Bexarotene


Curated chemical-gene interactions from CTD
Entrez gene IDGene symbolInteraction typeReference
100043194 SULT2A2 Decreases expression PMID:16648578
100384898 UGT2B3 Decreases expression PMID:16648578
10062 NR1H3 Decreases expression PMID:32123961
10095 ARPC1B Increases expression PMID:16648578
10144 FAM13A Decreases expression PMID:17630414
10209 EIF1 Decreases expression PMID:17178900
10237 SLC35B1 Increases expression PMID:16648578
10247 RIDA Decreases expression PMID:16648578
1026 CDKN1A Increases expression PMID:19067706
1036 CDO1 Decreases expression PMID:16648578
10434 LYPLA1 Decreases expression PMID:16648578
1054 CEBPG Decreases expression PMID:17178900
10550 ARL6IP5 Increases expression PMID:17178900
10675 CSPG5 Increases expression PMID:16648578
107460 RDH2 Increases expression PMID:16648578
10797 MTHFD2 Decreases expression PMID:17178900
10808 HSPH1 Decreases expression PMID:16648578
10957 PNRC1 Increases expression PMID:17178900
109579 ES2 Decreases expression PMID:16648578
10959 TMED2 Increases expression PMID:16648578
10961 ERP29 Increases expression PMID:16648578
10962 MLLT11 Increases expression PMID:17178900
10965 ACOT2 Increases expression PMID:16648578
10974 ADIRF Increases expression PMID:17178900
11001 SLC27A2 Decreases expression PMID:16648578
11067 DEPP1 Increases expression PMID:17178900
11140 CDC37 Increases expression PMID:16648578
11186 RASSF1 Decreases expression PMID:17849452
112 ADCY6 Decreases expression PMID:16648578
112417 UGT2B37 Decreases expression PMID:16648578
1130 LYST Increases expression PMID:17630414
11330 CTRC Increases expression PMID:16648578
1135 CHRNA2 Increases expression PMID:16648578; PMID:17630414
113868 ACAA1A Increases expression PMID:16648578
1152 CKB Increases expression PMID:16648578
120 ADD3 Increases expression PMID:17178900
121340 SP7 Decreases expression PMID:25932594
127 ADH4 Increases expression PMID:17630414
1303 COL12A1 Decreases expression PMID:16648578
13117 CYP4A10 Increases expression PMID:16648578
1312 COMT Affects expression PMID:16648578
1365 CLDN3 Increases expression PMID:16648578
1366 CLDN7 Increases expression PMID:16648578
1373 CPS1 Decreases expression PMID:16648578
1376 CPT2 Increases expression PMID:16648578
14194 FH1 Decreases expression PMID:16648578
1466 CSRP2 Decreases expression PMID:16648578
147 ADRA1B Decreases expression PMID:16648578
1491 CTH Decreases expression PMID:17178900
1512 CTSH Increases expression PMID:17178900
1528 CYB5A Decreases expression PMID:16648578
154 ADRB2 Decreases expression PMID:17178900
1544 CYP1A2 Decreases expression PMID:16648578
1545 CYP1B1 Increases expression PMID:16648578
1555 CYP2B6 Increases expression PMID:31312845
156 GRK2 Increases expression PMID:16648578
1592 CYP26A1 Increases expression PMID:17178900
1593 CYP27A1 Increases expression PMID:16648578
1601 DAB2 Decreases expression PMID:16648578
1613 DAPK3 Decreases expression PMID:16648578
16194 IL6RA Decreases expression PMID:16648578
1628 DBP Decreases expression PMID:16648578
1632 ECI1 Increases expression PMID:16648578
16369 IRS3 Increases expression PMID:17630414
1645 AKR1C1 Increases expression PMID:17178900
1649 DDIT3 Decreases expression PMID:16648578
168002 DACT2 Increases expression PMID:17630414
171380 CYP2T1 Decreases expression PMID:17630414
1717 DHCR7 Increases expression PMID:16648578
1737 DLAT Increases expression PMID:16648578
1781 DYNC1I2 Decreases expression PMID:16648578
17836 MUG1 Decreases expression PMID:16648578
