42 nM | | | NPASS |
| NCI-H1648 | Homo sapiens | | | = 38.07 nM | | | NPASS |
| NCI-H1650 | Homo sapiens | | | = 149.39 nM | | | NPASS |
| NCI-H1651 | Homo sapiens | | | = 14.95 nM | | | NPASS |
| NCI-H1666 | Homo sapiens | | | = 18.71 nM | | | NPASS |
| NCI-H1693 | Homo sapiens | | | = 26.69 nM | | | NPASS |
| NCI-H1703 | Homo sapiens | | | = 6.515 nM | | | NPASS |
| NCI-H1755 | Homo sapiens | | | = 208.78 nM | | | NPASS |
| NCI-H1770 | Homo sapiens | | | = 157.32 nM | | | NPASS |
| NCI-H1792 | Homo sapiens | | | = 40.12 nM | | | NPASS |
| NCI-H1838 | Homo sapiens | | | = 253.14 nM | | | NPASS |
| NCI-H441 | Homo sapiens | | | = 28.46 nM | | | NPASS |
| NCI-H720 | Homo sapiens | | | = 44.69 nM | | | NPASS |
| NCI-H460 | Homo sapiens | | = 6.9 nM | = 330.0 nM|= 180.0 nM|= 6.2 nM|> 25000.0 nM|> 1000.0 nM|= 13.0 nM|< 40.0 nM|= 30.0 nM|= 5.0 nM|= 2.0 nM|= 3.0 nM|= 24.12 nM|= 190.0 nM|= 110.0 nM|= 5370.0 nM|= 120.0 nM|= 790.0 nM | | | NPASS |
| NOS-1 | Homo sapiens | | | = 91.86 nM | | | NPASS |
| NTERA-2-cl-D1 | Homo sapiens | | | = 0.2738 nM | | | NPASS |
| NUGC-3 | Homo sapiens | | | = 3.136 nM | | | NPASS |
| NY | Homo sapiens | | | = 4356.62 nM | | | NPASS |
| OAW-28 | Homo sapiens | | | = 7.263 nM | | | NPASS |
| OAW-42 | Homo sapiens | | | = 8.99 nM | | | NPASS |
| OC-314 | Homo sapiens | | | = 2.506 nM | | | NPASS |
| OCI-AML2 | Homo sapiens | | | = 0.8868 nM | | | NPASS |
| OCUB-M | Homo sapiens | | | = 38.13 nM | | | NPASS |
| OE19 | Homo sapiens | | | = 3273.33 nM | | | NPASS |
| OE33 | Homo sapiens | | | = 25.55 nM | | | NPASS |
| OMC-1 | Homo sapiens | | | = 78.21 nM | | | NPASS |
| ONS-76 | Homo sapiens | | | = 2.406 nM | | | NPASS |
| OS-RC-2 | Homo sapiens | | | = 9.968 nM | | | NPASS |
| OVCAR-3 | Homo sapiens | | | = 956.65 nM | | | NPASS |
| OVCAR-4 | Homo sapiens | | | = 188.55 nM | | | NPASS |
| OVCAR-5 | Homo sapiens | | | = 43.33 nM | | | NPASS |
| OVCAR-8 | Homo sapiens | | | = 7.272 nM | | | NPASS |
| P12-Ichikawa | Homo sapiens | | | = 0.1016 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 330.0 nM|= 8.5 nM|= 61000.0 nM|= 33.0 nM|= 5.6 nM|> 10000.0 nM|= 5385.0 nM|= 500.0 nM|= 24.0 nM|= 0.004 nM|> 10.0 nM|= 5.0 nM|= 15.0 nM|= 25.0 nM|= 26.0 nM|= 0.08 ug.mL-1|= 4.0 nM|= 28.7 nM|= 3280.0 nM|= 6.0 nM|= 1700.0 nM|= 60.0 nM|= 30.0 nM|> 25000.0 nM|= 52.0 nM|= 57.0 nM|= 260.0 nM|= 15200.0 nM|< 100.0 nM|= 10.0 nM|< 1000.0 nM|= 6.8 nM|= 423.0 nM|= 37.1 nM|< 10.0 nM|= 300.0 nM|= 2780.0 nM|= 10070.0 nM|= 1980.0 nM|= 474.0 nM|= 786.0 nM|= 131.0 nM|= 120.0 nM|= 3600.0 nM|= 6300.0 nM|= 40.0 nM|= 0.15 nM|= 70.0 nM|= 220.0 nM|= 710.0 nM|= 960.0 nM|< 3.0 nM|= 140.0 nM|= 100.0 nM|= 190.0 nM|<= 100.0 nM|= 1290.0 nM|= 20.0 nM|= 2820.0 nM|= 7000.0 nM|= 7100.0 nM|= 5.5 nM|= 3.0 nM|= 35.0 nM|= 9520.0 nM|= 11360.0 nM|= 17650.0 nM|= 59130.0 nM|= 29810.0 nM|> 100000.0 nM|= 1410.0 nM|= 1270.0 nM|= 460.0 nM|= 1520.0 nM|= 80.0 nM|= 1.4 nM|= 130.0 nM|= 600.0 nM|= 1120.0 nM|= 310.0 nM|= 13700.0 nM|= 110.0 nM|= 400.0 nM|= 830.0 nM|= 1060.0 nM|= 590.0 nM|= 380.0 nM|= 350.0 nM|= 4540.0 nM|= 890.0 nM|= 1240.0 nM|= 6700.0 nM|= 3040.0 nM|= 1840.0 nM|= 5930.0 nM | | | NPASS |
| NCI-H446 | Homo sapiens | | | = 56.63 nM|> 200000.0 nM | | | NPASS |
| NOMO-1 | Homo sapiens | | | = 1.557 nM | | | NPASS |
| NKM-1 | Homo sapiens | | | = 0.441 nM | | | NPASS |
| NCI-H510A | Homo sapiens | | | = 1.699 nM | | | NPASS |
| NCI-H520 | Homo sapiens | | | = 25.01 nM | | | NPASS |
| NCI-H520 | | | | = 162.01 nM | | | NPASS |
| NCI-H526 | Homo sapiens | | | = 1.028 nM | | | NPASS |
| NCI-H596 | | | | = 2968.73 nM | | | NPASS |
| NCI-H630 | Homo sapiens | | | = 282.32 nM | | | NPASS |
| NCI-H650 | Homo sapiens | | | = 54.96 nM | | | NPASS |
| NCI-H661 | Homo sapiens | | | = 13.55 nM | | | NPASS |
| NCI-H69 | Homo sapiens | | | = 1.0 nM|= 311.44 nM | | | NPASS |
| NCI-H1155 | Homo sapiens | | | = 1.188 nM | | | NPASS |
| NCI-H727 | Homo sapiens | | | = 1009.34 nM | | | NPASS |
| NCI-H747 | Homo sapiens | | | = 296.49 nM | | | NPASS |
| NCI-H810 | Homo sapiens | | | = 50.3 nM | | | NPASS |
| NCI-H82 | Homo sapiens | | | = 588.29 nM | | | NPASS |
| NCI-H928 | | | | = 7.8 nM | | | NPASS |
| NCI-N87 | Homo sapiens | | | = 8.743 nM|= 2320.0 nM | | | NPASS |
| NEC8 | Homo sapiens | | | = 3.108 nM | | | NPASS |
| NH-12 | Homo sapiens | | | = 3.793 nM | | | NPASS |
| NHDF | Homo sapiens | | | = 5380.0 nM | | | NPASS |
| NMC-G1 | Homo sapiens | | | = 19.82 nM | | | NPASS |
| NCI-H1092 | Homo sapiens | | | = 43.18 nM | | | NPASS |
| MC-IXC | Homo sapiens | | | = 0.513 nM | | | NPASS |
| NBsusSR | Homo sapiens | | | = 0.1936 nM | | | NPASS |
| MCF-10A | Homo sapiens | | | = 2190.0 nM|= 2580.0 nM | | | NPASS |
| MCF-12A | Homo sapiens | | | < 10.0 nM | | | NPASS |
| MCF10 | Homo sapiens | | | = 24770.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | = 72.0 nM | = 3.1 nM|= 0.02 ug.mL-1|= 320.0 nM|= 40.0 nM|= 10000.0 nM|= 200.0 nM|= 1100.0 nM|= 3.0 nM|= 10.0 nM|= 7420.0 nM|= 60.0 nM|= 1220.0 nM|= 20.0 nM|= 14200.0 nM|= 2430.0 nM|= 650.0 nM|= 70.0 nM|= 11120.0 nM|= 1.6 nM|= 56.0 nM|= 2600.0 nM|= 1800.0 nM|= 3910.0 nM|< 100.0 nM|= 80.0 nM|< 1000.0 nM|< 10.0 nM|= 6.427 nM|= 26.0 nM|= 3.3 nM|< 0.024 ug.mL-1|= 65.1 nM|= 0.5 nM|= 0.6 nM|<= 100.0 nM|= 6000.0 nM|< 1.8 nM|= 71300.0 nM|= 30.0 nM|= 87.5 nM|= 28660.0 nM|= 73.0 nM|= 13620.0 nM|= 340.0 nM|= 160.0 nM|= 420.0 nM|= 680.0 nM|= 84.0 nM|= 1670.0 nM|= 2500.0 nM|= 18600.0 nM|= 560.0 nM|= 2800.0 nM|= 21.0 nM|= 350.0 nM | | | NPASS |
| MDA-MB-157 | Homo sapiens | | | = 20.0 nM|= 7.569 nM | | | NPASS |
| MDA-MB-175-VII | Homo sapiens | | | = 83.02 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 291.0 nM|= 4160.0 nM|= 1100.0 nM|= 920.0 nM|= 680.0 nM|= 300.0 nM|= 4200.0 nM|= 330.0 nM|= 970.0 nM|= 2700.0 nM|< 10.0 nM|= 229.98 nM|= 162.0 nM|= 342.0 nM|= 2110.0 nM|= 5770.0 nM|= 307.0 nM|= 540.0 nM|= 16440.0 nM|= 0.32 nM|= 28.4 nM|= 23980.0 nM|= 8830.0 nM|= 264.0 nM|> 6400.0 nM|= 420.0 nM|= 1060.0 nM|= 490.0 nM|= 241.0 nM|> 100000.0 nM|= 170.0 nM | | | NPASS |
| MDA-MB-361 | Homo sapiens | | | = 170.0 nM|= 34.43 nM | | | NPASS |
| MDA-MB-415 | Homo sapiens | | | = 134.42 nM | | | NPASS |
| MDA-MB-435 | Homo sapiens | | | = 15.0 nM|= 375.0 nM|= 710.0 nM|= 43.6 nM|< 1.0 nM|= 1000.0 nM|= 2700.0 nM|= 310.0 nM | | | NPASS |
| MDA-MB-436 | Homo sapiens | | | = 31860.0 nM | | | NPASS |
