| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Neuronal acetylcholine receptor subunit alpha-7 | Homo sapiens | P36544 | 740 nM|38000 nM|83000 nM|113000 nM|91000 nM|1584.89 nM|4710 nM | 7600 nM|21000 nM | 1.06 nM | 2000 nM|1610 nM|620 nM|7200 nM|6300 nM|630 nM|12000 nM|24000 nM|2110 nM|3000 nM|1000 nM|1023.29 nM|3800 nM|6290 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-7 | Mus musculus | P49582 | | | | 480 nM|244 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-7 | Rattus norvegicus | Q05941 | 54000 nM|13000 nM|109648 nM|108700 nM|43000000 nM|1500 nM|1071.52 nM|23000 nM|47000 nM | 16 nM | | 130 nM|>10000 nM|668 nM|170 nM|517 nM|4000 nM|610 nM|770 nM|15000 nM|450 nM|234 nM|250 nM|480 nM|460 nM|469 nM|1400 nM|340 nM|1748 nM|6290 nM|750 nM|16000 nM|176 nM|230 nM|400 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-9 | Rattus norvegicus | P43144 | | 2.4 nM | 5 nM | 1000 nM | BindingDB |
| Neuronal acetylcholine receptor; alpha2/beta4 | Rattus norvegicus | P12392 | | | | = 112.0 nM|= 110.0 nM|= 70.0 nM | NPASS |
| Neuronal acetylcholine receptor; alpha2/beta2 | Homo sapiens | Q15822 | | | | = 5.5 nM | NPASS |
| Neuronal acetylcholine receptor; alpha2/beta2 | Rattus norvegicus | P12390 | | | | = 15.0 nM|= 12.0 nM|= 5.5 nM | NPASS |
| Neuronal acetylcholine receptor; alpha2/beta4 | Homo sapiens | Q15822 | | | | = 103.0 nM|= 70.0 nM | NPASS |
| Neuronal acetylcholine receptor; alpha3/alpha6/beta2/beta3 | Homo sapiens | Q05901 | = 127.0 nM | = 84.8 nM | | | NPASS |
| Neuronal acetylcholine receptor subunit alpha-6/beta-3 | Rattus norvegicus | | | | | = 3.3 nM | NPASS |
| Neuronal acetylcholine receptor subunit beta-4 | Rattus norvegicus | P12392 | | | | 73 nM|= 73.0 nM | BindingDB, NPASS |
| Neuronal acetylcholine receptor subunit alpha-6 | Gallus gallus | P49581 | | | | 20 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-4 | Mus musculus | O70174 | | 7.0 nM | | | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-4/beta-4 | Rattus norvegicus | P09483|P12392 | | | | 40 nM|46 nM|72 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-4/beta-4 | Homo sapiens | P30926|P43681 | 7100 nM | | | 129 nM|23 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-4/beta-2 | Rattus norvegicus | P09483|P12390 | 4000 nM|590 nM|1000 nM|7.3 nM|10000 nM|14000 nM|591 nM|77 nM|19000 nM | 3.8 nM | | 1.4 nM|1 nM|1.3 nM|12 nM|10 nM|0.84 nM|1.5 nM|1.1 nM|10.00 nM|9.8 nM|6.8 nM|3 nM|2.3 nM|2 nM|4.0 nM|11.1 nM|1.26 nM|1.01 nM|8.0 nM|0.940000 nM|10.0 nM|35 nM|2.0 nM|1.8 nM|2.8 nM|13 nM|14 nM|4.1 nM|11 nM|5.6 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-4/beta-2 | Mus musculus | | = 720.0 nM|= 724.44 nM | | | | NPASS |