1788 DNMT3A Decreases expression PMID:17849452
1831 TSC22D3 Increases expression PMID:17178900
1843 DUSP1 Decreases expression PMID:16648578; PMID:17178900
1847 DUSP5 Decreases expression PMID:17178900
189 AGXT Increases expression PMID:16648578
1891 ECH1 Increases expression PMID:23292798
19 ABCA1 Increases expression PMID:25932594
1910 EDNRB Increases expression PMID:16648578
19349 RAB7 Increases expression PMID:16648578
1950 EGF Increases expression PMID:16648578
1960 EGR3 Decreases expression PMID:17178900
1962 EHHADH Increases expression PMID:16648578; PMID:17630414
1969 EPHA2 Decreases expression PMID:17178900
197 AHSG Decreases expression PMID:16648578
2023 ENO1 Increases expression PMID:16648578
20249 SCD1 Increases expression PMID:17178900; PMID:17630414; PMID:23292798
20250 SCD2 Increases expression PMID:16648578; PMID:17630414
2052 EPHX1 Increases expression PMID:23292798
2053 EPHX2 Increases expression PMID:23292798
20716 SERPINA3N Decreases expression PMID:16648578
2099 ESR1 Decreases expression PMID:17849452
2100 ESR2 Decreases activity PMID:25752796
2147 F2 Decreases expression PMID:16648578
2167 FABP4 Increases expression PMID:21622945; PMID:25932594
2168 FABP1 Decreases expression PMID:16648578
2169 FABP2 Decreases expression PMID:17630414
2180 ACSL1 Increases expression PMID:23292798
2194 FASN Increases expression PMID:16648578; PMID:17630414
221357 GSTA5 Increases expression PMID:23292798
2222 FDFT1 Increases expression PMID:16648578
224 ALDH3A2 Decreases expression PMID:16648578
2243 FGA Decreases expression PMID:16648578
2244 FGB Decreases expression PMID:16648578
226 ALDOA Increases expression PMID:16648578
226143 CYP2C23 Decreases expression PMID:16648578
2266 FGG Decreases expression PMID:16648578
229 ALDOB Decreases expression PMID:16648578
22943 DKK1 Increases expression PMID:17178900
230 ALDOC Increases expression PMID:16648578
2326 FMO1 Decreases expression PMID:16648578
2335 FN1 Increases expression PMID:16648578
23764 MAFF Decreases expression PMID:17178900
24300 CYP2B1 Increases expression PMID:23292798
24303 CYP2D3 Increases expression PMID:16648578
24540 LRE3 Increases expression PMID:16648578
24737 RT1-EC2 Increases expression PMID:16648578
24862 UGT2B Decreases expression PMID:16648578
24895 CYP2A2 Decreases expression PMID:16648578
249 ALPL Increases expression PMID:16648578
24977 RT1-CL Increases expression PMID:16648578
25011 CYP2C12 Decreases expression PMID:16648578
252931 CYP3A18 Decreases expression PMID:16648578
25475 LGALS5 Increases expression PMID:16648578
25642 CYP3A23-3A1 Affects expression PMID:16648578; PMID:16648578; PMID:23292798
25797 QPCT Increases expression PMID:16648578
25915 NDUFAF3 Increases expression PMID:16648578
26063 DECR2 Increases expression PMID:16648578
2617 GARS1 Decreases expression PMID:17178900
2621 GAS6 Decreases expression PMID:16648578
26358 ALDH1A7 Decreases expression PMID:16648578
2638 GC Decreases expression PMID:16648578
2642 GCGR Decreases expression PMID:16648578
2691 GHRH Increases expression PMID:16648578
27044 SND1 Increases expression PMID:16648578
27284 SULT1B1 Decreases expression PMID:16648578
27306 HPGDS Increases expression PMID:16648578
2819 GPD1 Increases expression PMID:23292798
2824 GPM6B Increases expression PMID:17178900
2834 PRLHR Increases expression PMID:16648578
284541 CYP4A22 Increases expression PMID:16648578
2879 GPX4 Increases expression PMID:16648578
288 ANK3 Decreases expression PMID:16648578
2905 GRIN2C Increases expression PMID:17630414