| MDA-MB-453 | Homo sapiens | | | < 10.0 nM|= 6.965 nM | | | NPASS |
| MDA-MB-468 | Homo sapiens | | | = 14760.0 nM|= 1710.0 nM | | | NPASS |
| ME-180 | Homo sapiens | | | = 2.692 nM | | | NPASS |
| MEF | Mus musculus | | | = 5.87 ug.mL-1 | | | NPASS |
| MEG-01 | Homo sapiens | | | = 39.51 nM | | | NPASS |
| MEL-HO | Homo sapiens | | | = 7.628 nM | | | NPASS |
| MEL-JUSO | Homo sapiens | | | = 35.62 nM | | | NPASS |
| MFE-280 | Homo sapiens | | | = 21.56 nM | | | NPASS |
| MC116 | Homo sapiens | | | = 15.86 nM | | | NPASS |
| MFE-296 | Homo sapiens | | | < 1000.0 nM | | | NPASS |
| P30-OHK | Homo sapiens | | | = 2.792 nM | | | NPASS |
| M059J | Homo sapiens | | | = 4.095 nM|= 5500.0 nM | | | NPASS |
| LNCaP-Clone-FGC | Homo sapiens | | | = 31.03 nM | | | NPASS |
| LOX IMVI | Homo sapiens | | | = 48.0 nM|= 3.72 nM | | | NPASS |
| LS-1034 | Homo sapiens | | | = 9492.4 nM | | | NPASS |
| LS-123 | Homo sapiens | | | = 7325.59 nM | | | NPASS |
| LS-411N | Homo sapiens | | | = 58.08 nM | | | NPASS |
| LS-513 | Homo sapiens | | | = 19.37 nM | | | NPASS |
| LU-134-A | Homo sapiens | | | = 0.5865 nM | | | NPASS |
| LU-135 | Homo sapiens | | | = 28.16 nM | | | NPASS |
| LU-139 | Homo sapiens | | | = 16.44 nM | | | NPASS |
| LU-99A | Homo sapiens | | | = 3.854 nM | | | NPASS |
| LX-1 | Homo sapiens | | | = 120.0 nM | | | NPASS |
| LXF-289 cell line | | | | = 7.054 nM | | | NPASS |
| Leishmania donovani | Leishmadonovani | | = 7840.0 nM|= 3794.0 nM|= 12820.0 nM|= 6582.0 nM | | | | NPASS |
| Leishmania infantum | Leishmaitum | | | = 34400.0 nM|= 1120.0 nM | | | NPASS |
| Lewis lung carcinoma cell line | | | | = 33.0 nM | | | NPASS |
| LoVo | Homo sapiens | | | = 3100.0 nM|= 14.93 nM|= 0.32 nM|= 1540.0 nM | | | NPASS |
| Lu-65 | Homo sapiens | | | = 276.33 nM | | | NPASS |
| Lu-99 cell line | | | | = 0.001 ug.mL-1 | | | NPASS |
| Lu1 | Homo sapiens | | | = 28.7 nM | | | NPASS |
| M14 | Homo sapiens | | | = 9.948 nM | | | NPASS |
| NCI-H1048 | Homo sapiens | | | = 0.5292 nM | | | NPASS |
| MFH-ino | Homo sapiens | | | = 27.08 nM | | | NPASS |
| MG-63 | Homo sapiens | | | = 7.654 nM | | | NPASS |
| MX1 | Homo sapiens | | | = 1700.0 nM | | | NPASS |
| MZ1-PC | Homo sapiens | | | = 20.33 nM | | | NPASS |
| MZ2-MEL | Homo sapiens | | | = 14.11 nM | | | NPASS |
| MZ7-mel | Homo sapiens | | | = 8.612 nM | | | NPASS |
| Macrophage | Mus musculus | | = 18320.0 nM | | | | NPASS |
| MeWo | Homo sapiens | | | = 46.97 nM | | | NPASS |
| Melanoma-associated antigen E1 | | Q9HCI5 | | >55182 nM | | | BindingDB |
| Mo | Homo sapiens | | | = 111.97 nM | | | NPASS |
| Multidrug resistance-associated protein 4 | Homo sapiens | O15439 | | = 7400.0 nM | | | NPASS |
| NB-4 | Homo sapiens | | | = 2010.0 nM | | | NPASS |
| NB10 | Homo sapiens | | | = 0.6143 nM | | | NPASS |
| NB12 | Homo sapiens | | | = 44.02 nM | | | NPASS |
| NB13 | Homo sapiens | | | = 28.8 nM | | | NPASS |
| NB14 | Homo sapiens | | | = 0.9071 nM | | | NPASS |
| NB17 | Homo sapiens | | | = 2.175 nM | | | NPASS |
| NB5 | Homo sapiens | | | = 1.925 nM | | | NPASS |
| NB6 | Homo sapiens | | | = 182.71 nM | | | NPASS |
| NB69 | Homo sapiens | | | = 0.5694 nM | | | NPASS |
| NB7 | Homo sapiens | | | = 16.8 nM | | | NPASS |
| MV4-11 | Homo sapiens | | | = 0.7058 nM | | | NPASS |
| MFM-223 | Homo sapiens | | | = 5270.72 nM | | | NPASS |
| MT4 | Homo sapiens | | | = 4.0 nM | | | NPASS |
| MS-1 | Homo sapiens | | | = 2.774 nM | | | NPASS |
| MGC-803 | Homo sapiens | | | = 9450.0 nM|= 2960.0 nM|= 4270.0 nM|> 150000.0 nM|= 17760.0 nM | | | NPASS |
| MHCC97H | Homo sapiens | | | = 0.32 nM | | | NPASS |
| MHH-ES-1 | Homo sapiens | | | = 0.1293 nM | | | NPASS |
| MHH-NB-11 | Homo sapiens | | | = 0.8418 nM | | | NPASS |
| MHH-PREB-1 | Homo sapiens | | | = 2.733 nM | | | NPASS |
| MIA PaCa-2 | Homo sapiens | | | = 400.0 nM|= 2.759 nM|= 190.0 nM|= 180.0 nM | | | NPASS |
| MKN-1 | Homo sapiens | | | = 37.91 nM | | | NPASS |
| MKN-28 | Homo sapiens | | | = 51.21 nM | | | NPASS |
| MKN-45 | Homo sapiens | | | = 17.0 nM|= 27.5 nM | | | NPASS |
| MKN-7 | Homo sapiens | | | = 144.23 nM | | | NPASS |
| ML-2 | Homo sapiens | | | = 2.165 nM | | | NPASS |
| MLMA | Homo sapiens | | | = 8.145 nM | | | NPASS |
| MMAC-SF | Homo sapiens | | | = 38.4 nM | | | NPASS |
| MN-60 | Homo sapiens | | | = 5.083 nM | | | NPASS |
| MOLT-13 | Homo sapiens | | | = 1.787 nM | | | NPASS |
| MOLT-16 | Homo sapiens | | | = 0.7318 nM | | | NPASS |
| MOLT-4 | Homo sapiens | | | = 1.616 nM|= 0.04 nM | | | NPASS |
| MPP-89 | Homo sapiens | | | = 27.24 nM | | | NPASS |
| MRC5 | Homo sapiens | | | = 890.0 nM|= 1700.0 nM|= 800.0 nM|= 1.7 10^-5 uM|= 9020.0 nM | | | NPASS |
| MSTO-211H | Homo sapiens | | | = 8.238 nM | | | NPASS |
| P388 | Mus musculus | | | = 32.0 nM|= 0.005 ug.mL-1|= 0.00474 ug.mL-1|= 7.0 nM|= 13.0 nM|= 10.0 nM|= 32.1 nM|= 0.004 nM|= 9.0 nM|> 10000.0 nM|= 4.0 nM|= 14.0 nM | | | NPASS |
| SK-MEL-30 | Homo sapiens | | | = 2281.97 nM | | | NPASS |
| PA-1 | Homo sapiens | | | = 0.981 nM | | | NPASS |
| SiHa | Homo sapiens | | | = 86.88 nM | | | NPASS |
| Somatostatin receptor | Homo sapiens | P32745 | | = 2.21 nM | | | NPASS |
| Somatostatin receptor type 1/2/3/4/5 | Homo sapiens | P30872|P30874|P31391|P32745|P35346 | | 2.2 nM | | | BindingDB |
| T-24 | Homo sapiens | | | = 88.0 nM|= 6.0 nM|= 1.614 nM|= 6800.0 nM|= 3090.0 nM | | | NPASS |
| T47D | Homo sapiens | | | = 207.0 nM|= 9170.0 nM|< 1000.0 nM|< 10.0 nM|= 1530.0 nM|= 13.52 nM|= 70.0 nM|= 300.0 nM|= 280.0 nM|= 750.0 nM|= 1840.0 nM|= 310.0 nM|= 80.0 nM|= 1620.0 nM|= 11170.0 nM|= 4100.0 nM|= 2100.0 nM|= 2310.0 nM|= 490.0 nM|= 250.0 nM|= 3670.0 nM|= 90.0 nM | | | NPASS |
| T84 | Homo sapiens | | | = 4602.33 nM | | | NPASS |
| T98G | Homo sapiens | | | = 27.15 nM | | | NPASS |
| TCC-SUP | Homo sapiens | | | = 39.04 nM | | | NPASS |
| TE-1 | Homo sapiens | | | = 35.11 nM | | | NPASS |
| TE-10 | Homo sapiens | | | = 147.61 nM | | | NPASS |
| TE-11 | Homo sapiens | | | = 16.33 nM | | | NPASS |
| TE-12 | Homo sapiens | | | = 265.25 nM | | | NPASS |
| TE-5 | Homo sapiens | | | = 7.38 nM | | | NPASS |
| TE-6 | Homo sapiens | | | = 178.5 nM | | | NPASS |
| TE-8 | Homo sapiens | | | = 4.17 nM | | | NPASS |
| TE-9 | Homo sapiens | | | = 23.65 nM | | | NPASS |
| TERT-RPE1 | Homo sapiens | | | > 40000.0 nM|= 27200.0 nM | | | NPASS |
| TGBC11TKB | Homo sapiens | | | = 12.24 nM | | | NPASS |
