| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Alpha-2B adrenergic receptor | Homo sapiens | P18089 | | | | 455 nM | BindingDB |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Rattus norvegicus | P22002 | | | | 1250 nM | BindingDB |
| Reverse transcriptase | Human immunodeficiency virus 1 | | | >564000 nM | | | BindingDB |
| Murine T-cell line | Mus musculus | | | = 27600.0 nM | | | NPASS |
| Human immunodeficiency virus type 1 reverse transcriptase | Human immunodeficiency virus 1 | Q72547 | | > 200.0 ug.mL-1 | | | NPASS |
| Cytochrome P450 2D6 | Homo sapiens | P10635 | | | | 80 nM|= 80.0 nM | BindingDB, NPASS |
| B-cell line | Mus musculus | | | = 40500.0 nM | | | NPASS |
| Alpha-2c adrenergic receptor | Homo sapiens | P18825 | | | | = 161.0 nM | NPASS |
| Alpha-2b adrenergic receptor | Homo sapiens | P18089 | | | | = 455.0 nM | NPASS |
| Alpha-2a adrenergic receptor | Homo sapiens | P08913 | | | | = 1218.0 nM | NPASS |
| Alpha-2C adrenergic receptor | Homo sapiens | P18825 | | | | 161 nM | BindingDB |
| Voltage-gated L-type calcium channel alpha-1C subunit | Rattus norvegicus | P22002 | | | | = 1250.0 nM | NPASS |
| Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor | Rattus norvegicus | P19328|P22086|P22909 | | 17500 nM | | 15800 nM | BindingDB |
| Alpha-2A adrenergic receptor | Homo sapiens | P08913 | | | | 1218 nM | BindingDB |
| Alpha-1d adrenergic receptor | Homo sapiens | P25100 | | | | = 253.0 nM | NPASS |
| Alpha-1b adrenergic receptor | Homo sapiens | P35368 | | | | = 517.0 nM | NPASS |
| Alpha-1a adrenergic receptor | Homo sapiens | P35348 | | | = 251.19 nM | = 142.0 nM|= 29.0 nM | NPASS |
| Alpha-1D adrenergic receptor | Homo sapiens | P25100 | | | | 253 nM | BindingDB |
| Alpha-1B adrenergic receptor | Homo sapiens | P35368 | | | | 517 nM | BindingDB |
| Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor | Rattus norvegicus | P15823|P23944|P43140 | | 220 nM | | | BindingDB |
| Alpha-1A adrenergic receptor | Homo sapiens | P35348 | | | | 29 nM|142 nM | BindingDB |
| Adrenergic receptor alpha-2 | Rattus norvegicus | P22909 | | = 17500.0 nM | = 9332.54 nM | = 15800.0 nM | NPASS |
| Adrenergic receptor alpha-2 | Homo sapiens | P18089 | | = 1038000.0 nM|= 211000.0 nM|= 871000.0 nM|= 340000.0 nM | = 330000.0 nM|= 25000.0 nM|= 37000.0 nM|= 5600.0 nM|= 2500000.0 nM|= 640000.0 nM|= 1300000.0 nM|= 170000.0 nM | | NPASS |
| Adrenergic receptor alpha-1 | Rattus norvegicus | P43140 | | = 220.0 nM | = 562.34 nM | | NPASS |
| Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor | Homo sapiens | P08913|P18089|P18825 | | 211000 nM|340000 nM|871000 nM|1038000 nM | 640000 nM|25000 nM|330000 nM|2500000 nM | | BindingDB |