2907 GRINA Increases expression PMID:16648578
2921 CXCL3 Decreases expression PMID:16648578
29229 SPT1 Decreases expression PMID:16648578
29298 CYP2C7 Decreases expression PMID:16648578
294269 RT1-DA Increases expression PMID:16648578
2949 GSTM5 Increases expression PMID:17630414
2998 GYS2 Affects expression PMID:16648578; PMID:23292798
30 ACAA1 Increases expression PMID:17630414
3015 H2AZ1 Decreases expression PMID:16648578
3053 SERPIND1 Decreases expression PMID:16648578
31 ACACA Increases expression PMID:23292798
3148 HMGB2 Decreases expression PMID:16648578
315571 OR8G20B Increases expression PMID:16648578
3169 FOXA1 Increases expression PMID:16648578
3170 FOXA2 Decreases expression PMID:16648578
3240 HP Decreases expression PMID:16648578
3291 HSD11B2 Increases activity PMID:31927052
3291 HSD11B2 Increases expression PMID:31927052
3294 HSD17B2 Decreases expression PMID:16648578
3301 DNAJA1 Decreases expression PMID:16648578
3308 HSPA4 Decreases expression PMID:16648578
3313 HSPA9 Increases expression PMID:16648578
3315 HSPB1 Increases expression PMID:16648578
332 BIRC5 Decreases expression PMID:17849452; PMID:19067706
334 APLP2 Increases expression PMID:16648578
336 APOA2 Affects expression PMID:16648578; PMID:8668150
338 APOB Decreases expression PMID:16648578
3397 ID1 Increases expression PMID:17178900
34 ACADM Increases expression PMID:23292798
341 APOC1 Decreases expression PMID:16648578
345 APOC3 Decreases expression PMID:16648578
3459 IFNGR1 Increases expression PMID:16648578
347 APOD Increases expression PMID:17849452
3479 IGF1 Decreases expression PMID:15591091
3481 IGF2 Increases expression PMID:16648578
3484 IGFBP1 Increases expression PMID:16648578
3485 IGFBP2 Increases expression PMID:16648578; PMID:17630414
3486 IGFBP3 Decreases expression PMID:16648578
3489 IGFBP6 Increases expression PMID:17178900
3491 CCN1 Decreases expression PMID:17178900
351 APP Increases expression PMID:16648578
3565 IL4 Decreases expression PMID:15781672
3600 IL15 Increases expression PMID:17178900
3606 IL18 Decreases expression PMID:16648578
361523 CYP2B2 Increases expression PMID:16648578
3638 INSIG1 Increases expression PMID:16648578
364 AQP7 Decreases expression PMID:16648578
3645 INSRR Increases expression PMID:16648578
3659 IRF1 Increases expression PMID:16648578
367 AR Decreases activity PMID:25752796
367 AR Increases expression PMID:16648578
3679 ITGA7 Decreases expression PMID:16648578
3694 ITGB6 Increases expression PMID:17178900
3699 ITIH3 Decreases expression PMID:16648578
3708 ITPR1 Increases expression PMID:17178900
3713 IVL Decreases expression PMID:8853895
3728 JUP Increases expression PMID:16648578
375 ARF1 Increases expression PMID:16648578
376497 SLC27A1 Increases expression PMID:10777552
38 ACAT1 Increases expression PMID:16648578; PMID:17630414
3827 KNG1 Affects expression PMID:16648578; PMID:17849452
383 ARG1 Decreases expression PMID:16648578
3852 KRT5 Decreases expression PMID:8853895
3861 KRT14 Decreases expression PMID:8853895
3866 KRT15 Increases expression PMID:17178900
3872 KRT17 Decreases expression PMID:17178900
387496 RASL11A Increases expression PMID:16648578
3921 RPSA Increases expression PMID:16648578
3945 LDHB Decreases expression PMID:16648578
3958 LGALS3 Decreases expression PMID:16648578
3991 LIPE Decreases expression PMID:16648578
3998 LMAN1 Decreases expression PMID:16648578
4015 LOX Decreases expression PMID:16648578
4017 LOXL2 Increases expression PMID:17178900
4036 LRP2 Decreases expression PMID:16648578