| TGBC1TKB | Homo sapiens | | | = 109.97 nM | | | NPASS |
| Serotonin 2b (5-HT2b) receptor | Homo sapiens | P41595 | | = 970.0 nM | | = 617.0 nM | NPASS |
| TGBC24TKB | Homo sapiens | | | = 53.71 nM | | | NPASS |
| Serine/threonine-protein kinase Chk1 | Homo sapiens | O14757 | 2.1 nM|= 2.1 nM | | | | BindingDB, NPASS |
| SW982 | Homo sapiens | | | = 4.062 nM | | | NPASS |
| SW-620 | Homo sapiens | | = 1.2 nM|= 0.15 nM | = 4.082 nM | | | NPASS |
| SW1088 | Homo sapiens | | | = 27.77 nM | | | NPASS |
| SW13 | Homo sapiens | | | = 2.993 nM | | | NPASS |
| SW1417 | Homo sapiens | | | = 52.7 nM | | | NPASS |
| SW1463 | Homo sapiens | | | = 51.69 nM | | | NPASS |
| SW1573 | Homo sapiens | | | = 2.348 nM | | | NPASS |
| SW1710 | Homo sapiens | | | = 33.57 nM | | | NPASS |
| SW1783 | Homo sapiens | | | = 24.57 nM | | | NPASS |
| SW1990 | Homo sapiens | | | = 37.88 nM|= 200.0 nM | | | NPASS |
| SW48 | Homo sapiens | | | = 3.017 nM | | | NPASS |
| SW480 | Homo sapiens | | | = 0.01 ug.mL-1|= 290.0 nM|= 210.0 nM | | | NPASS |
| SW626 | Homo sapiens | | | = 28.7 nM|= 76.9 nM | | | NPASS |
| SW684 | Homo sapiens | | | = 711.49 nM | | | NPASS |
| SW756 | Homo sapiens | | | = 4.211 nM | | | NPASS |
| SW780 | Homo sapiens | | | = 25.78 nM | | | NPASS |
| SW837 | Homo sapiens | | | = 48.92 nM | | | NPASS |
| SW872 | Homo sapiens | | | = 24.16 nM | | | NPASS |
| SW900 | Homo sapiens | | | = 31.84 nM | | | NPASS |
| SW948 | Homo sapiens | | | = 160.0 nM|= 260.2 nM | | | NPASS |
| Saccharomyces cerevisiae | Saccharomyces cerevisiae | | | > 200000.0 nM|= 0.16 ug.mL-1|= 0.014 ug.mL-1|> 100.0 ug.mL-1|= 0.18 ug.mL-1|= 0.06 ug.mL-1 | | | NPASS |
| SW 962 | Homo sapiens | | | = 20.51 nM | | | NPASS |
| THP-1 | Homo sapiens | | = 160.0 nM | = 600.0 nM|= 71.0 nM|= 1890.0 nM | | | NPASS |
| TK-10 | Homo sapiens | | | = 55.79 nM | | | NPASS |
| UACC-893 | Homo sapiens | | | = 383.65 nM | | | NPASS |
| UMC-11 | Homo sapiens | | | = 2511.11 nM | | | NPASS |
| UMUC3 | Homo sapiens | | | = 3.093 nM | | | NPASS |
| UO-31 | Homo sapiens | | | = 34.07 nM | | | NPASS |
| VA-ES-BJ | Homo sapiens | | | = 3.469 nM | | | NPASS |
| VM-CUB-1 | Homo sapiens | | | = 2.21 nM | | | NPASS |
| VMRC-RCZ | Homo sapiens | | | = 47.35 nM | | | NPASS |
| Vero | Chlorocebus aethiops | | | = 0.054 ug.mL-1|= 0.02 ug.mL-1|= 0.6 ug.mL-1|= 58.0 ug.mL-1 | | | NPASS |
| WI-38 | Homo sapiens | | | = 0.4 ug.mL-1|= 0.03 ug.mL-1|= 30.0 nM|= 8370.0 nM | | | NPASS |
| WIL2-NS | Homo sapiens | | | = 5.0 nM | | | NPASS |
| WM-115 | Homo sapiens | | | = 102.32 nM | | | NPASS |
| WiDr | Homo sapiens | | | = 17.0 nM|= 0.07 ug.mL-1 | | | NPASS |
| YAPC | Homo sapiens | | | = 29.6 nM | | | NPASS |
| YH-13 | Homo sapiens | | | = 11.65 nM | | | NPASS |
| YKG-1 | Homo sapiens | | | = 5.453 nM | | | NPASS |
| ZR-75-1 | Homo sapiens | | | < 10.0 nM | | | NPASS |
| ZR-75-30 | Homo sapiens | | | = 261.0 nM|= 240.0 nM | | | NPASS |
| no-10 | Homo sapiens | | | = 174.04 nM | | | NPASS |
| no-11 | Homo sapiens | | | = 113.08 nM | | | NPASS |
| UACC-62 | Homo sapiens | | | = 31.03 nM | | | NPASS |
| TI-73 | Homo sapiens | | | = 14.55 nM | | | NPASS |
| UACC-257 | Homo sapiens | | | = 115.96 nM | | | NPASS |
| U-937 | Homo sapiens | | | = 680.0 nM|= 32.0 nM|= 15.0 nM|= 300.0 nM|= 1980.0 nM|= 18240.0 nM|= 1810.0 nM | | | NPASS |
| TYK-nu | Homo sapiens | | | = 4.94 nM | | | NPASS |
| Telomerase reverse transcriptase | Homo sapiens | O14746 | | >300000 nM|> 300000.0 nM | | | BindingDB, NPASS |
| Topoisomerase I subunit B | Leishmamajor | | 670 nM | | | | BindingDB |
| Type II restriction enzyme BamHI | Bacillus amyloliquefaciens | P23940 | | >300000 nM | | | BindingDB |
| Type II restriction enzyme EcoRI | Escherichia coli | P00642 | | >300000 nM | | | BindingDB |
| Type II restriction enzyme HindIII | Haemophilus influe (strain ATCC 51907 / DSM 11121 / KW20 / Rd) | P43870 | | >300000 nM | | | BindingDB |
| Type II restriction enzyme PstI | Providencia stuartii | P00640 | | >300000 nM | | | BindingDB |
| Type II restriction enzyme ScaI | Streptomyces caespitosus | O52691 | | >300000 nM | | | BindingDB |
| Type-2 restriction enzyme BamHI | Bacillus amyloliquefaciens | P23940 | | > 300000.0 nM | | | NPASS |
| Type-2 restriction enzyme EcoRI | Escherichia coli | P00642 | | > 300000.0 nM | | | NPASS |
| Type-2 restriction enzyme HindIII | Haemophilus influe (strain ATCC 51907 / DSM 11121 / KW20 / Rd) | P43870 | | > 300000.0 nM | | | NPASS |
| Type-2 restriction enzyme PstI | Providencia stuartii | P00640 | | > 300000.0 nM | | | NPASS |
| Type-2 restriction enzyme ScaI | Streptomyces caespitosus | O52691 | | > 300000.0 nM | | | NPASS |
| Tyrosyl-DNA phosphodiesterase 1 | Homo sapiens | Q9NUW8 | | >111000 nM|> 111000.0 nM|= 0.0 nM | | | BindingDB, NPASS |
| Tyrosyl-DNA phosphodiesterase 2 | Homo sapiens | O95551 | | >111000 nM|> 111000.0 nM|= 0.0 nM | | | BindingDB, NPASS |
| U-118-MG | Homo sapiens | | | = 19.0 nM | | | NPASS |
| U-251 | Homo sapiens | | | = 1.869 nM | | | NPASS |
| U-266 | Homo sapiens | | | = 69.51 nM | | | NPASS |
| U-87 MG | Homo sapiens | | | = 6.632 nM|< 1850.0 nM | | | NPASS |
| U2OS | Homo sapiens | | | = 13.54 nM | | | NPASS |
| P388CPT5 | Mus musculus | | | = 2800.0 nM | | | NPASS |
| SW 954 | Homo sapiens | | | = 20.35 nM | | | NPASS |
| SU-DHL-2 | Homo sapiens | | | = 940.0 nM | | | NPASS |
| RPMI 8402 | Homo sapiens | | | = 5.0 nM|= 6.0 nM|> 10000.0 nM | | | NPASS |
| RPMI-2650 | Homo sapiens | | | = 2.217 nM | | | NPASS |
| RPMI-7951 | Homo sapiens | | | = 4.753 nM|= 220.0 nM | | | NPASS |
| RPMI-8226 | Homo sapiens | | | = 6.0 nM|= 29.49 nM|= 2.05 ug.mL-1 | | | NPASS |
| RPMI-8866 | Homo sapiens | | | = 1.725 nM | | | NPASS |
| RS4-11 | Homo sapiens | | | = 0.9022 nM | | | NPASS |
| RT-112 | Homo sapiens | | | = 14.88 nM | | | NPASS |
| RVH-421 | Homo sapiens | | | = 71.47 nM | | | NPASS |
| RXF 393 | Homo sapiens | | | = 4.662 nM | | | NPASS |
| Raji | Homo sapiens | | | = 1000.0 nM|= 3270.0 nM | | | NPASS |
| Ramos-2G6-4C10 | Homo sapiens | | | = 10.51 nM | | | NPASS |
| Renca | Mus musculus | | | = 304.0 nM | | | NPASS |
| Reverse transcriptase | Human immunodeficiency virus 1 | | | >574000 nM | | | BindingDB |
| Ribonuclease pancreatic | Bos taurus | P61823 | | >300000 nM|> 300000.0 nM | | | BindingDB, NPASS |