| Neuronal acetylcholine receptor subunit alpha-4/beta-2 | Mus musculus | O70174|Q9ERK7 | 724 nM|720 nM | | | | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-4/beta-2 | Human | P17787|P43681 | 2400 nM | 370 nM | | 10 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-4/beta-2 | Homo sapiens | P17787|P43681 | 2100 nM|4000 nM|5000 nM|290 nM|1 nM|3000 nM|295.12 nM|295 nM|9400 nM|6600 nM|300 nM|2400 nM|800 nM | 430 nM|427 nM|426.58 nM|370 nM|1.2 nM|4.9 nM | | 8.60 nM|2.3 nM|1.2 nM|2.1 nM|2 nM|9.1 nM|4.9 nM|4 nM|1.5 nM|5.5 nM|1.6 nM|>10000 nM|9.46 nM|12.59 nM|0.600000 nM|2.0 nM|10.0 nM|0.045000 nM|1.1 nM|2.2 nM|1.000000 nM|<1.000000 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-4 | Rattus norvegicus | P09483 | | 1.65 nM | | >10000 nM|1 nM|0.84 nM|8.3 nM|74 nM|10 nM|40 nM|1.5 nM|7 nM|4 nM|6.0 nM|0.94 nM|22 nM|150 nM | BindingDB |
| Neuronal acetylcholine receptor; alpha3/beta2 | Homo sapiens | P32297 | = 132000.0 nM | = 3.8 nM | | = 47.0 nM|= 29.0 nM | NPASS |
| Neuronal acetylcholine receptor subunit alpha-4 | Homo sapiens | P43681 | 4700 nM|6600 nM | | | 1.05 nM|26.25 nM|1 nM|6690 nM|4.9 nM|7.7 nM|4.6 nM|2 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-4 | Gallus gallus | P09482 | | | | 1.9 nM|= 1.9 nM | BindingDB, NPASS |
| Neuronal acetylcholine receptor subunit alpha-3/beta-4 | Rattus norvegicus | P04757|P12392 | 86000 nM|24000 nM|35000 nM|1514 nM|1500 nM | >10000 nM | | 443 nM|530 nM|481 nM|440 nM|290 nM|288 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-3/beta-4 | Rat | P04757|P12392 | 23000 nM | >10000 nM | | 440 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-5 | Rattus norvegicus | P20420 | | | | 156 nM | BindingDB |
| Neuronal acetylcholine receptor; alpha3/beta2 | Rattus norvegicus | P12390 | | | | = 43.0 nM|= 1.0 nM|= 47.0 nM|= 29.0 nM | NPASS |
| Nicotinic acetylcholine receptor alpha 5 subunit | Musca domestica | | | 11900 nM | | | BindingDB |
| Neuronal acetylcholine receptor; alpha3/beta4 | Rattus norvegicus | P12392 | = 86000.0 nM|= 35000.0 nM|= 23000.0 nM|= 24000.0 nM|= 1500.0 nM|= 1513.56 nM | > 10000.0 nM | | = 530.0 nM|= 443.0 nM|= 440.0 nM|= 220.0 nM|= 199.53 nM|= 600.0 nM|= 630.96 nM|= 260.0 nM|= 481.0 nM|= 251.19 nM|= 250.0 nM|= 230.0 nM|= 290.0 nM|= 288.4 nM | NPASS |
| Neuronal acetylcholine receptor subunit alpha-3/beta-4 | Mus musculus | | | | | = 167.0 nM | NPASS |
| Transient receptor potential cation channel subfamily A member 1 | Homo sapiens | O75762 | 17000 nM|457088190 nM|457000000 nM|= 17000.0 nM|= 457088189.61 nM|= 2000.0 nM | | | | BindingDB, NPASS |
| Striatum | Rattus norvegicus | | = 199.53 nM|= 200.0 nM | | | | NPASS |
| Solute carrier family 22 member 2 | Rattus norvegicus | Q9R0W2 | | | | 50500 nM|= 50500.0 nM | BindingDB, NPASS |
| Solute carrier family 22 member 1 | Rattus norvegicus | Q63089 | | | | 64300 nM|= 64300.0 nM | BindingDB, NPASS |
| Soluble acetylcholine receptor | Aplysia californica | Q8WSF8 | | | | = 2511.89 nM|= 598.0 nM|= 30.0 nM | NPASS |
| Soluble acetylcholine receptor | Aplysia californica | | | | | 280 nM|598 nM|2511.89 nM|30 nM | BindingDB |
| Sigma opioid receptor | Homo sapiens | Q99720 | | > 10000.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily A member 1 | Mus musculus | Q8BLA8 | 10000 nM|= 10000.0 nM | | | | BindingDB, NPASS |
