| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Muscarinic acetylcholine receptor M4 | Homo sapiens | P08173 | | | | >10000 nM | BindingDB |
| Muscarinic acetylcholine receptor M5 | Homo sapiens | P08912 | | | | 35.13 nM | BindingDB |
| N9 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | = 109630.0 nM | = 10600.0 nM|> 164000.0 nM|= 4.65 ug.mL-1|= 19400.0 nM|= 10106700.0 nM|= 7794400.0 nM|= 4700.0 nM | | | NPASS |
| Neuraminidase | InflueA virus (A/WSN/1933(H1N1)) | P03470 | | 87700 nM|>100000 nM|52200 nM | | | BindingDB |
| Neuraminidase | InflueA virus (A/Puerto Rico/8/1934(H1N1)) | P03468 | | = 31.14 ug.mL-1 | | | NPASS |
| Neuraminidase | InflueA virus (strain A/Puerto Rico/8/1934 H1N1) | P03468 | | 50700 nM|51000 nM | | | BindingDB |
| Muscarinic acetylcholine receptor M3 | Homo sapiens | P20309 | | | | >10000 nM | BindingDB |
| Neuraminidase | InflueA virus (strain A/USSR/90/1977 H1N1) | P03469 | | 95900 nM|96800 nM|= 95900.0 nM|= 96800.0 nM | | | BindingDB, NPASS |
| Neuraminidase | InflueA virus | B4URF0 | | = 52200.0 nM|= 87700.0 nM|> 100000.0 nM|= 34400.0 nM | | = 33800.0 nM | NPASS |
| Muscarinic acetylcholine receptor M2 | Homo sapiens | P08172 | | | | >10000 nM | BindingDB |
| Leishmania amazonensis | Leishmaamazonensis | | | = 4400.0 nM | | | NPASS |
| Mu-type opioid receptor | Homo sapiens | P35372 | | | | >10000 nM | BindingDB |
| Monoamine oxidase A | Homo sapiens | P21397 | | = 3890.0 nM | | | NPASS |
| Mitogen-activated protein kinase 14 | Homo sapiens | Q16539 | | 6.59e+4 nM | | | BindingDB |
| Meloidogyne incognita | Meloidogyne incognita | | > 1000.0 ug.mL-1 | | | | NPASS |
| Lysine-specific histone demethylase 1A | Homo sapiens | O60341 | | 2160 nM | | | BindingDB |
| Lysine-specific histone demethylase 1 | Homo sapiens | O60341 | | = 2160.0 nM | | | NPASS |
| Leishmania donovani | Leishmadonovani | | | = 49140.0 nM | | | NPASS |
| L929 | Mus musculus | | = 250000.0 nM|> 250000.0 nM | > 100000.0 nM | | | NPASS |
| L-lactate dehydrogenase A chain | Homo sapiens | P00338 | | >500000 nM|> 500000.0 nM | | | BindingDB, NPASS |
| Kappa-type opioid receptor | Homo sapiens | P41145 | | | | >10000 nM | BindingDB |
| Neuromedin-U receptor 2 | Homo sapiens | Q9GZQ4 | 1200 nM|= 1200.0 nM | | | | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M1 | Homo sapiens | P11229 | | | | >10000 nM | BindingDB |
| No relevant target | | | | = 2.5 ug.mL-1 | | | NPASS |
| Tyrosinase | Homo sapiens | P14679 | | = 0.856 ug.mL-1 | | | NPASS |
| Nonstructural protein 5 | Dengue virus | V5TFZ2 | | = 2100.0 nM | | | NPASS |
| n.a. | | | | = 1170.0 nM|= 2530.0 nM|= 4700.0 nM | | | NPASS |
| Xanthine dehydrogenase/oxidase | Homo sapiens | P47989 | | 52200 nM | | | BindingDB |
| Xanthine dehydrogenase | Homo sapiens | P47989 | | = 52200.0 nM | | | NPASS |
| Verticillium dahliae | Verticillium dahliae | | | = 80.0 ug.mL-1 | | | NPASS |
| Vasopressin V2 receptor | Homo sapiens | P30518 | | | | >10000 nM | BindingDB |
| Vasopressin V1b receptor | Homo sapiens | P47901 | | | | >10000 nM | BindingDB |
