| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D | Homo sapiens | P27815|Q07343|Q08493|Q08499 | | | | 163000 nM | BindingDB |
| Xanthine dehydrogenase/oxidase | Homo sapiens | P47989 | | >200000 nM | | | BindingDB |
| Adenosine receptor A2a/A2b | Rattus norvegicus | P29276|P30543 | | | | 6600 nM|47000 nM | BindingDB |
| Adenosine receptor A2a/A2b | Homo sapiens | P29274|P29275 | | | | 1900 nM | BindingDB |
| Adenosine receptor A1 | Cavia porcellus | P47745 | | | | 11500 nM | BindingDB |
| Adenosine receptor A2a | Cavia porcellus | P46616 | | | | 67100.0 nM | BindingDB |
| Adenosine receptor A1 | Rattus norvegicus | P25099 | | | | >10000 nM|17000 nM|9000 nM|36000 nM | BindingDB |
| Adenosine receptor A2a | Homo sapiens | P29274 | 75900.0 nM | | | >10000 nM | BindingDB |