| S-117 | Homo sapiens | | | = 78.15 nM | | | NPASS |
| SAOS-2 | Homo sapiens | | | = 17.77 nM | | | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM | | | NPASS |
| SAS | Homo sapiens | | | = 1.241 nM|= 6000.0 nM | | | NPASS |
| SBC-1 | Homo sapiens | | | = 27.79 nM | | | NPASS |
| RO82-W-1 | Homo sapiens | | | = 14.91 nM | | | NPASS |
| SBC-5 | Homo sapiens | | | = 32.15 nM | | | NPASS |
| RMG-I | Homo sapiens | | | = 244.5 nM | | | NPASS |
| RH-18 | Homo sapiens | | | = 389.64 nM | | | NPASS |
| PANC-03-27 | Homo sapiens | | | = 7.103 nM | | | NPASS |
| PANC-08-13 | Homo sapiens | | | = 44.89 nM | | | NPASS |
| PANC-1 | Homo sapiens | | | = 180.0 nM|= 90.0 nM | | | NPASS |
| PBMC | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| PC-14 | Homo sapiens | | | = 13.58 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 57.0 nM|= 310.0 nM|= 1414.4 nM|= 52.0 nM|= 1400.0 nM|= 16240.0 nM|= 30.0 nM|= 12.0 nM|= 9.753 nM|= 78.0 nM|= 1200.0 nM|= 10.0 nM|= 2500.0 nM|= 100.0 nM|= 6960.0 nM|= 400.0 nM|> 40000.0 nM|= 18240.0 nM|= 2400.0 nM | | | NPASS |
| PC-3M | Homo sapiens | | | = 480.0 nM|= 190.0 nM | | | NPASS |
| PFSK-1 | Homo sapiens | | | = 26.03 nM | | | NPASS |
| PSN1 | Homo sapiens | | | = 3.069 nM | | | NPASS |
| Panc1005 | Homo sapiens | | | = 19.68 nM | | | NPASS |
| Panel (56 tumour cell lines) | | | | = 40.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 0.83 nM|= 1.41 nM|= 1.12 nM|= 1.32 nM|= 0.89 nM|= 0.56 nM|= 794.33 nM|= 1258.93 nM|= 1000.0 nM|= 501.19 nM | | | NPASS |
| QG-56 | | | | = 0.00463 ug.mL-1 | | | NPASS |
| QIMR-WIL | Homo sapiens | | | = 0.7753 nM | | | NPASS |
| RCC10RGB | Homo sapiens | | | = 113.62 nM | | | NPASS |
| RCM-1 | Homo sapiens | | | = 28.66 nM | | | NPASS |
| RD | Homo sapiens | | | = 15.74 nM|= 4490.0 nM|= 1240.0 nM|= 1720.0 nM | | | NPASS |
| RERF-LC-MS | Homo sapiens | | | = 22.87 nM | | | NPASS |
| RH-1 | Homo sapiens | | | = 3.86 nM | | | NPASS |
| RKO | Homo sapiens | | | = 4.23 nM|< 1850.0 nM|= 61.7 nM | | | NPASS |
| SW 1116 | Homo sapiens | | | = 190.35 nM | | | NPASS |
| SCC-15 | Homo sapiens | | | = 18.57 nM | | | NPASS |
| SCC-4 | Homo sapiens | | | = 19.26 nM | | | NPASS |
| SK-N-AS | Homo sapiens | | | = 5.377 nM | | | NPASS |
| SK-N-DZ | Homo sapiens | | | = 21.69 nM | | | NPASS |
| SK-N-FI | Homo sapiens | | | = 106.62 nM | | | NPASS |
| SK-NEP-1 | Homo sapiens | | | = 1.227 nM | | | NPASS |
| SK-OV-3 | Homo sapiens | | | = 37.0 nM|= 20.0 nM|= 51.0 nM|= 14.0 nM|= 1.54 ug.mL-1|= 2544.0 nM|= 7210.91 nM|= 5.5 nM|= 5500.0 nM|= 3820.0 nM|= 2560.0 nM|= 4860.0 nM | | | NPASS |
| SK-PN-DW | Homo sapiens | | | = 1.16 nM | | | NPASS |
| SK-UT-1 | Homo sapiens | | | = 3.067 nM | | | NPASS |
| SK-VLB | Homo sapiens | | | = 41.0 nM|= 53.0 nM | | | NPASS |
| SKG-IIIa | Homo sapiens | | | = 4.582 nM | | | NPASS |
| SMMC-7721 | Homo sapiens | | | = 20.0 nM|= 3.0 nM|= 1080.0 nM|= 450.0 nM|> 10000.0 nM|= 3950.0 nM | | | NPASS |
| SN12C | Homo sapiens | | | = 4.503 nM | | | NPASS |
| SNB-75 | Homo sapiens | | | = 17.34 nM | | | NPASS |
| SNU-387 | Homo sapiens | | | = 256.33 nM | | | NPASS |
| SNU-423 | Homo sapiens | | | = 128.79 nM | | | NPASS |
| SNU-449 | Homo sapiens | | | = 194.29 nM | | | NPASS |
| SNU-5 | Homo sapiens | | | = 42.71 nM | | | NPASS |
| SNU-638 | Homo sapiens | | | = 98.0 nM|= 280.0 nM | | | NPASS |
| SNU-C2B | Homo sapiens | | | = 35.38 nM | | | NPASS |
| SNU1 | Homo sapiens | | | = 1.088 nM | | | NPASS |
| SK-MES-1 | Homo sapiens | | | = 10.0 nM|= 10.78 nM | | | NPASS |
| SCC-25 | Homo sapiens | | | = 56.73 nM | | | NPASS |
| SK-MEL3 | Homo sapiens | | | = 329.41 nM | | | NPASS |
| SK-MEL-28 | Homo sapiens | | | = 40.0 nM|= 17.13 nM|< 10.0 nM|= 2260.0 nM | | | NPASS |
| SCC-9 | Homo sapiens | | | = 33.19 nM | | | NPASS |
| SCH | Homo sapiens | | | = 628.09 nM | | | NPASS |
| SF-126 | Homo sapiens | | | = 2.835 nM | | | NPASS |
| SF-268 | Homo sapiens | | = 59.0 nM | = 40.0 nM|= 190.0 nM|= 70.0 nM|= 3.379 nM | | | NPASS |
| SF-295 | Homo sapiens | | | = 7.909 nM | | | NPASS |
| SF-539 | Homo sapiens | | | = 9.009 nM | | | NPASS |
| SGC-7901 | Homo sapiens | | | < 1850.0 nM|= 5800.0 nM | | | NPASS |
| SH-4 | Homo sapiens | | | = 59.8 nM | | | NPASS |
| SH-SY5Y | Homo sapiens | | | = 610.0 nM | | | NPASS |
| SHP77 | Homo sapiens | | | = 1543.63 nM | | | NPASS |
| SJRH30 | Homo sapiens | | | = 298.06 nM | | | NPASS |
| SJSA-1 | Homo sapiens | | | = 18.0 nM | | | NPASS |
| SK-BR-3 | Homo sapiens | | | = 20.0 nM|< 10.0 nM|= 210.0 nM | | | NPASS |
| SK-HEP1 | Homo sapiens | | | = 7.253 nM|= 900.0 nM | | | NPASS |
| SK-LMS-1 | Homo sapiens | | | = 180.87 nM | | | NPASS |
| SK-LU-1 | Homo sapiens | | | = 4.713 nM | | | NPASS |
| SK-MEL-1 | Homo sapiens | | | = 51.29 nM | | | NPASS |
| SK-MEL-2 | Homo sapiens | | | = 75.0 nM|= 165.0 nM|= 6.88 ug.mL-1|= 7860.0 nM|= 54.75 nM | | | NPASS |
| SK-MEL-24 | Homo sapiens | | | = 38.51 nM|= 460.0 nM | | | NPASS |
| LNCaP | Homo sapiens | | | = 86.1 nM | | | NPASS |
| LN-405 | Homo sapiens | | | = 517.64 nM | | | NPASS |
| LB2518-MEL | Homo sapiens | | | = 87.25 nM | | | NPASS |
| LK-2 | Homo sapiens | | | = 35.53 nM | | | NPASS |
| CWR22R | Homo sapiens | | | = 9.314 nM | | | NPASS |
| Ca-Ski | Homo sapiens | | | = 4.97 nM|= 1800.0 nM | | | NPASS |
| Ca9-22 | Homo sapiens | | | = 2.211 nM | | | NPASS |
| CaR-1 | Homo sapiens | | | = 6.427 nM | | | NPASS |
| Caco-2 | Homo sapiens | | | = 9550.0 nM | | | NPASS |
| Calu-3 | Homo sapiens | | | = 32.8 nM | | | NPASS |
| Calu-6 | Homo sapiens | | | = 178.95 nM | | | NPASS |
| LN-229 | Homo sapiens | | | = 0.32 nM | | | NPASS |
| Canalicular multispecific organic anion transporter 2 | Homo sapiens | O15438 | | > 133000.0 nM | | | NPASS |
| Caov-3 cell line | | | | = 2900000.0 nM|= 30.0 nM | | | NPASS |
| Capan-2 | Homo sapiens | | | = 452.29 nM | | | NPASS |
| ChaGo-K-1 | Homo sapiens | | | = 304.67 nM | | | NPASS |
| Col2 | Homo sapiens | | | = 45.0 nM | | | NPASS |
| Cystic fibrosis transmembrane conductance regulator | Human | P13569 | >50000 nM | | | | BindingDB |
| D-247MG | Homo sapiens | | | = 39.54 nM | | | NPASS |
| D-263MG | Homo sapiens | | | = 9.114 nM | | | NPASS |
| D-336MG | Homo sapiens | | | = 5.205 nM | | | NPASS |
| D-392MG | Homo sapiens | | | = 17.73 nM | | | NPASS |
| D-423MG | Homo sapiens | | | = 2.551 nM | | | NPASS |
