
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| ATP-binding cassette sub-family G member 2 | Homo sapiens | Q9UNQ0 | = 2140.0 nM|= 1180.0 nM | NPASS | |||
| BV-2 | Mus musculus | = 28510.0 nM | NPASS | ||||
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens | Q9UNQ0 | 2140 nM|1180 nM | BindingDB | |||
| DU-145 | Homo sapiens | = 30800.0 nM | NPASS | ||||
| LNCaP | Homo sapiens | = 15600.0 nM | NPASS | ||||
| PC-3 | Homo sapiens | = 14900.0 nM | NPASS |