| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Sorbitol dehydrogenase | Homo sapiens | Q00796 | | 106000 nM|= 106000.0 nM | | | BindingDB, NPASS |
| Xanthine dehydrogenase | Homo sapiens | P47989 | | = 131000.0 nM | | | NPASS |
| Xanthine dehydrogenase/oxidase | Homo sapiens | P47989 | | 131000 nM | | | BindingDB |
| Tyrosinase | Homo sapiens | P14679 | | | | 3400 nM|= 3400.0 nM | BindingDB, NPASS |
| Serine racemase | Homo sapiens | Q9GZT4 | | >10000000 nM|> 10000000.0 nM | | | BindingDB, NPASS |
| U-937 | Homo sapiens | | | > 2000000.0 nM | | | NPASS |
| SK-MEL-28 | Homo sapiens | | | = 1200.0 nM | | | NPASS |
| Aldo-keto reductase family 1 member B1 | Homo sapiens | P15121 | | 62000 nM | | | BindingDB |
| Aldose reductase | Homo sapiens | P15121 | | = 62000.0 nM | | | NPASS |
| SK-MEL3 | Homo sapiens | | | = 6800.0 nM | | | NPASS |
| D-aspartate oxidase | Homo sapiens | Q99489 | | 7579000 nM|= 7579000.0 nM | | | BindingDB, NPASS |
| D-amino-acid oxidase | Homo sapiens | P14920 | | 943 nM|440 nM|35 nM|= 943.0 nM|= 440.0 nM|= 34.67 nM | 6300 nM|4000 nM|5600 nM|= 6300.0 nM|= 4000.0 nM|= 5600.0 nM | 156 nM|13 nM|= 156.0 nM|= 3690.0 nM|= 265.0 nM|= 13.0 nM | BindingDB, NPASS |