| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Microtubule-associated protein tau | Homo sapiens | P10636 | | >= 200000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 1590.0 nM|= 18300.0 nM|= 22.22 ug.mL-1|> 50.0 ug.mL-1|= 1.83 ug.mL-1|= 47370.0 nM | | | NPASS |
| Mitogen-activated protein kinase 14 | Homo sapiens | Q16539 | | 6.76e+4 nM | | | BindingDB |
| Mitogen-activated protein kinase 10 | Homo sapiens | P53779 | | 8.95e+4 nM | | | BindingDB |
| Nitric oxide synthase, endothelial | Bos taurus | P29473 | 2.0 nM | | | | BindingDB |
| Intestinal-type alkaline phosphatase | Homo sapiens | P09923 | >100000 nM | | | | BindingDB |
| L929 | Mus musculus | | = 300000.0 nM|= 350000.0 nM | | | | NPASS |
| M18 aspartyl aminopeptidase | Plasmodium falciparum (isolate 3D7) | | | 1376 nM | | | BindingDB |
| Liver microsomes | Rattus norvegicus | | | = 25000000.0 nM | | | NPASS |
| Liver microsome | Rattus norvegicus | | | = 29.0 ug.mL-1 | | | NPASS |
| LNCaP | Homo sapiens | | = 13000.0 nM | | | | NPASS |
| Intestinal-type alkaline phosphatase 1 | Rattus norvegicus | P15693 | | 1360 nM | | | BindingDB |
| Nitric-oxide synthase, endothelial | Bos taurus | P29473 | = 2.0 nM | | | | NPASS |
| M18 aspartyl aminopeptidase | Plasmodium falciparum 3D7 | Q8I2J3 | | = 1376.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | > 500000.0 nM | | | NPASS |
| U373 MG | Homo sapiens | | | > 500000.0 nM | | | NPASS |
| Procathepsin L | Homo sapiens | P07711 | | >59642 nM | | | BindingDB |
| Intestinal alkaline phosphatase | Mus musculus | P24822 | | = 1360.0 nM | | | NPASS |
| Xanthine dehydrogenase/oxidase | Homo sapiens | P47989 | | >100000 nM | | | BindingDB |
| Xanthine dehydrogenase | Homo sapiens | P47989 | | > 100000.0 nM | | | NPASS |
| Vero | Chlorocebus aethiops | | | = 184100.0 nM | | | NPASS |
| Trypanosoma brucei brucei | Trypanosoma brucei brucei | | | < 30000.0 nM | | | NPASS |
| Thrombin | Homo sapiens | P00734 | | = 150000.0 nM | = 5190000.0 nM | | NPASS |
| Sucrase-isomaltase, intestinal | Rattus norvegicus | P23739 | | 650000 nM | | | BindingDB |
| Sucrase-isomaltase | Rattus norvegicus | P23739 | | = 650000.0 nM | | | NPASS |
| SK-OV-3 | Homo sapiens | | | > 500000.0 nM | | | NPASS |
| Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | | | >100000 nM | | | BindingDB |
| Radical scavenging activity | | | | = 8.5 ug.mL-1|= 49000.0 nM|= 1.7 ug.mL-1|= 1.61 ug.mL-1 | | | NPASS |
| Pyruvate kinase isozymes M1/M2 | Homo sapiens | P14618 | | = 1330.0 nM | | | NPASS |
| Prothrombin | Homo sapiens | P00734 | | 150000 nM | 5190000 nM | | BindingDB |
| Protein RecA | Mycobacterium tuberculosis | P9WHJ3 | > 380000.0 nM | | | | NPASS |
| Prostaglandin G/H synthase 1 | Ovis aries | P05979 | | 12200 nM|2000 nM | 25900 nM | | BindingDB |
| Plasmodium falciparum | Plasmodium falciparum | | | > 150000.0 nM|> 50000.0 nM | | | NPASS |
| Intestinal alkaline phosphatase | Homo sapiens | P09923 | > 100000.0 nM | | | | NPASS |
| DLD-1 | Homo sapiens | | | > 25000.0 nM|= 415000.0 nM | | | NPASS |
