| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Pyruvate kinase PKM | Homo sapiens | P14618 | | 1920000 nM | | | BindingDB |
| Protein-tyrosine phosphatase 2C | Homo sapiens | Q06124 | | = 2590.0 nM | | | NPASS |
| Protein-tyrosine phosphatase 1C | Homo sapiens | P29350 | | = 2140.0 nM | | | NPASS |
| Protease | Human immunodeficiency virus 1 | Q9YQ12 | | = 59200.0 nM | | | NPASS |
| Peroxisome proliferator-activated receptor gamma | Homo sapiens | P37231 | | | | = 2560.0 nM | NPASS |
| NCI-N87 | Homo sapiens | | | = 3100.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | = 1200.0 nM | = 3300.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | > 20000.0 nM | > 50000.0 nM|= 400.0 nM | | | NPASS |
| Monoglyceride lipase | Homo sapiens | Q99685 | | = 48000.0 nM | | | NPASS |
| MIA PaCa-2 | Homo sapiens | | | = 1900.0 nM | | | NPASS |
| Pyruvate kinase isozymes M1/M2 | Homo sapiens | P14618 | | = 1920000.0 nM | | | NPASS |
| Papain | Carica papaya | P00784 | | 122000 nM|= 122000.0 nM | | | BindingDB, NPASS |
| RAW264.7 | Mus musculus | | | = 18170.0 nM | | | NPASS |
| Telomerase reverse transcriptase | Homo sapiens | O14746 | | 5000 nM|500 nM|= 5000.0 nM|= 500.0 nM | | | BindingDB, NPASS |
| Replicase polyprotein 1a | Severe acute respiratory syndrome coronavirus | P0C6U8 | | 1600 nM|17100 nM|89100 nM | | 11200 nM | BindingDB |
| Replicase polyprotein 1ab | Human SARS coronavirus | P0C6X7 | | 89100 nM | | | BindingDB |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | P0DTD1 | | = 1571.0 nM | | | NPASS |
| SARS coronavirus 3C-like proteinase | SARS coronavirus | P0C6U8 | | = 89100.0 nM|= 1600.0 nM|= 17100.0 nM | | = 11200.0 nM | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | > 200000.0 nM | | | | NPASS |
| SGC-7901 | Homo sapiens | | | = 250000.0 nM | | | NPASS |
| MGC-803 | Homo sapiens | | | > 5000.0 nM | | | NPASS |
| Toxoplasma gondii | Toxoplasma gondii | | | = 2500.0 nM | | | NPASS |
| Tryptophan 2,3-dioxygenase | Homo sapiens | P48775 | | > 10000.0 nM | | | NPASS |
| Tyrosine-protein phosphatase non-receptor type 11 | Homo sapiens | Q06124 | | 2590 nM | | | BindingDB |
| Tyrosine-protein phosphatase non-receptor type 6 | Homo sapiens | P29350 | | 2140 nM | | | BindingDB |
| U-937 | Homo sapiens | | | > 5000.0 nM | | | NPASS |
| Replicase polyprotein 1a | SARS-CoV | P0C6U8 | | 800 nM | | | BindingDB |
| MDA-MB-231 | Homo sapiens | | | = 115900.0 nM|= 7695.0 nM | | | NPASS |
| SAOS-2 | Homo sapiens | | > 20000.0 nM | | | | NPASS |
| Liver carboxylesterase 1 | Homo sapiens | P23141 | | | | 6890 nM | BindingDB |
| A549 | Homo sapiens | | | = 53200.0 nM|= 6680.0 nM|= 2200.0 nM | | | NPASS |
| AGS | Homo sapiens | | | = 10000.0 nM|= 6800.0 nM | | | NPASS |
| Acetylcholinesterase | Homo sapiens | P22303 | | >140000 nM|> 140000.0 nM | | >100000 nM|> 100000.0 nM | BindingDB, NPASS |
| Acyl coenzyme A:cholesterol acyltransferase | Homo sapiens | P23141 | | | | = 6890.0 nM | NPASS |
| Aldo-keto reductase family 1 member B1 | Homo sapiens | P15121 | | 8690 nM | | | BindingDB |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus | P07943 | | 1140 nM|1148 nM | | | BindingDB |
| Aldose reductase | Homo sapiens | P15121 | | = 8690.0 nM | | | NPASS |
| Apoptotic protease-activating factor 1 | Homo sapiens | O14727 | | 4820 nM|>100000 nM|> 100000.0 nM|= 4820.0 nM | | | BindingDB, NPASS |
| BGC-823 | Homo sapiens | | | = 2800.0 nM | | | NPASS |
| CWR22R | Homo sapiens | | | = 6700.0 nM | | | NPASS |
| Carboxylesterase 2 | Homo sapiens | O00748 | | | | = 69.4 nM|= 2450.0 nM | NPASS |
| Caspase-9 | Homo sapiens | P55211 | | 11200 nM | | | BindingDB |
| Aldose reductase | Rattus norvegicus | P07943 | | = 1140.0 nM|= 1148.15 nM | | | NPASS |
| DNA-(apurinic or apyrimidinic site) endonuclease | Homo sapiens | P27695 | | | 0.880000 nM | | BindingDB |
| Cocaine esterase | Homo sapiens | O00748 | | | | 69 nM|2450 nM | BindingDB |
| L02 | Homo sapiens | | | = 78500.0 nM|= 65290.0 nM | | | NPASS |
| Indoleamine 2,3-dioxygenase | Homo sapiens | P14902 | | > 10000.0 nM | | | NPASS |
| Hypoxia inducible factors; HIF-1-alpha, HIF-2-alpha | Homo sapiens | | | = 7530.0 nM|= 6180.0 nM | | | NPASS |
| Histone-lysine N-methyltransferase EZH2/Polycomb protein EED/Polycomb protein SUZ12 | Homo sapiens | O75530|Q15022|Q15910 | | 28100 nM | | | BindingDB |
| HepG2 | Homo sapiens | | | = 65700.0 nM|= 4910.0 nM|= 23850.0 nM|= 23900.0 nM | | | NPASS |
| LNCaP | Homo sapiens | | | = 500.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | = 900.0 nM | = 7793.5 nM|> 5000.0 nM | | | NPASS |
| Endothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha | Homo sapiens | Q16665|Q99814 | | 7530 nM|6180 nM | | | BindingDB |
| EZH2/SUZ12/EED complex | Homo sapiens | Q15022 | | = 28100.0 nM | | | NPASS |
| Dengue virus type 2 NS3 protein | Dengue virus type 2 (strain Thailand/16681/1984) (DENV-2) | P29990 | | > 100000.0 nM | | | NPASS |
| DNA-(apurinic or apyrimidinic site) lyase | Homo sapiens | P27695 | | | = 0.88 nM | | NPASS |
| HeLa | Homo sapiens | | | = 193200.0 nM|= 3470.0 nM | | | NPASS |