| CW-2 | Homo sapiens | | | = 35.45 nM | | | NPASS |
| D-502MG | Homo sapiens | | | = 22.59 nM | | | NPASS |
| CTV-1 | Homo sapiens | | | = 0.9054 nM | | | NPASS |
| CT26.WT | Mus musculus | | | = 430.0 nM | | | NPASS |
| CNE-2 | Homo sapiens | | | = 100.0 nM|= 980.0 nM | | | NPASS |
| COLO 205 | Homo sapiens | | | = 5.4 nM|= 50.0 nM | | | NPASS |
| COLO-320-HSR | Homo sapiens | | | = 62.09 nM | | | NPASS |
| COLO-668 | Homo sapiens | | | = 22.32 nM | | | NPASS |
| COLO-678 | Homo sapiens | | | = 3682.73 nM | | | NPASS |
| COLO-679 | Homo sapiens | | | = 4791.52 nM | | | NPASS |
| COLO-680N | Homo sapiens | | | = 72.45 nM | | | NPASS |
| COLO-684 | Homo sapiens | | | = 13.82 nM | | | NPASS |
| COLO-741 | Homo sapiens | | | = 109.27 nM | | | NPASS |
| COLO-792 | Homo sapiens | | | = 169.17 nM | | | NPASS |
| COLO-800 | Homo sapiens | | | = 0.4281 nM | | | NPASS |
| COLO-824 | Homo sapiens | | | = 269.5 nM | | | NPASS |
| COLO-829 | Homo sapiens | | | = 11.67 nM | | | NPASS |
| COR-L105 | Homo sapiens | | | = 184.93 nM | | | NPASS |
| COR-L23 | Homo sapiens | | | = 6.849 nM | | | NPASS |
| COR-L88 | Homo sapiens | | | = 40.93 nM | | | NPASS |
| CP50-MEL-B | Homo sapiens | | | = 72.08 nM | | | NPASS |
| CP66-MEL | Homo sapiens | | | = 208.15 nM | | | NPASS |
| CT26 | Mus musculus | | | = 34.0 nM | | | NPASS |
| CTB-1 | Homo sapiens | | | = 0.4292 nM | | | NPASS |
| CNE | Homo sapiens | | | = 340.0 nM | | | NPASS |
| D-542MG | Homo sapiens | | | = 291.41 nM | | | NPASS |
| D283 Med | | | | = 3.198 nM | | | NPASS |
| DNA topoisomerase type IB small subunit | Leishmamajor | Q95Z89 | = 670.0 nM | | | | NPASS |
| DOHH-2 | Homo sapiens | | | = 0.6022 nM | | | NPASS |
| DOK | Homo sapiens | | | = 18.92 nM | | | NPASS |
| DSH1 | Homo sapiens | | | = 15.75 nM | | | NPASS |
| DU-145 | Homo sapiens | | | = 10.0 nM|= 3200.0 nM|= 1460.0 nM|= 3570.0 nM|= 940.0 nM|= 660.0 nM|= 1000.0 nM|= 400.0 nM|= 20.0 nM|= 610.0 nM|= 310.0 nM|= 2370.0 nM|= 15.0 nM|= 9290.0 nM|= 1060.0 nM|= 28.7 nM|= 2281.94 nM|= 390.0 nM|= 800.0 nM|= 4010.0 nM|= 110.0 nM|= 950.0 nM|= 29.0 nM|= 100.0 nM|= 50.0 nM|= 16.0 nM|= 1990.0 nM|= 70.0 nM|= 33.45 nM|= 210.0 nM | | | NPASS |
| DU-4475 | Homo sapiens | | | = 3.067 nM | | | NPASS |
| Daoy | Homo sapiens | | | = 0.4809 nM | | | NPASS |
| Deoxyribonuclease-1 | Bos taurus | P00639 | | >300000 nM|> 300000.0 nM | | | BindingDB, NPASS |
| Deoxyribonuclease-2-alpha | Sus scrofa | O62855 | | >300000 nM|> 300000.0 nM | | | BindingDB, NPASS |
| Detroit 551 | Homo sapiens | | | = 990.0 nM | | | NPASS |
| Detroit562 | Homo sapiens | | | = 13.34 nM | | | NPASS |
| DoTc2-4510 | Homo sapiens | | | = 4.032 nM | | | NPASS |
| EC-GI-10 | Homo sapiens | | | = 7.904 nM | | | NPASS |
| ECC10 | Homo sapiens | | | = 3.853 nM | | | NPASS |
| EFM-19 | Homo sapiens | | | = 126.89 nM | | | NPASS |
| EFO-21 | Homo sapiens | | | = 20.32 nM | | | NPASS |
| EFO-27 | Homo sapiens | | | = 80.99 nM | | | NPASS |
| EGI-1 | Homo sapiens | | | = 25.07 nM | | | NPASS |
| EKVX | Homo sapiens | | | = 436.37 nM | | | NPASS |
| DNA topoisomerase II alpha | Homo sapiens | P11388 | | > 300000.0 nM | | | NPASS |
| D-566MG | Homo sapiens | | | = 0.1315 nM | | | NPASS |
| DNA topoisomerase I | Mus musculus | Q04750 | | = 40000.0 nM|= 12000.0 nM | | | NPASS |
| DNA topoisomerase I | Homo sapiens | P11387 | = 350.0 nM | = 700.0 nM|= 679.0 nM|= 127000.0 nM|= 680.0 nM|= 300.0 nM|= 4000.0 nM|= 17000.0 nM|= 9000.0 nM|= 20000.0 nM|= 2200.0 nM|= 3750.0 nM|= 4950.0 nM|= 4750.0 nM|= 25.0 nM|= 2500.0 nM|= 27000.0 nM|= 62900.0 nM|= 62000.0 nM|= 224.0 nM|= 2430.0 nM | | | NPASS |
| DB | Homo sapiens | | | = 1.161 nM | | | NPASS |
| DBTRG-05MG | Homo sapiens | | | = 40.86 nM | | | NPASS |
| DC3F | Cricetulus griseus | | | = 6.0 nM | | | NPASS |
| DEL | Homo sapiens | | | = 0.8157 nM | | | NPASS |
| DJM-1 | Homo sapiens | | | = 436.47 nM | | | NPASS |
| DK-MG | Homo sapiens | | | = 84.75 nM | | | NPASS |
| DLD-1 | Homo sapiens | | | = 14000000.0 nM|= 210.0 nM | | | NPASS |
| DMS-114 | Homo sapiens | | | = 81.1 nM | | | NPASS |
| DMS-273 | Homo sapiens | | | = 6.072 nM | | | NPASS |
| DMS-79 | Homo sapiens | | | = 31.85 nM | | | NPASS |
| DNA ligase | Enterobacteria phage T4 | P00970 | | >300000 nM|> 300000.0 nM | | | BindingDB, NPASS |
| DNA topoisomerase | Bos taurus | | | 17000 nM | | | BindingDB |
| DNA topoisomerase | Bos taurus | A0JN73 | | = 17000.0 nM | | | NPASS |
| DNA topoisomerase 1 | Chlorocebus aethiops | Q7YR26 | | 27000 nM|= 27000.0 nM | | | BindingDB, NPASS |
| DNA topoisomerase 1 | Homo sapiens | P11387 | 350 nM | 127000 nM|679 nM|1400 nM|4000 nM|17000 nM|9000 nM|700 nM|1600 nM|680 nM|300 nM|20000 nM|2200 nM|224 nM|4950 nM|4750 nM|3750 nM|2500 nM|25 nM|27000 nM|62900 nM|62 nM | | | BindingDB |
| DNA topoisomerase 1 | Human | P11387 | | 2.0e+4 nM | | | BindingDB |
| DNA topoisomerase 1 | Mus musculus | Q04750 | | 40000 nM|12000 nM | | | BindingDB |
| DNA topoisomerase 2-alpha | Homo sapiens | P11388 | | >300000 nM | | | BindingDB |
| DNA topoisomerase 2-alpha | Human | P11388 | | >3.50e+5 nM | | | BindingDB |
| DNA topoisomerase I | Leishmadonovani (strain BPK282A1) | E9BRC0 | | = 21920.0 nM|= 9200.0 nM | | | NPASS |
| EM-2 | Homo sapiens | | | = 4.08 nM | | | NPASS |
| CHP-212 | Homo sapiens | | | = 1.026 nM | | | NPASS |
| CGTH-W-1 | Homo sapiens | | | = 3.275 nM | | | NPASS |
| A498 | Homo sapiens | | | = 7.077 nM | | | NPASS |
| A549 | Homo sapiens | | | = 2530.0 nM|= 8.0 nM|= 330000.0 nM|= 14.0 nM|= 67.0 nM|= 69.0 nM|= 3120.0 nM|= 4.0 nM|= 10.0 nM|= 58.0 nM|= 3100.0 nM|= 47.0 nM|= 40.0 nM|= 5.379 nM|= 57.0 nM|= 30.0 nM|= 3600.0 nM|= 0.072 ug.mL-1|= 91.0 nM|= 260.0 nM|= 33.8 nM|= 2610.0 nM|= 15.8 nM|= 14.09 nM|= 99.0 nM|= 37050.0 nM|= 650.0 nM|< 10.0 nM|= 16.0 nM|= 1300.0 nM|= 1.0 nM|= 26450.0 nM|= 100.0 nM|= 1600.0 nM|= 350.0 nM|= 9.0 nM|= 240.0 nM|= 6.0 nM|= 8.63 nM|= 700.0 nM|= 13640.0 nM|< 1000.0 nM|= 5500.0 nM|= 8870.0 nM|= 5930.0 nM|= 2210.0 nM|= 1310.0 nM|= 4430.0 nM|= 0.32 nM|= 90.0 nM|= 2800.0 nM|= 3320.0 nM|= 39.0 nM|= 32110.0 nM|= 50880.0 nM|= 1560.0 nM|= 1000.0 nM|= 170.0 nM|= 8900.0 nM|= 470.0 nM|= 32100.0 nM|= 74.0 nM|= 370.0 nM|< 1850.0 nM | | | NPASS |
| A673 | Homo sapiens | | | = 0.8149 nM | | | NPASS |
| A704 | Homo sapiens | | | = 15.35 nM | | | NPASS |
| ABC-1 | Homo sapiens | | | = 3.468 nM | | | NPASS |
| ACHN | Homo sapiens | | | = 6.663 nM | | | NPASS |
