| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| MCF7 | Homo sapiens | | | = 55000.0 nM | | | NPASS |
| MES-SA | Homo sapiens | | | = 30000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 23000.0 nM|= 21000.0 nM | | | NPASS |
| Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | Q07820 | | | | 2270 nM|= 2270.0 nM | BindingDB, NPASS |
| DU-145 | Homo sapiens | | | = 29000.0 nM | | | NPASS |
| Apoptosis regulator Bcl-2 | Homo sapiens | P10415 | | | | 1700 nM|= 1700.0 nM | BindingDB, NPASS |
| Induced myeloid leukemia cell differentiation protein Mcl-1 [172-327] | Homo sapiens | Q07820 | | | 1.350e+6 nM | | BindingDB |