4060 LUM Decreases expression PMID:16648578
4071 TM4SF1 Increases expression PMID:17178900
4090 SMAD5 Increases expression PMID:17178900
4094 MAF Increases expression PMID:17178900
4129 MAOB Decreases expression PMID:16648578
4131 MAP1B Increases expression PMID:16648578
4133 MAP2 Increases expression PMID:16648578
4139 MARK1 Increases expression PMID:16648578
4199 ME1 Increases expression PMID:16648578; PMID:23292798
4214 MAP3K1 Increases expression PMID:16648578
43 ACHE Decreases expression PMID:16648578
4312 MMP1 Decreases expression PMID:17178900
432 ASGR1 Increases expression PMID:16648578
4323 MMP14 Decreases expression PMID:16648578
43973 LIP1 Decreases expression PMID:16648578
440 ASNS Decreases expression PMID:17178900
4513 COX2 Decreases expression PMID:17178900
4582 MUC1 Increases expression PMID:16648578
472 ATM Increases activity PMID:19067706
476 ATP1A1 Increases expression PMID:16648578
4761 NEUROD2 Increases expression PMID:16648578
481 ATP1B1 Decreases expression PMID:16648578
4843 NOS2 Decreases expression PMID:17849452
4852 NPY Increases expression PMID:17630414
4946 OAZ1 Increases expression PMID:16648578
495 ATP4A Increases expression PMID:16648578
4953 ODC1 Decreases expression PMID:17178900
5004 ORM1 Decreases expression PMID:16648578
5034 P4HB Increases expression PMID:16648578
51 ACOX1 Increases expression PMID:16648578; PMID:23292798
51129 ANGPTL4 Increases expression PMID:21622945
51144 HSD17B12 Increases expression PMID:16648578
51179 HAO2 Decreases expression PMID:17630414
513 ATP5F1D Increases expression PMID:16648578
5138 PDE2A Decreases expression PMID:16648578
51421 AMOTL2 Decreases expression PMID:17178900
5164 PDK2 Increases expression PMID:16648578
5166 PDK4 Increases expression PMID:16648578
5168 ENPP2 Decreases expression PMID:16648578
51703 ACSL5 Increases expression PMID:23292798
5196 PF4 Increases expression PMID:17630414
5241 PGR Decreases activity PMID:25752796
5265 SERPINA1 Decreases expression PMID:16648578
527 ATP6V0C Increases expression PMID:16648578
5291 PIK3CB Increases expression PMID:16648578
5325 PLAGL1 Decreases expression PMID:16648578
5327 PLAT Increases expression PMID:17178900
5329 PLAUR Decreases expression PMID:17178900
5346 PLIN1 Increases expression PMID:25932594
5352 PLOD2 Increases expression PMID:17178900
54150 RDH7 Decreases expression PMID:16648578
54205 CYCS Decreases expression PMID:17178900
5422 POLA1 Increases expression PMID:16648578
5444 PON1 Decreases expression PMID:16648578
5447 POR Increases expression PMID:16648578
54541 DDIT4 Increases expression PMID:17178900
54677 CROT Increases expression PMID:16648578
5516 PPP2CB Increases expression PMID:16648578
5518 PPP2R1A Increases expression PMID:16648578
5538 PPT1 Decreases expression PMID:16648578
5577 PRKAR2B Decreases expression PMID:16648578
55862 ECHDC1 Increases expression PMID:23292798
5621 PRNP Decreases expression PMID:16648578
5623 PSPN Increases expression PMID:16648578
56266 CYP4F1 Decreases expression PMID:16648578
5660 PSAP Increases expression PMID:16648578
56603 CYP26B1 Increases expression PMID:17849452
56902 PNO1 Decreases expression PMID:17178900
5701 PSMC2 Increases expression PMID:16648578
5710 PSMD4 Increases expression PMID:16648578
57142 RTN4 Increases expression PMID:17630414
57175 CORO1B Increases expression PMID:16648578
5733 PTGER3 Decreases expression PMID:17849452
5734 PTGER4 Decreases expression PMID:17849452
57582 KCNT1 Increases expression PMID:16648578
5763 PTMS Increases expression PMID:16648578