| ACN | Homo sapiens | | | = 85.66 nM | | | NPASS |
| AGS | Homo sapiens | | | = 20.0 nM|= 16.13 nM|= 23760.0 nM | | | NPASS |
| ALL-PO | Homo sapiens | | | = 1.534 nM | | | NPASS |
| AM-38 | Homo sapiens | | | = 4.408 nM | | | NPASS |
| AN3-CA | Homo sapiens | | | = 33.98 nM | | | NPASS |
| ASPC1 | Homo sapiens | | | = 168.37 nM | | | NPASS |
| ATN-1 | Homo sapiens | | | = 2.043 nM | | | NPASS |
| ATP-binding cassette sub-family C member 2 | Homo sapiens | Q92887 | | >133000 nM | | | BindingDB |
| ATP-binding cassette sub-family C member 3 | Homo sapiens | O15438 | | >133000 nM | | | BindingDB |
| ATP-binding cassette sub-family C member 4 | Homo sapiens | O15439 | | 7400 nM | | | BindingDB |
| AU565 | Homo sapiens | | | = 3.68 nM | | | NPASS |
| BALL-1 | Homo sapiens | | | = 108.94 nM | | | NPASS |
| BB30-HNC | Homo sapiens | | | = 21.55 nM | | | NPASS |
| A4-Fuk | Homo sapiens | | | = 1.749 nM | | | NPASS |
| BB49-HNC | Homo sapiens | | | = 120.28 nM | | | NPASS |
| A388 | Homo sapiens | | | = 10.12 nM | | | NPASS |
| A2780 | Homo sapiens | | | = 7.0 nM|= 280.0 nM|= 4.0 nM|= 200.0 nM|= 0.07 ug.mL-1|= 300.0 nM|= 260.0 nM|= 2.902 nM|= 13.0 nM|= 900.0 nM|= 29.0 nM | | | NPASS |
| 23132-87 | Homo sapiens | | | = 19.46 nM | | | NPASS |
| 4T1 | Mus musculus | | | = 170.0 nM | | | NPASS |
| 5637 | Homo sapiens | | | = 4.183 nM | | | NPASS |
| 639-V | Homo sapiens | | | = 0.1714 nM | | | NPASS |
| 647-V | Homo sapiens | | | = 0.8964 nM | | | NPASS |
| 697 | Homo sapiens | | | = 2.029 nM | | | NPASS |
| 769-P | Homo sapiens | | | = 25.34 nM | | | NPASS |
| 786-0 | Homo sapiens | | | = 5.021 nM | | | NPASS |
| 8-MG-BA | Homo sapiens | | | = 1.502 nM | | | NPASS |
| 8305C | Homo sapiens | | | = 93.98 nM | | | NPASS |
| 833K | | | | = 10.0 nM | | | NPASS |
| 8505C | Homo sapiens | | | = 3.301 nM | | | NPASS |
| A-375 | Homo sapiens | | | = 3.688 nM|= 187.0 nM|= 13.0 nM|= 660.0 nM | | | NPASS |
| A-427 | Homo sapiens | | | = 24.0 nM|= 4.251 nM | | | NPASS |
| A-431 | Homo sapiens | | | = 11.0 nM|= 1552.36 nM | | | NPASS |
| A101D | Homo sapiens | | | = 257.84 nM | | | NPASS |
| A172 | Homo sapiens | | | = 140.0 nM|= 12.76 nM | | | NPASS |
| A204 | Homo sapiens | | | = 4.525 nM | | | NPASS |
| A2058 | Homo sapiens | | | = 3.599 nM | | | NPASS |
| A3-KAW | Homo sapiens | | | = 1.669 nM | | | NPASS |
| CHL-1 | Homo sapiens | | | = 6.091 nM | | | NPASS |
| BB65-RCC | Homo sapiens | | | = 1.853 nM | | | NPASS |
| BE-13 | Homo sapiens | | | = 4.564 nM | | | NPASS |
| CAKI-1 | Homo sapiens | | | = 5.354 nM | | | NPASS |
| CAKI-2 | Homo sapiens | | | = 3960.0 nM | | | NPASS |
| CAL-120 | Homo sapiens | | | = 594.73 nM | | | NPASS |
| CAL-12T | Homo sapiens | | | = 262.05 nM | | | NPASS |
| CAL-27 | Homo sapiens | | | = 2.018 nM | | | NPASS |
| CAL-33 | Homo sapiens | | | = 5.997 nM | | | NPASS |
| CAL-39 | Homo sapiens | | | = 19.16 nM | | | NPASS |
| CAL-51 | Homo sapiens | | | = 29.74 nM | | | NPASS |
| CAL-54 | Homo sapiens | | | = 4.758 nM | | | NPASS |
| CAL-62 | Homo sapiens | | | = 0.9836 nM | | | NPASS |
| CAL-72 | Homo sapiens | | | = 150.57 nM | | | NPASS |
| CAL-85-1 | Homo sapiens | | | = 7923.68 nM | | | NPASS |
| CAMA-1 | Homo sapiens | | | = 70.0 nM|= 87.43 nM | | | NPASS |
| CAPAN-1 | Homo sapiens | | | = 14.95 nM|= 210.0 nM | | | NPASS |
| CAS-1 | Homo sapiens | | | = 121.91 nM | | | NPASS |
| CCD 19Lu | Homo sapiens | | | = 2.0 ug.mL-1 | | | NPASS |
| CCRF-CEM | Homo sapiens | | | = 0.005 ug.mL-1|= 5300.0 nM|= 0.84 nM|= 3.0 nM|= 40.0 nM|= 5.0 nM|= 5.547 nM|= 80.0 nM|= 2.0 nM | | | NPASS |
| CCRF-SB | Homo sapiens | | | = 3.0 nM | | | NPASS |
| CFPAC-1 | Homo sapiens | | | = 14.75 nM | | | NPASS |
| CA46 | Homo sapiens | | | = 520.0 nM | | | NPASS |
| BCPAP | Homo sapiens | | | = 3.041 nM | | | NPASS |
| C8166 | Homo sapiens | | | = 41.48 nM | | | NPASS |
| C3A | Homo sapiens | | | = 56.87 nM | | | NPASS |
| BEN | Homo sapiens | | | = 107.08 nM | | | NPASS |
| BFTC-905 | Homo sapiens | | | = 0.1398 nM | | | NPASS |
| BFTC-909 | Homo sapiens | | | = 6.925 nM | | | NPASS |
| BGC-823 | Homo sapiens | | | = 9670.0 nM|= 9700.0 nM|= 210.0 nM|= 57.0 nM | | | NPASS |
| BHT-101 | Homo sapiens | | | = 1.822 nM | | | NPASS |
| BHY | Homo sapiens | | | = 5.31 nM | | | NPASS |
| BJ | Homo sapiens | | = 7.67 nM | > 40000.0 nM | | | NPASS |
| BPH-1 | Homo sapiens | | | = 2.082 nM | | | NPASS |
| BT-20 | Homo sapiens | | | = 70.0 nM|< 10.0 nM|= 25.99 nM | | | NPASS |
| BT-474 | Homo sapiens | | | = 12750.0 nM|= 1985.76 nM | | | NPASS |
| BT-549 | Homo sapiens | | | = 17.64 nM | | | NPASS |
| BV-173 | Homo sapiens | | | = 2.381 nM | | | NPASS |
| BXPC-3 | Homo sapiens | | | = 240.0 nM|= 116.78 nM|= 62.5 nM | | | NPASS |
| Becker | Homo sapiens | | | = 23.34 nM | | | NPASS |
| Bel-7402 | Homo sapiens | | | = 7.0 nM|= 2.72 ug.mL-1|= 12500.0 nM|= 170.0 nM|= 260.0 nM|= 14.0 nM | | | NPASS |
| Bile salt export pump | Homo sapiens | O95342 | | >135000 nM|>133000 nM|> 135000.0 nM|> 133000.0 nM | | | BindingDB, NPASS |
| C-33-A | Homo sapiens | | | = 6.477 nM | | | NPASS |
| C2BBe1 | Homo sapiens | | | = 2.438 nM | | | NPASS |
| C32 | Homo sapiens | | | = 13.37 nM | | | NPASS |
| C6 | Rattus norvegicus | | | < 1850.0 nM | | | NPASS |
| EOL1 | Homo sapiens | | | = 0.2708 nM | | | NPASS |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens | Q92887 | | > 133000.0 nM | | | NPASS |
| ES1 | Homo sapiens | | | = 0.09574 nM | | | NPASS |
| IST-SL1 | Homo sapiens | | | = 34.38 nM | | | NPASS |
| Integrase | Human immunodeficiency virus 1 | | | >100000 nM | | | BindingDB |
| J-RT3-T3-5 | Homo sapiens | | | = 2.579 nM | | | NPASS |
| J82 | Homo sapiens | | | = 4.722 nM | | | NPASS |
| JAR | Homo sapiens | | | = 14.54 nM | | | NPASS |
| JEG-3 | Homo sapiens | | | = 13.12 nM | | | NPASS |
| JVM-2 | Homo sapiens | | | = 3029.5 nM | | | NPASS |
| JVM-3 | Homo sapiens | | | = 2.504 nM | | | NPASS |
| IST-MES1 | Homo sapiens | | | = 10.56 nM | | | NPASS |
| Jurkat | Homo sapiens | | | = 5.6 nM|= 1.4 nM|= 26.0 nM|= 110.0 nM|= 85.0 nM|= 22000.0 nM|= 51500.0 nM|= 100.0 nM | | | NPASS |
| K562 | Homo sapiens | | | = 57.0 nM|= 40.0 nM|= 1400.0 nM|= 80.0 nM|= 2.0 nM|= 590.0 nM|= 1180.0 nM|= 1077.74 nM|= 31.0 nM|= 400.0 nM|= 130.0 nM|= 5370.0 nM|< 3.0 nM|= 90.0 nM|= 711.0 nM|= 70.0 nM|= 320.0 nM|= 2690.0 nM|= 580.0 nM | | | NPASS |