| K562 | Homo sapiens | | | = 897000.0 nM | | | NPASS |
| Tyrosinase | Agaricus bisporus | O42713 | | = 70000.0 nM|= 130000.0 nM | | | NPASS |
| Trypsin | Homo sapiens | P35030 | | = 16000.0 nM | | = 17500.0 nM | NPASS |
| Trypsin | Homo sapiens | P07477|P07478|P35030 | | 16000 nM | | 17500 nM | BindingDB |
| Trypanosoma cruzi | Trypanosoma cruzi | | | = 49140.0 nM | | | NPASS |
| Trypanosoma brucei rhodesiense | Trypanosoma brucei rhodesiense | | | = 6900.0 nM | | | NPASS |
| Solute carrier organic anion transporter family member 2B1 | Homo sapiens | O94956 | | = 138038.43 nM|= 136900.0 nM | | | NPASS |
| Sodium-dependent serotonin transporter | Homo sapiens | P31645 | | | | >10000 nM | BindingDB |
| Sodium-dependent noradrenaline transporter | Homo sapiens | P23975 | | | | >10000 nM | BindingDB |
| Sodium-dependent dopamine transporter | Bos taurus | P27922 | | | | >10000 nM | BindingDB |
| Serum albumin | Bos taurus | P02769 | | = 41900.0 nM | | | NPASS |
| SK-OV-3 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| SK-MEL-2 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Radical scavenging activity | | | = 4.8 ug|= 15.5 ug | = 12340.0 nM|= 12300.0 nM|= 1.83 ug.mL-1|= 38700.0 nM|= 4700.0 nM | | | NPASS |
| RAW264.7 | Mus musculus | | | = 15070.0 nM|= 27500.0 nM|= 44500.0 nM | | | NPASS |
| Prolyl endopeptidase | Homo sapiens | P48147 | | > 200000.0 nM | | | NPASS |
| Polyphenol oxidase 2 | Agaricus bisporus | O42713 | | 70000 nM|130000 nM | | | BindingDB |
| Nonstructural protein 3 | Zika virus | | | 104000 nM | | | BindingDB |
| Histamine H1 receptor | Rattus norvegicus | P31390 | | | | >10000 nM | BindingDB |
| Sialidase | Clostridium perfringens | P10481 | | 30900 nM|= 30900.0 nM | | | BindingDB, NPASS |
| Glutamate receptor ionotropic, NMDA 1 | Rattus norvegicus | P35439 | | | | >10000 nM | BindingDB |
| BV-2 | Mus musculus | | | = 24290.0 nM | | | NPASS |
| BT-549 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Alpha-chymotrypsin | Bos taurus | P00766 | | = 296000.0 nM|= 281000.0 nM | | | NPASS |
| Alpha-2c adrenergic receptor | Homo sapiens | P18825 | | | | = 9637.0 nM | NPASS |
| Alpha-2a adrenergic receptor | Homo sapiens | P08913 | | | | = 9340.0 nM | NPASS |
| Alpha-2C adrenergic receptor | Homo sapiens | P18825 | | | | 9637 nM | BindingDB |
| Alpha-2B adrenergic receptor | Homo sapiens | P18089 | | | | >10000 nM | BindingDB |
| Alpha-2A adrenergic receptor | Homo sapiens | P08913 | | | | 9340 nM | BindingDB |
| Alpha-1B adrenergic receptor | Homo sapiens | P35368 | | | | >10000 nM | BindingDB |
| Alpha-1A adrenergic receptor | Homo sapiens | P35348 | | | | >10000 nM | BindingDB |
| Aldose reductase | Rattus norvegicus | P07943 | | = 13000.0 nM | | | NPASS |
| Aldose reductase | Homo sapiens | P15121 | | = 294500.0 nM | | | NPASS |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus | P07943 | | 13000 nM | | | BindingDB |
| Albumin | Bos taurus | P02769 | | 41900 nM | | | BindingDB |
| Acetylcholinesterase | Homo sapiens | P22303 | | 12 nM|= 12.0 nM|= 113300.0 nM | | >300000 nM|> 300000.0 nM | BindingDB, NPASS |
