Flufenacet

Target genes for Flufenacet is obtained based on ToxCast assay component endpoints.
Chemical nameGene identifierToxCast assay component endpoint name
FlufenacetCREB3ATG_CRE_CIS_up
FlufenacetCSF1BSK_hDFCGF_MCSF_down
FlufenacetCYP1A1CLD_CYP1A1_48hr
FlufenacetCYP1A2CLD_CYP1A2_48hr
FlufenacetCYP2B6CLD_CYP2B6_24hr
FlufenacetCYP2B6CLD_CYP2B6_6hr
FlufenacetCYP2C19NVS_ADME_hCYP2C19
FlufenacetCYP2C18NVS_ADME_hCYP2C18
FlufenacetCYP3A4CLD_CYP3A4_48hr
FlufenacetESR2TOX21_ERb_BLA_Antagonist_ratio
FlufenacetESRRATOX21_ERR_Antagonist
FlufenacetESRRATOX21_PGC_ERR_Antagonist
FlufenacetETS1ATG_Ets_CIS_dn
FlufenacetFOXO1ATG_FoxO_CIS_dn
FlufenacetFOXO3ATG_FoxO_CIS_dn
FlufenacetFOSATG_AP_1_CIS_up
FlufenacetNR3C1ATG_GRE_CIS_dn
FlufenacetNR3C1TOX21_GR_BLA_Antagonist_ratio
FlufenacetHLA-DRABSK_BE3C_HLADR_down
FlufenacetCXCL10BSK_KF3CT_IP10_down
FlufenacetCXCL10BSK_hDFCGF_IP10_down
FlufenacetARTOX21_AR_BLA_Antagonist_ratio
FlufenacetARACEA_AR_antagonist_80hr
FlufenacetARTOX21_AR_LUC_MDAKB2_Antagonist_0.5nM_R1881
FlufenacetJUNATG_AP_1_CIS_up
FlufenacetSMAD1ATG_BRE_CIS_up
FlufenacetACHENVS_ENZ_hAChE
FlufenacetMMP1BSK_hDFCGF_MMP1_up
FlufenacetMTF1ATG_MRE_CIS_up
FlufenacetNFIAATG_NFI_CIS_up
FlufenacetNFE2L2ATG_NRF2_ARE_CIS_up
FlufenacetNFE2L2TOX21_ARE_BLA_agonist_ratio
FlufenacetNFKB1ATG_NF_kB_CIS_up
FlufenacetPGRTOX21_PR_BLA_Antagonist_ratio
FlufenacetPOU2F1ATG_Oct_MLP_CIS_up
FlufenacetPPARGTOX21_PPARg_BLA_antagonist_ratio
FlufenacetPPARGATG_PPARg_TRANS_up
FlufenacetBCHENVS_ENZ_hES
FlufenacetCCL2BSK_4H_MCP1_down
FlufenacetSELPBSK_4H_Pselectin_down
FlufenacetSLC6A3NVS_TR_hDAT
FlufenacetSLC6A4NVS_TR_hSERT
FlufenacetSULT2A1CLD_SULT2A_24hr
FlufenacetTSPONVS_MP_hPBR
FlufenacetTNFBSK_LPS_TNFa_up
FlufenacetNR1H2ATG_LXRb_TRANS_up
FlufenacetVCAM1BSK_hDFCGF_VCAM1_down
FlufenacetVDRATG_VDRE_CIS_up
FlufenacetXBP1ATG_Xbp1_CIS_up
FlufenacetNR1I2ATG_PXR_TRANS_up
FlufenacetNR1I2ATG_PXRE_CIS_up
FlufenacetNR1I3ATG_PBREM_CIS_up
FlufenacetNR1I3TOX21_CAR_Agonist
FlufenacetNR1H4TOX21_FXR_BLA_antagonist_ratio

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