| KALS-1 | Homo sapiens | | | = 69.89 nM | | | NPASS |
| KARPAS-299 | Homo sapiens | | | = 2892.53 nM | | | NPASS |
| KARPAS-45 | Homo sapiens | | | = 134.47 nM | | | NPASS |
| KATO III stomach cancer cell lines | | | | = 46000000.0 nM|= 1170.0 nM | | | NPASS |
| KB | Homo sapiens | | = 3.6 nM|= 0.01 ug.mL-1 | = 9.0 nM|= 40.0 nM|= 70.0 nM|= 30.0 nM|= 35.0 nM|= 1040.0 nM|= 0.01 ug.mL-1|= 0.04 ug.mL-1|= 8.0 nM|< 0.005 ug.mL-1|= 20.0 nM|= 28.7 nM|= 3.0 nM|= 38.0 nM|= 1220.0 nM|< 13.0 nM|= 8.8 nM|= 121.0 nM|= 37.0 nM|= 50.0 nM | | | NPASS |
| KB 3-1 | Homo sapiens | | | = 10.0 nM|= 20.0 nM | | | NPASS |
| KB VCR R | | | | = 9.0 nM|= 0.03 ug.mL-1 | | | NPASS |
| K5 | Homo sapiens | | | = 3.201 nM | | | NPASS |
| IST-MEL1 | Homo sapiens | | | = 3.81 nM | | | NPASS |
| IMR-90 | Homo sapiens | | | = 430.0 nM | | | NPASS |
| IMR-32 | Homo sapiens | | | = 80.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 117.2 nM|= 500.0 nM|= 1080.0 nM|= 0.19 ug.mL-1|= 72.0 nM|= 200.0 nM|= 1850.0 nM|= 860.0 nM|= 630.0 nM|= 1220.0 nM|= 580.0 nM|= 940.0 nM|= 400.0 nM|= 1100.0 nM|= 8.9 nM|= 1500.0 nM|= 8930.0 nM|= 1010.0 nM|= 1570.0 nM|= 0.28 ug.mL-1|= 24.0 nM|= 130.0 nM|= 420.0 nM|= 11620.0 nM|= 180.0 nM|= 410.0 nM|= 14000.0 nM|= 1590.0 nM|= 6130.0 nM|= 19800.0 nM|= 590.0 nM|= 60010.0 nM|= 90.0 nM|= 60.0 nM|= 10100.0 nM|= 3800.0 nM|= 2620.0 nM|= 120.0 nM|= 1370.0 nM|= 80.0 nM|= 1300.0 nM|> 50000.0 nM|= 660.0 nM|= 6510.0 nM|= 1660.0 nM|= 8280.0 nM|= 6000.0 nM|= 230.0 nM | | | NPASS |
| Hep 3B2 | Homo sapiens | | | = 434.29 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 6.3 nM|= 0.09 ug.mL-1|= 30.0 nM|= 300.0 nM|= 130.0 nM|= 200.0 nM|= 455.0 nM|= 60.0 nM|= 6400.0 nM|= 20.0 nM|< 100.0 nM|= 10.0 nM|= 32300.0 nM|= 600.0 nM|= 50.0 nM|< 1000.0 nM|= 4920.0 nM|= 13200.0 nM|= 500.0 nM|= 430.0 nM|= 4370.0 nM|= 370.0 nM|= 6080.0 nM|= 1360.0 nM|= 4790.0 nM|= 660.0 nM|= 5690.0 nM|= 400.0 nM|= 40.0 nM|= 110.0 nM|= 33.16 nM|< 1850.0 nM|= 3500.0 nM | | | NPASS |
| Heterogeneous nuclear ribonucleoprotein A1 | Homo sapiens | P09651 | | | 82.7 nM|= 82.7 nM | | BindingDB, NPASS |
| Histone deacetylase | Homo sapiens | O15379|P56524|Q13547|Q8WUI4|Q92769|Q969S8|Q96DB2|Q9BY41|Q9UBN7|Q9UKV0|Q9UQL6 | | 50 nM | | | BindingDB |
| Histone deacetylase | Homo sapiens | Q13547|O15379|Q9UBN7|Q92769|Q9UQL6|Q8WUI4|Q9BY41|Q96DB2|P56524|Q9UKV0|Q969S8 | | = 50.0 nM | | | NPASS |
| Hs-578T | Homo sapiens | | | = 144.69 nM | | | NPASS |
| HuCCT-1 | Homo sapiens | | | = 73.21 nM | | | NPASS |
| HuO-3N1 | Homo sapiens | | | = 12.65 nM | | | NPASS |
| HuO9 | Homo sapiens | | | = 2.881 nM | | | NPASS |
| HuP-T3 | Homo sapiens | | | = 36.35 nM | | | NPASS |
| HuP-T4 | Homo sapiens | | | = 0.8814 nM | | | NPASS |
| HuTu80 | Homo sapiens | | | = 3.382 nM | | | NPASS |
| Huh-7 | Homo sapiens | | | < 100.0 nM|= 150.0 nM|= 60.0 nM|= 115.84 nM|= 0.32 nM|= 2.3 nM|< 1850.0 nM | | | NPASS |
| Human immunodeficiency virus type 1 integrase | Human immunodeficiency virus 1 | Q7ZJM1 | | > 100000.0 nM | | | NPASS |
| Human immunodeficiency virus type 1 reverse transcriptase | Human immunodeficiency virus 1 | Q72547 | | > 200.0 ug.mL-1 | | | NPASS |
| IA-LM | Homo sapiens | | | = 12.0 nM | | | NPASS |
| IGR-1 | Homo sapiens | | | = 151.26 nM | | | NPASS |
| IGROV-1 | Homo sapiens | | | = 1650.0 nM|= 12.0 nM|= 36.34 nM | | | NPASS |
| KE-37 | Homo sapiens | | | = 1.535 nM | | | NPASS |
| KG-1 | Homo sapiens | | | = 2310.0 nM | | | NPASS |
| KG-1 | | | | = 1.11 nM|= 1600.0 nM | | | NPASS |
| KGN | Homo sapiens | | | = 10.59 nM | | | NPASS |
| KYSE-510 | Homo sapiens | | | = 6.754 nM | | | NPASS |
| KYSE-520 cell line | | | | = 82.56 nM | | | NPASS |
| KYSE-70 cell line | | | | = 92.14 nM | | | NPASS |
| Kasumi 1 | | | | = 4.066 nM | | | NPASS |
| L-363 | Homo sapiens | | | = 1.869 nM | | | NPASS |
| L-428 | Homo sapiens | | | = 148.3 nM | | | NPASS |
| L02 | Homo sapiens | | | = 2150.0 nM|> 150000.0 nM|= 140.0 nM | | | NPASS |
| L1210 | Mus musculus | | | = 30.0 nM|= 23.0 nM|= 330.0 nM|= 15.0 nM|= 126.0 nM|= 14.0 nM|= 180.0 nM|= 60.0 nM|= 510.0 nM | | | NPASS |
| L2987 | Homo sapiens | | | = 400.0 nM | | | NPASS |
| LAMA-84 | Homo sapiens | | | = 7.02 nM | | | NPASS |
| LAN-6 | Homo sapiens | | | = 124.47 nM | | | NPASS |
| LB1047-RCC | Homo sapiens | | | = 7.897 nM | | | NPASS |
| LB2241-RCC | Homo sapiens | | | = 2.076 nM | | | NPASS |
| LB373-MEL-D | Homo sapiens | | | = 91.19 nM | | | NPASS |
| LB771-HNC | Homo sapiens | | | = 196.84 nM | | | NPASS |
| LB831-BLC | Homo sapiens | | | = 18.37 nM | | | NPASS |
| LC-2-ad | Homo sapiens | | | = 2.806 nM | | | NPASS |
| LCLC-103H cell line | | | | = 20.49 nM | | | NPASS |
| LCLC-97TM1 | Homo sapiens | | | = 8.136 nM | | | NPASS |
| KYSE-450 | Homo sapiens | | | = 23.73 nM | | | NPASS |
| HUVEC | Homo sapiens | | | = 200.0 nM|= 10.0 nM|= 60.0 nM|= 12.0 nM | | | NPASS |
| KYSE-410 | Homo sapiens | | | = 78.11 nM | | | NPASS |
| KYSE-180 | Homo sapiens | | | = 13.18 nM | | | NPASS |
| KINGS-1 | Homo sapiens | | | = 332.9 nM | | | NPASS |
| KLE | Homo sapiens | | | = 411.5 nM | | | NPASS |
| KM-H2 | Homo sapiens | | | = 55.67 nM | | | NPASS |
| KM12 | Homo sapiens | | | = 74.99 nM | | | NPASS |
| KMOE-2 | Homo sapiens | | | = 11.26 nM | | | NPASS |
| KNS-42 | Homo sapiens | | | = 33.14 nM | | | NPASS |
| KNS-62 | Homo sapiens | | | = 7.701 nM | | | NPASS |
| KNS-81-FD | Homo sapiens | | | = 19.42 nM | | | NPASS |
| KOSC-2 | Homo sapiens | | | = 4.393 nM | | | NPASS |
| KP-4 | Homo sapiens | | | = 3.162 nM | | | NPASS |
| KP-N-YN | Homo sapiens | | | = 102.97 nM | | | NPASS |
| KP-N-YS | Homo sapiens | | | = 736.29 nM | | | NPASS |
| EPLC-272H | Homo sapiens | | | = 72.8 nM | | | NPASS |
| KU-19-19 | Homo sapiens | | | = 22.03 nM | | | NPASS |
| KU812 cell line | | | | = 8.365 nM | | | NPASS |
| KURAMOCHI | Homo sapiens | | | = 3634.01 nM | | | NPASS |
| KY821 | Homo sapiens | | | = 8.123 nM | | | NPASS |
| KYSE-140 | Homo sapiens | | | = 69.74 nM | | | NPASS |
| KYSE-150 cell line | | | | = 245.96 nM | | | NPASS |
| KYSE-270 | Homo sapiens | | | = 5.223 nM | | | NPASS |
| HTC-C3 | Homo sapiens | | | = 31.47 nM | | | NPASS |
| KS-1 | Homo sapiens | | | = 57.87 nM | | | NPASS |
| HT1197 | Homo sapiens | | | = 1093.19 nM | | | NPASS |
| G-402 | Homo sapiens | | | = 24.5 nM | | | NPASS |