| A549 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| 5-hydroxytryptamine receptor 7 | Homo sapiens | P34969 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 6 | Homo sapiens | P50406 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 5A | Homo sapiens | P47898 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 3A | Homo sapiens | P46098 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 1D | Homo sapiens | P28221 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 1A | Homo sapiens | P08908 | | | | >10000 nM | BindingDB |
| Glycogen synthase kinase-3 beta | Homo sapiens | P49841 | 27960 nM | | | | BindingDB |
| Beta-1 adrenergic receptor | Rattus norvegicus | P18090 | | | | >10000 nM | BindingDB |
| Beta-2 adrenergic receptor | Rattus norvegicus | P10608 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 2C | Rattus norvegicus | P08909 | | | | >10000 nM | BindingDB |
| Beta-secretase 1 | Homo sapiens | P56817 | | = 3.8 nM | | | NPASS |
| Giardia intestinalis | Giardia intestinalis | | | = 178.7 ug.mL-1 | | | NPASS |
| Beta-lactamase | Enterobacter cloacae | P05364 | | >500000 nM|> 500000.0 nM | | | BindingDB, NPASS |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus | P62813 | | | | >10000 nM | BindingDB |
| Filobasidiella neoformans | Cryptococcus neoformans | | | = 30.0 ug.mL-1 | | | NPASS |
| Epoxide hydratase | Homo sapiens | P34913 | | = 24300.0 nM | | | NPASS |
| Entamoeba histolytica | Eoeba histolytica | | | = 119.7 ug.mL-1|= 120.7 ug.mL-1 | | | NPASS |
| Dipeptidyl peptidase IV | Homo sapiens | P27487 | | = 145000.0 nM | | | NPASS |
| Dihydroorotate dehydrogenase (fumarate) | Leishmamajor | Q4QEW7 | | = 1531000.0 nM|= 1584893.19 nM | | | NPASS |
| Dihydroorotate dehydrogenase (fumarate) | Leishmamajor | | | 1584893 nM|1531000 nM | | | BindingDB |
| Dengue virus | Dengue virus | | | = 1700.0 nM | | | NPASS |
| Delta-type opioid receptor | Sus scrofa | P79291 | | | | >10000 nM | BindingDB |
| D(4) dopamine receptor | Rattus norvegicus | P30729 | | | | >10000 nM | BindingDB |
| Genome polyprotein | Zika virus | A0A024AXB9 | | = 104000.0 nM | | | NPASS |
| D(2) dopamine receptor | Rattus norvegicus | P61169 | | | | >10000 nM | BindingDB |
| D(3) dopamine receptor | Rattus norvegicus | P19020 | | | | >10000 nM | BindingDB |
| Bifunctional epoxide hydrolase 2 | Homo sapiens | P34913 | | 24300 nM | | | BindingDB |
| Candida albicans | Candida albicans | | | > 50.0 ug.mL-1 | | | NPASS |
| Cholinesterase | Homo sapiens | P06276 | | | | 501200 nM | BindingDB |
| Chymotrypsinogen A | Bos taurus | P00766 | | 281000 nM|296000 nM | | | BindingDB |
| Butyrylcholinesterase | Homo sapiens | P06276 | | | | = 501200.0 nM | NPASS |
| Cytochrome P450 3A4 | Homo sapiens | P08684 | | >80000 nM|> 80000.0 nM | | | BindingDB, NPASS |
| D(1A) dopamine receptor | Homo sapiens | P21728 | | | | >10000 nM | BindingDB |
| D(1B) dopamine receptor | Homo sapiens | P21918 | | | | >10000 nM | BindingDB |
| Cystic fibrosis transmembrane conductance regulator | Homo sapiens | P13569 | | | 65800 nM|= 65800.0 nM | | BindingDB, NPASS |