For more information regarding the endpoints, refer to the 'ToxCast Endpoints' file on the
DOWNLOAD page.
ToxCast Endpoints for intended target type: RNA
Assay Name | Tissue | Target Gene ID | Target HGNC Symbol | Target UniProt ID | Response | AC50 value |
---|
LTEA_HepaRG_ABCC2 | Liver | 1244 | ABCC2 | Q92887 | Activatory | 9.92 μM |
LTEA_HepaRG_ABCG2 | Liver | 9429 | ABCG2 | Q9UNQ0 | Activatory | 9.40 μM |
LTEA_HepaRG_CYP2B6 | Liver | 1555 | CYP2B6 | P20813 | Activatory | 5.80 μM |
LTEA_HepaRG_CYP2C19 | Liver | 1557 | CYP2C19 | P33261 | Activatory | 15.42 μM |
LTEA_HepaRG_CYP2C8 | Liver | 1558 | CYP2C8 | P10632 | Activatory | 12.70 μM |
LTEA_HepaRG_CYP2C9 | Liver | 1559 | CYP2C9 | P11712 | Activatory | 6.12 μM |
LTEA_HepaRG_CYP2E1 | Liver | 1571 | CYP2E1 | P05181 | Inhibitory | 10.06 μM |
LTEA_HepaRG_CYP3A4 | Liver | 1576 | CYP3A4 | P08684 | Activatory | 7.10 μM |
LTEA_HepaRG_CYP3A7 | Liver | 1551 | CYP3A7 | P24462 | Activatory | 5.99 μM |
LTEA_HepaRG_UGT1A1 | Liver | 54658 | UGT1A1 | P22309 | Activatory | 7.77 μM |
ToxCast Endpoints for intended target type: Protein
Assay Name | Tissue | Target Gene ID | Target HGNC Symbol | Target UniProt ID | Response | AC50 value |
---|
BSK_3C_TissueFactor | Vascular | 2152 | F3 | P13726 | Inhibitory | 3.97 μM |
TOX21_p450_CYP1A2_Antagonist | | 1544 | CYP1A2 | P05177 | Loss | 3.96 μM |
TOX21_p450_CYP1A2_Antagonist | | 1544 | CYP1A2 | P05177 | Loss | 4.06 μM |
No ToxCast endpoints for intended target type: Molecular Messengers
No ToxCast endpoints for intended target type: Pathway
No ToxCast endpoints for intended target type: Cellular
No ToxCast endpoints for intended target type: Extracellular