| GAK | Homo sapiens | | | = 218.07 nM | | | NPASS |
| GAMG | Homo sapiens | | | = 1.527 nM | | | NPASS |
| GB-1 | Homo sapiens | | | = 4.677 nM | | | NPASS |
| GCIY | Homo sapiens | | | = 66.15 nM | | | NPASS |
| GCT | Homo sapiens | | | = 5.023 nM | | | NPASS |
| GI-1 | Homo sapiens | | | = 3.365 nM | | | NPASS |
| GI-ME-N | Homo sapiens | | | = 33.89 nM | | | NPASS |
| GMS-10 | Homo sapiens | | | = 7.311 nM | | | NPASS |
| GOTO | Homo sapiens | | | = 0.7058 nM | | | NPASS |
| GP5d | Homo sapiens | | | = 12.49 nM | | | NPASS |
| GR-ST | Homo sapiens | | | = 0.701 nM | | | NPASS |
| HT55 | Homo sapiens | | | = 192.44 nM | | | NPASS |
| H-EMC-SS | Homo sapiens | | | = 95.58 nM | | | NPASS |
| H22 | Mus musculus | | | = 540.0 nM | | | NPASS |
| H4 | Homo sapiens | | | = 0.6154 nM | | | NPASS |
| H9 | Homo sapiens | | | = 0.3582 nM | | | NPASS |
| HAL-01 | Homo sapiens | | | = 2.551 nM | | | NPASS |
| HC-1 | Homo sapiens | | | = 3.344 nM | | | NPASS |
| G-401 | Homo sapiens | | | = 19.16 nM | | | NPASS |
| HCC 2998 | Homo sapiens | | | = 150.28 nM | | | NPASS |
| G-361 | Homo sapiens | | | = 2544.45 nM | | | NPASS |
| FTC-133 | Homo sapiens | | | = 4.567 nM | | | NPASS |
| ES3 | Homo sapiens | | | = 0.9311 nM | | | NPASS |
| ES4 | Homo sapiens | | | = 1.474 nM | | | NPASS |
| ES5 | Homo sapiens | | | = 0.7735 nM | | | NPASS |
| ES6 | Homo sapiens | | | = 88.05 nM | | | NPASS |
| ES7 | Homo sapiens | | | = 0.02543 nM | | | NPASS |
| ES8 | Homo sapiens | | | = 0.7956 nM | | | NPASS |
| ESS-1 | Homo sapiens | | | = 7.079 nM | | | NPASS |
| ETK-1 | Homo sapiens | | | = 34.89 nM | | | NPASS |
| EW-1 | Homo sapiens | | | = 1.777 nM | | | NPASS |
| EW-11 | Homo sapiens | | | = 2.659 nM | | | NPASS |
| EW-13 | Homo sapiens | | | = 3.267 nM | | | NPASS |
| EW-16 | Homo sapiens | | | = 0.1214 nM | | | NPASS |
| EW-18 | Homo sapiens | | | = 150.08 nM | | | NPASS |
| EW-22 | Homo sapiens | | | = 0.5566 nM | | | NPASS |
| EW-24 | Homo sapiens | | | = 4.033 nM | | | NPASS |
| EW-3 | Homo sapiens | | | = 0.3192 nM | | | NPASS |
| Erythrocyte | | | = 429.9 ug.mL-1 | | | | NPASS |
| Eukaryotic translation initiation factor 2-alpha kinase 3 | Homo sapiens | Q9NZJ5 | > 55700.0 nM | | | | NPASS |
| Eukaryotic translation initiation factor 2-alpha kinase 3 | Human | Q9NZJ5 | >55700 nM | | | | BindingDB |
| FaDu | Homo sapiens | | | = 0.5392 nM | | | NPASS |
| HCC1187 | Homo sapiens | | | = 314.07 nM | | | NPASS |
| GT3TKB | Homo sapiens | | | = 1.759 nM | | | NPASS |
| HCC1419 | Homo sapiens | | | = 4155.69 nM | | | NPASS |
| HL-60 | Homo sapiens | | | = 66.0 nM|= 5.0 nM|= 18.0 nM|= 13.0 nM|= 130000.0 nM|= 89.0 nM|= 800.0 nM|= 6.0 nM|= 65.0 nM|= 67.0 nM|= 590.0 nM|= 100.0 nM|= 17.0 nM|= 600.0 nM|= 3.734 nM|= 60.0 nM|= 15.0 nM|= 920.0 nM|= 19.0 nM|= 6.7 nM|= 20.0 nM|= 70.0 nM|= 420.0 nM|< 64.0 nM|= 1700.0 nM|= 910.0 nM | | | NPASS |
| HLE | Homo sapiens | | | = 5.753 nM | | | NPASS |
| HMV-2 cell line | | | | = 8.887 nM | | | NPASS |
| HN | Homo sapiens | | | = 1.399 nM | | | NPASS |
| HO-1-N-1 | Homo sapiens | | | = 0.8385 nM | | | NPASS |
| HOC-21 cell line | | | | = 0.0147 ug.mL-1 | | | NPASS |
| HCC1395 | Homo sapiens | | | = 1367.35 nM | | | NPASS |
| HOP-92 | Homo sapiens | | | = 8.787 nM | | | NPASS |
| HOS | Homo sapiens | | | = 1.398 nM | | | NPASS |
| HPAF-II | Homo sapiens | | | = 55.12 nM | | | NPASS |
| HSC-2 | Homo sapiens | | | = 11.7 nM | | | NPASS |
| HSC-3 | Homo sapiens | | | = 3.015 nM | | | NPASS |
| HSC-4 | Homo sapiens | | | = 0.1816 nM | | | NPASS |
| HT | Homo sapiens | | | = 29.71 nM | | | NPASS |
| HT-1080 | Homo sapiens | | | = 80.0 nM|= 0.3944 nM | | | NPASS |
| HT-1376 | Homo sapiens | | | = 1780.55 nM | | | NPASS |
| HT-144 | Homo sapiens | | | = 17.86 nM | | | NPASS |
| HT-29 | Homo sapiens | | = 60.0 nM | = 46.0 nM|= 1400.0 nM|= 80.0 nM|= 87.8 nM|= 30.0 nM|= 14.0 nM|= 3160.0 nM|= 8810.0 nM|= 2000.0 nM|= 90.0 nM|= 120.0 nM|= 400.0 nM|= 850.0 nM|= 1220.0 nM|= 1070.0 nM|= 260.0 nM|= 10000.0 nM|= 85.52 nM|= 0.7 nM|= 60.0 nM|> 100000.0 nM|= 70.0 nM|> 150000.0 nM|= 1370.0 nM | | | NPASS |
| HT-3 | Homo sapiens | | | = 0.2119 nM | | | NPASS |
| HH | Homo sapiens | | | = 13.52 nM | | | NPASS |
| HGC-27 | Homo sapiens | | | = 4.073 nM|> 150000.0 nM|= 166.0 nM | | | NPASS |
| HOP-62 | Homo sapiens | | | = 3293.6 nM | | | NPASS |
| HEL | Homo sapiens | | | = 6.311 nM | | | NPASS |
| HCC1569 | Homo sapiens | | | = 267.54 nM | | | NPASS |
| HCC1806 | Homo sapiens | | | = 3.143 nM | | | NPASS |
| HEp-2 | Homo sapiens | | | = 0.02 ug.mL-1|= 700.0 nM|= 3040.0 nM|= 3010.0 nM | | | NPASS |
| HCC1954 | Homo sapiens | | | = 266.61 nM | | | NPASS |
| HCC2218 | Homo sapiens | | | = 55.5 nM | | | NPASS |
| HCC38 | Homo sapiens | | | = 12.86 nM | | | NPASS |
| HCC70 | Homo sapiens | | | = 45.46 nM|= 44.0 nM | | | NPASS |
| HCCLM9 | Homo sapiens | | | > 150000.0 nM | | | NPASS |
| HCE-4 | Homo sapiens | | | = 1.814 nM | | | NPASS |
| HCC1937 | Homo sapiens | | | = 349.21 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | = 1000.0 nM|= 9.0 nM|= 2.0 nM|= 2770.0 nM|= 130.0 nM|= 2300.0 nM|= 3970.0 nM|= 22.9 nM|< 100.0 nM|< 1000.0 nM|= 110.0 nM|< 10.0 nM|= 5.051 nM|= 16.0 nM|= 70.0 nM|= 90.0 nM|= 120.0 nM|= 11.5 nM|= 159.0 nM|= 1880.0 nM|= 30.0 nM|= 8.5 nM|= 20.0 nM|= 13.0 nM|= 400.0 nM|= 50.0 nM|= 250.0 nM|= 40.0 nM|< 1850.0 nM|= 600.0 nM|= 17.0 nM|= 2.01 nM | | | NPASS |
| HCT-15 | Homo sapiens | | | = 18.0 nM|= 80.0 nM|= 83.0 nM|= 3.0 nM|= 640.0 nM|= 760.0 nM|= 500.0 nM|= 67.0 nM|= 800.0 nM|= 0.096 ug.mL-1|= 166.0 nM|= 260.0 nM|= 9920.0 nM|= 1380.0 nM|= 776.97 nM|= 420.0 nM|= 2820.0 nM|= 520.0 nM|= 300.0 nM|= 6080.0 nM|= 600.0 nM|= 50.0 nM|= 20.0 nM|= 49.0 nM|= 1590.0 nM | | | NPASS |
| HCT-8 | Homo sapiens | | | = 7.0 nM|< 0.005 ug.mL-1|= 3150.0 nM|= 3200.0 nM|< 13.0 nM|= 260.0 nM|= 24.0 nM | | | NPASS |
| HCE-T | Homo sapiens | | | = 5.469 nM | | | NPASS |
| HD-MY-Z | Homo sapiens | | | = 1.634 nM | | | NPASS |
| HDLM-2 | Homo sapiens | | | = 486.07 nM | | | NPASS |
| HEC-1 | Homo sapiens | | | = 18.13 nM | | | NPASS |
| HEC-1B cell line | | | | = 8640.0 nM|= 60.0 nM | | | NPASS |
| HEK-293T | Homo sapiens | | | = 5650.0 nM|= 30.0 nM|= 690.0 nM | | | NPASS |
| HEK293 | Homo sapiens | | | = 7940.0 nM|= 1010.0 nM|= 780.0 nM|= 280.0 nM|= 10.0 nM|= 54690.0 nM|= 0.56 nM|= 1610.0 nM|= 600.0 nM|= 8750.0 nM|= 5.6 nM | | | NPASS |