5788 PTPRC Increases expression PMID:16648578
581 BAX Increases activity PMID:19067706
581 BAX Increases expression PMID:19067706
5824 PEX19 Decreases expression PMID:16648578
5825 ABCD3 Increases expression PMID:16648578; PMID:23292798
59 ACTA2 Increases expression PMID:16648578
59088 PRL8A4 Increases expression PMID:16648578
5915 RARB Increases expression PMID:17178900; PMID:35483669
595 CCND1 Affects expression PMID:16648578; PMID:17178900
5973 RENBP Increases expression PMID:16648578
5978 REST Increases expression PMID:16648578
6035 RNASE1 Increases expression PMID:16648578
6130 RPL7A Increases expression PMID:16648578
6142 RPL18A Increases expression PMID:16648578
6146 RPL22 Increases expression PMID:16648578
6187 RPS2 Increases expression PMID:16648578
619412 NEDD4A Increases expression PMID:16648578
6256 RXRA Increases activity PMID:21218783
6258 RXRG Decreases expression PMID:17849452
6280 S100A9 Increases expression PMID:16648578; PMID:17178900
6281 S100A10 Decreases expression PMID:16648578
6285 S100B Decreases expression PMID:16648578
6289 SAA2 Increases expression PMID:16648578
6319 SCD Increases expression PMID:17178900; PMID:32123961
6342 SCP2 Decreases expression PMID:16648578
6356 CCL11 Decreases expression PMID:16648578
6383 SDC2 Decreases expression PMID:16648578
641371 ACOT1 Increases expression PMID:16648578; PMID:17630414
6421 SFPQ Decreases expression PMID:16648578
6427 SRSF2 Decreases expression PMID:17178900
644076 GLYCAM1 Increases expression PMID:16648578
6469 SHH Increases expression PMID:26096596
6478 SIAH2 Decreases expression PMID:17178900
6507 SLC1A3 Decreases expression PMID:16648578
6514 SLC2A2 Increases expression PMID:16648578
6533 SLC6A6 Increases expression PMID:16648578
6541 SLC7A1 Decreases expression PMID:17178900
6623 SNCG Decreases expression PMID:16648578
663 BNIP2 Decreases expression PMID:17178900
6652 SORD Decreases expression PMID:16648578
6675 UAP1 Decreases expression PMID:17178900
6678 SPARC Increases expression PMID:17178900
6690 SPINK1 Increases expression PMID:16648578
6694 SPP2 Decreases expression PMID:16648578
6696 SPP1 Decreases expression PMID:16648578
6715 SRD5A1 Decreases expression PMID:16648578
6720 SREBF1 Increases expression PMID:23292798; PMID:32123961
6817 SULT1A1 Decreases expression PMID:16648578
6822 SULT2A1 Decreases expression PMID:16648578
685222 CYP2B15 Increases expression PMID:16648578
6865 TACR2 Increases expression PMID:16648578
687 KLF9 Affects expression PMID:16648578; PMID:26096596
70 ACTC1 Increases expression PMID:16648578
7018 TF Increases expression PMID:16648578
7038 TG Increases expression PMID:16648578
7043 TGFB3 Increases expression PMID:16648578
7051 TGM1 Decreases expression PMID:8853895
7052 TGM2 Increases expression PMID:17178900; PMID:21622945; PMID:25932594
7067 THRA Decreases activity PMID:25752796
7071 KLF10 Decreases expression PMID:17178900
71 ACTG1 Increases expression PMID:16648578
713 C1QB Increases expression PMID:16648578
7132 TNFRSF1A Increases expression PMID:16648578
7145 TNS1 Increases expression PMID:16648578
7157 TP53 Increases activity PMID:19067706
7161 TP73 Increases expression PMID:19067706
7168 TPM1 Increases expression PMID:16648578
7170 TPM3 Increases expression PMID:16648578
7171 TPM4 Increases expression PMID:16648578
718 C3 Decreases expression PMID:16648578
722 C4BPA Decreases expression PMID:16648578
7276 TTR Decreases expression PMID:16648578
7422 VEGFA Increases expression PMID:16648578
7494 XBP1 Decreases expression PMID:17178900
