
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| Endothelin-1 receptor | Homo sapiens | P25101 | 40000 nM | BindingDB | |||
| Endothelin-1 receptor | Rattus norvegicus | P26684 | 580000 nM | BindingDB | |||
| Endothelin receptor type B | Homo sapiens | P24530 | >500000 nM | BindingDB | |||
| Endothelin receptor ET-A | Homo sapiens | P25101 | = 40000.0 nM | NPASS | |||
| Endothelin receptor ET-A | Rattus norvegicus | P26684 | = 580000.0 nM | NPASS | |||
| Endothelin receptor ET-B | Homo sapiens | P24530 | > 500000.0 nM | NPASS |