| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Neuronal acetylcholine receptor; alpha2/beta2 | Rattus norvegicus | P12390 | | | | = 18000.0 nM | NPASS |
| Neuronal acetylcholine receptor; alpha4/beta2 | Rattus norvegicus | P12390 | | | | = 37000.0 nM | NPASS |
| Neuronal acetylcholine receptor; alpha3/beta2 | Rattus norvegicus | P12390 | | | | = 37000.0 nM | NPASS |
| Neuronal acetylcholine receptor; alpha3/beta4 | Rattus norvegicus | P12392 | | | | = 48000.0 nM | NPASS |
| Neuronal acetylcholine receptor; alpha4/beta4 | Rattus norvegicus | P12392 | | | | = 34000.0 nM | NPASS |
| Solute carrier family 22 member 2 | Mus musculus | O70577 | | 217000 nM|= 217000.0 nM | | | BindingDB, NPASS |
| Sodium- and chloride-dependent creatine transporter 1 | Rattus norvegicus | P28570 | | | | 42000 nM | BindingDB |
| Solute carrier family 22 member 1 | Mus musculus | O08966 | | 55000 nM|= 55000.0 nM | | | BindingDB, NPASS |
| Solute carrier family 22 member 1 | Rattus norvegicus | Q63089 | | 1452000 nM|398000 nM|= 1452000.0 nM|= 398000.0 nM | | | BindingDB, NPASS |
| Solute carrier family 22 member 2 | Rattus norvegicus | Q9R0W2 | | 1450000 nM|159000 nM|= 1450000.0 nM|= 159000.0 nM | | | BindingDB, NPASS |
| Neuronal acetylcholine receptor subunit alpha-4/beta-4 | Rattus norvegicus | P09483|P12392 | | | | 34000 nM | BindingDB |
| Nicotinic acetylcholine receptor | Rattus leucopus | | | | | >10000 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-4/beta-2 | Rattus norvegicus | P09483|P12390 | | | | 37000 nM | BindingDB |
| Acetylcholinesterase | Tetronarce californica | P04058 | | 3010000 nM | | | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-4 | Homo sapiens | P43681 | | | | 7000 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-3/beta-4 | Rattus norvegicus | P04757|P12392 | | | | 48000 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-3/beta-2 | Rattus norvegicus | P04757|P12390 | | | | 37000 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-3 | Rattus norvegicus | P04757 | | | | >10000 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-2/beta-2 | Rattus norvegicus | P12389|P12390 | | | | 18000 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-2 | Rattus norvegicus | P12389 | | | | >10000 nM | BindingDB |
| Neuronal acetylcholine receptor | Rattus norvegicus | Q05941 | | | | = 42000.0 nM | NPASS |
| High affinity choline transporter 1 | Mus musculus | Q8BGY9 | | 1600 nM | | 680.77 nM | BindingDB |
| Creatine transporter | Rattus norvegicus | P28570 | | | | = 42000.0 nM | NPASS |
| Choline transporter | Mus musculus | Q8BGY9 | | = 1600.0 nM | | | NPASS |
| Choline O-acetyltransferase | Rattus norvegicus | P32738 | | | | 7600000 nM|400000 nM | BindingDB |
| Acetylcholinesterase | Homo sapiens | P22303 | | 3013006.02 nM|= 3013006.02 nM | | | BindingDB, NPASS |
| Neuronal acetylcholine receptor subunit alpha-4 | Rattus norvegicus | P09483 | | | | >10000 nM | BindingDB |