| Human immunodeficiency virus | Human immunodeficiency virus | | | = 34.1 ug.mL-1 | | | NPASS |
| Human immunodeficiency virus type 1 reverse transcriptase | Human immunodeficiency virus 1 | Q72547 | | > 100000.0 nM | | | NPASS |
| 6-phosphogluconate dehydrogenase | Homo sapiens | P52209 | | > 1000000.0 nM | | | NPASS |
| 6-phosphogluconate dehydrogenase, decarboxylating | Homo sapiens | P52209 | | >1000000 nM | | | BindingDB |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus | P07943 | | >30000 nM | | | BindingDB |
| Aldose reductase | Rattus norvegicus | P07943 | | > 30000.0 nM | | | NPASS |
| Alkaline phosphatase placental-like | Homo sapiens | P10696 | = 51300.0 nM | | | | NPASS |
| Alkaline phosphatase, germ cell type | Homo sapiens | P10696 | 51300 nM | | | | BindingDB |
| Alpha-amylase 1A | Homo sapiens | P0DUB6 | | | | | BindingDB |
| Alpha-synuclein | Homo sapiens | P37840 | | 29900 nM|800 nM|= 29900.0 nM|= 800.0 nM | | | BindingDB, NPASS |
| Amyloid-beta A4 protein | Homo sapiens | P05067 | | = 5300.0 nM | | | NPASS |
| Anthrax toxin receptor 2 | Homo sapiens | P58335 | | >300000 nM|> 300000.0 nM | | | BindingDB, NPASS |
| Apoptosis regulator Bcl-2 | Homo sapiens | P10415 | | | | >100000 nM|> 100000.0 nM | BindingDB, NPASS |
| Arginase | Leishmaamazonensis | | | 1600 nM | | 200 nM | BindingDB |
| Arginase | Leishmaamazonensis | O96394 | | = 1600.0 nM | | = 200.0 nM | NPASS |
| Beta-secretase 1 | Homo sapiens | P56817 | | = 4500.0 nM | | | NPASS |
| Alkaline phosphatase, tissue-nonspecific isozyme | Homo sapiens | P05186 | | 407 nM|= 407.0 nM | | | BindingDB, NPASS |
| Carbonic anhydrase 1 | Homo sapiens | P00915 | | | | 2.32e+3 nM | BindingDB |
| HeLa | Homo sapiens | | | > 25000.0 nM | | | NPASS |
| Candida albicans | Candida albicans | | | > 50.0 ug.mL-1 | | | NPASS |
| Glucose-6-phosphate 1-dehydrogenase | Saccharomyces cerevisiae S288c | P11412 | | > 1000000.0 nM | | | NPASS |
| Glucose-6-phosphate 1-dehydrogenase | Saccharomyces cerevisiae (strain ATCC 204508 / S288c) | P11412 | | >1000000 nM | | | BindingDB |
| Giardia intestinalis | Giardia intestinalis | | | = 1.0 ug.mL-1 | | | NPASS |
| Fatty acid synthase | Homo sapiens | P49327 | | >100000 nM|> 100000.0 nM | | | BindingDB, NPASS |
| Entamoeba histolytica | Eoeba histolytica | | | = 1.92 ug.mL-1 | | | NPASS |
| Filobasidiella neoformans | Cryptococcus neoformans | | | > 50.0 ug.mL-1 | | | NPASS |
| DNA polymerase beta | Rattus norvegicus | P06766 | | 18500 nM|= 18500.0 nM | | | BindingDB, NPASS |
| Cyclooxygenase-1 | Ovis aries | P05979 | | = 2000.0 nM|= 12200.0 nM | = 25900.0 nM | | NPASS |
| Cathepsin L | Homo sapiens | P07711 | | > 59642.0 nM | | | NPASS |
| Carbonic anhydrase 6 | Human | P23280 | | | | 4.36e+3 nM | BindingDB |
| Carbonic anhydrase 4 | Homo sapiens | P22748 | | | | 3.98e+3 nM | BindingDB |
| Carbonic anhydrase 3 | Bovine | Q3SZX4 | | | | 8.93e+3 nM | BindingDB |
| Carbonic anhydrase 2 | Homo sapiens | P00918 | | | | 1.24e+3 nM | BindingDB |