| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| MCF7 | Homo sapiens | | | = 14110.0 nM|= 65000.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 10000.0 nM|= 63000.0 nM|= 31170.0 nM | | | NPASS |
| NACHT, LRR and PYD domains-containing protein 3 | Mus musculus | Q8R4B8 | | >10000 nM|> 10000.0 nM | | | BindingDB, NPASS |
| NCI-H460 | Homo sapiens | | | = 17000.0 nM | | | NPASS |
| NIH3T3 | Mus musculus | | | = 12200.0 nM|= 12190.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | = 1220.0 nM | = 2960.0 nM|= 15900.0 nM|= 14050.0 nM|= 17330.0 nM|= 15180.0 nM|= 17390.0 nM | | | NPASS |
| Neofusicoccum parvum | Neofusicoccum parvum | | | = 250000.0 nM | | | NPASS |
| P-glycoprotein 1 | Homo sapiens | P08183 | | = 42000.0 nM | | | NPASS |
| PANC-1 | Homo sapiens | | | = 50000.0 nM | | | NPASS |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens | P09917 | | 530 nM|3910 nM|9320 nM | | | BindingDB |
| Prostaglandin G/H synthase 1 | Homo sapiens | P23219 | | 700 nM | | | BindingDB |
| Liver microsome | Rattus norvegicus | | = 355000.0 nM | | | | NPASS |
| Quinone reductase 2 | Homo sapiens | P16083 | | = 5100.0 nM | | | NPASS |
| RAW264.7 | Mus musculus | | | = 30000.0 nM | | | NPASS |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens | P16083 | | 5100 nM | | | BindingDB |
| Vanilloid receptor | Homo sapiens | Q8NER1 | | > 10000.0 nM | | | NPASS |
| SK-MEL-2 | Homo sapiens | | | = 17000.0 nM | | | NPASS |
| T47D | Homo sapiens | | | = 35000.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily A member 1 | Rattus norvegicus | Q6RI86 | 3600 nM|= 3600.0 nM | 7500 nM|= 7500.0 nM | | | BindingDB, NPASS |
| Transient receptor potential cation channel subfamily V member 1 | Homo sapiens | Q8NER1 | | >10000 nM | | | BindingDB |
| Transthyretin | Homo sapiens | P02766 | | | = 4600.0 nM|= 1900.0 nM | = 3500.0 nM | NPASS |
| U-87 MG | Homo sapiens | | | = 34000.0 nM | | | NPASS |
| Prostaglandin G/H synthase 2 | Homo sapiens | P35354 | | 820 nM | | | BindingDB |
| LN-229 | Homo sapiens | | | = 14000.0 nM | | | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM | | | NPASS |
| J774 | Mus musculus | | | = 16700.0 nM|= 8700.0 nM|= 10500.0 nM | | | NPASS |
| L02 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| A2780 | Homo sapiens | | | = 15560.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 71700.0 nM|= 15860.0 nM|= 26000.0 nM | | | NPASS |
| ATP-dependent translocase ABCB1 | Homo sapiens | P08183 | | 42000 nM | | | BindingDB |
| Arachidonate 5-lipoxygenase | Homo sapiens | P09917 | | = 3910.0 nM|= 530.0 nM|= 9320.0 nM|= 1630.0 nM | | | NPASS |
| BXPC-3 | Homo sapiens | | | = 31000.0 nM | | | NPASS |
| Bcr/Abl fusion protein | Homo sapiens | P11274 | | = 10000.0 nM | | | NPASS |
| Breakpoint cluster region protein/Tyrosine-protein kinase ABL1 | Homo sapiens | P00519|P11274 | | 10000 nM | | | BindingDB |
| Caco-2 | Homo sapiens | | | = 14460.0 nM | | | NPASS |
| Cyclooxygenase-1 | Homo sapiens | P23219 | | = 700.0 nM | | | NPASS |
| Cyclooxygenase-2 | Homo sapiens | P35354 | | = 820.0 nM|= 5990.0 nM | | | NPASS |
| COLO 201 | Homo sapiens | | | = 29000.0 nM | | | NPASS |
| Cytochrome P450 1B1 | Homo sapiens | Q16678 | | = 1400.0 nM | | 910 nM|= 900.0 nM|= 910.0 nM | BindingDB, NPASS |
| Histone deacetylase 6 | Homo sapiens | Q9UBN7 | | = 550.5 nM | | | NPASS |
| Cytochrome P450 1A1 | Homo sapiens | P04798 | | | | 570 nM|= 570.0 nM | BindingDB, NPASS |
| HT-29 | Homo sapiens | | | = 23800.0 nM|> 60000.0 nM|= 28000.0 nM | | | NPASS |
| HT-1080 | Homo sapiens | | | = 93400.0 nM | | | NPASS |
| HL-60 | Homo sapiens | | | = 35000.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 9430.0 nM | | | NPASS |
| Eutypa lata | Eutypa lata | | | = 251000.0 nM | | | NPASS |
| Diplodia seriata | Diplodia seriata | | | = 163000.0 nM | | | NPASS |
| DLD-1 | Homo sapiens | | | = 16450.0 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | > 60000.0 nM|= 34080.0 nM | | | NPASS |