7533 YWHAH Decreases expression PMID:16648578
7704 ZBTB16 Increases expression PMID:23292798
7784 ZP3 Increases expression PMID:16648578
7786 MAP3K12 Increases expression PMID:16648578
7832 BTG2 Decreases expression PMID:16648578
7846 TUBA1A Increases expression PMID:16648578
79365 BHLHE41 Decreases expression PMID:16648578
79874 RABEP2 Increases expression PMID:16648578
8001 GLRA3 Increases expression PMID:16648578
811 CALR Increases expression PMID:16648578
8140 SLC7A5 Decreases expression PMID:17178900
818 CAMK2G Increases expression PMID:16648578
821 CANX Increases expression PMID:16648578
8292 COLQ Increases expression PMID:16648578
8303 SNN Decreases expression PMID:16648578
836 CASP3 Decreases expression PMID:17849452
839 CASP6 Decreases expression PMID:16648578
8431 NR0B2 Increases expression PMID:17630414; PMID:23292798; PMID:32123961
84879 MFSD2A Decreases expression PMID:17630414
8503 PIK3R3 Increases expression PMID:16648578
8522 GAS7 Increases expression PMID:16648578
8644 AKR1C3 Increases expression PMID:17178900
8647 ABCB11 Increases expression PMID:16648578
8663 EIF3C Decreases expression PMID:17630414
8673 VAMP8 Increases expression PMID:17178900
871 SERPINH1 Increases expression PMID:17630414
873 CBR1 Increases expression PMID:16648578
8775 NAPA Increases expression PMID:16648578
8811 GALR2 Increases expression PMID:16648578
8824 CES2 Increases expression PMID:16648578; PMID:17630414
8864 PER2 Decreases expression PMID:17178900
8878 SQSTM1 Increases expression PMID:16648578
891 CCNB1 Decreases expression PMID:19067706
898 CCNE1 Decreases expression PMID:17849452
9027 NAT8 Decreases expression PMID:17630414
9104 RGN Decreases expression PMID:16648578
9133 CCNB2 Decreases expression PMID:17849452
9230 RAB11B Increases expression PMID:16648578
9249 DHRS3 Increases expression PMID:17178900
929 CD14 Increases expression PMID:16648578
93 ACVR2B Increases expression PMID:16648578
9391 CIAO1 Decreases expression PMID:16648578
9415 FADS2 Increases expression PMID:17630414
9452 ITM2A Increases expression PMID:17178900
9456 HOMER1 Increases expression PMID:16648578
948 CD36 Increases expression PMID:16648578; PMID:23292798
951 CD37 Increases expression PMID:16648578
9524 TECR Increases expression PMID:16648578
9527 GOSR1 Increases expression PMID:16648578
9547 CXCL14 Decreases expression PMID:16648578
9588 PRDX6 Increases expression PMID:16648578
9590 AKAP12 Increases expression PMID:16648578
9592 IER2 Decreases expression PMID:17178900
9709 HERPUD1 Decreases expression PMID:17178900
972 CD74 Increases expression PMID:16648578
983 CDK1 Decreases expression PMID:19067706
9970 NR1I3 Increases activity PMID:31312845
9970 NR1I3 Increases expression PMID:17630414

DISCLAIMER

We have built a comprehensive resource which compiles potential endocrine disrupting chemicals (EDCs) based on the observed adverse effects or endocrine-mediated endpoints in published experiments on humans or rodents to support basic research. We are not responsible for any errors or omissions in the published research articles or supporting literature on potential EDCs compiled in this resource. Users are advised to exercise their own judgement on the weight of evidence for potential EDCs compiled in this resource. Importantly, our sole goal to build this resource on potential EDCs is to enable future basic research towards better understanding of the systems-level perturbations upon chemical exposure rather than influencing regulatory advice on chemical use.