| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| PC-3 | Homo sapiens | | | > 25000.0 nM | | | NPASS |
| DU-145 | Homo sapiens | | | = 20300.0 nM | | | NPASS |
| DU-4475 | Homo sapiens | | | = 6740.0 nM | | | NPASS |
| Ghrelin O-acyltransferase | Human | Q96T53 | | >1.000e+6 nM | | | BindingDB |
| HCT-116 | Homo sapiens | | | = 9580.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 13510.0 nM | | | NPASS |
| MDA-MB-468 | Homo sapiens | | | = 6090.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 5960.0 nM | | | NPASS |
| Steroid C26-monooxygenase | Mycobacterium tuberculosis (strain CDC 1551 / Oshkosh) | P9WPL4 | | | 3.6e+2 nM | | BindingDB |
| Steroid C26-monooxygenase | Mycobacterium tuberculosis (strain CDC 1551 / Oshkosh) | P9WPP0 | | | 1.2e+3 nM | | BindingDB |