| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial | Homo sapiens | Q16654 | | 345000 nM | | | BindingDB |
| [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial | Homo sapiens | Q15119 | | 192000 nM | | | BindingDB |
| Pyruvate dehydrogenase kinase isoform 4 | Homo sapiens | Q16654 | | = 345000.0 nM | | | NPASS |
| Pyruvate dehydrogenase kinase isoform 2 | Homo sapiens | Q15119 | | = 192000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | > 50000.0 nM|= 35500.0 nM | | | | NPASS |
| Carbonic anhydrase XIV | Homo sapiens | Q9ULX7 | | | | = 860.0 nM | NPASS |
| Carbonic anhydrase XII | Homo sapiens | O43570 | | | | = 950.0 nM | NPASS |
| Carbonic anhydrase IX | Homo sapiens | Q16790 | | | | = 890.0 nM | NPASS |
| Carbonic anhydrase VII | Homo sapiens | P43166 | | | | = 850.0 nM | NPASS |
| Carbonic anhydrase I | Homo sapiens | P00915 | | | | = 830.0 nM | NPASS |
| Carbonic anhydrase 9 | Homo sapiens | Q16790 | | | | 890 nM | BindingDB |
| Carbonic anhydrase 7 | Homo sapiens | P43166 | | | | 850 nM | BindingDB |
| Carbonic anhydrase 2 | Homo sapiens | P00918 | | | | 760 nM | BindingDB |
| Carbonic anhydrase 14 | Homo sapiens | Q9ULX7 | | | | 860 nM | BindingDB |
| Carbonic anhydrase 12 | Homo sapiens | O43570 | | | | 950 nM | BindingDB |
| Carbonic anhydrase 1 | Homo sapiens | P00915 | | | | 830 nM | BindingDB |
| Carbonic anhydrase II | Homo sapiens | P00918 | | | | = 760.0 nM | NPASS |