| Sigma non-opioid intracellular receptor 1 | Homo sapiens | Q99720 | | >10000 nM | | | BindingDB |
| Serotonin 3 (5-HT3) receptor | Homo sapiens | Q8WXA8 | | | | = 71000.0 nM | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM | | | NPASS |
| Neuronal acetylcholine receptor; alpha3/beta4 | Homo sapiens | P32297 | = 21000.0 nM|= 4300.0 nM|= 51000.0 nM|= 19830.0 nM|= 8000.0 nM|= 7943.28 nM|= 9400.0 nM|= 290.0 nM|= 7000.0 nM|> 1000.0 nM | = 430.0 nM|> 1000.0 nM | | = 320.0 nM|= 530.0 nM|= 394.0 nM|= 400.0 nM|= 260.0 nM|= 261.0 nM|= 1744.44 nM | NPASS |
| Resistance to inhibitors of cholinesterase protein 3 | Pig roundworm | F1L1D9 | 6210 nM | | | | BindingDB |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens | Q12809 | | 245471 nM|244300 nM|245470.89 nM | | | BindingDB |
| Nicotinic acetylcholine receptor alpha3/betaX | Homo sapiens | Q05901 | = 21000.0 nM | | | | NPASS |
| Nicotinic acetylcholine receptor alpha2/beta4 | Homo sapiens | P30926 | = 10000.0 nM | | | | NPASS |
| Nicotinic acetylcholine receptor alpha-4/beta-2 | Mus musculus | Q8R493 | | | | = 3.5 nM | NPASS |
| Nicotinic acetylcholine receptor alpha 5 subunit | Musca domestica | A9XFY4 | | = 11900.0 nM | | = 2480.0 nM | NPASS |
| Nicotinic acetylcholine receptor | Rattus leucopus | | | | | 8.9 nM|125 nM|2 nM|4000 nM|>10000 nM|1 nM|55.3 nM|9.4 nM|1633 nM|55.2 nM|2.31 nM|1.5 nM|6000 nM|22 nM|7.22 nM|0.96 nM|10 nM|5.3 nM|154 nM|960 nM|12 nM | BindingDB |
| Neuronal nicotinic acetylcholine receptor | Mus musculus | Q2MKA5 | | = 4.0 nM | | = 1.2 nM | NPASS |
| Neuronal acetylcholine receptors; alpha-3/beta-4, alpha-5, beta-2 | Homo sapiens | P30532 | = 30000.0 nM | | | | NPASS |
| Neuronal acetylcholine receptor; alpha4/beta4 | Rattus norvegicus | P12392 | | | | = 46.0 nM|= 40.0 nM|= 33.0 nM|= 31.62 nM|= 150.0 nM|= 158.49 nM|= 23.0 nM|= 5.5 nM|= 141.25 nM|= 140.0 nM|= 51.0 nM|= 72.0 nM|= 72.44 nM | NPASS |
| Neuronal acetylcholine receptor; alpha4/beta4 | Homo sapiens | P43681 | = 7100.0 nM | | | = 129.0 nM|= 23.0 nM|= 70.0 nM | NPASS |
| Neuronal acetylcholine receptor; alpha4/beta2 | Rattus norvegicus | P12390 | = 4000.0 nM|= 590.0 nM|= 7.3 nM|= 1000.0 nM|= 10000.0 nM|= 67.0 nM|= 67.61 nM|= 220.0 nM|= 210.0 nM|= 14000.0 nM|= 591.0 nM|= 77.0 nM|= 19000.0 nM | = 3.8 nM|= 1.65 nM | | = 1.05 nM|= 0.94 nM|= 12.0 nM|= 1.5 nM|= 1.01 nM|= 1.0 nM|= 1.4 nM|= 10.0 nM|= 8.0 nM|= 1.3 nM|= 2.3 nM|= 0.84 nM|= 2.0 nM|= 0.95 nM|= 35.0 nM|= 1.8 nM|= 4.0 nM|= 0.9333 nM|= 6.2 nM|= 6.31 nM|= 6.8 nM|= 3.0 nM|= 7.0 nM|= 22.0 nM|= 19.95 nM|= 4.9 nM|= 9.8 nM|= 11.1 nM|= 2.83 nM|= 7.586 nM|= 7.6 nM|= 11.0 nM|= 2.1 nM|= 13.0 nM|= 14.13 nM|= 4.1 nM|= 5.6 nM | NPASS |
| Neuronal acetylcholine receptor; alpha4/beta2 | Homo sapiens | P43681 | = 4000.0 nM|= 5000.0 nM|= 2100.0 nM|= 9332.54 nM|= 9400.0 nM|= 6600.0 nM|= 6606.93 nM|= 4700.0 nM|= 300.0 nM|= 290.0 nM|= 1.0 nM|= 3000.0 nM|= 295.12 nM|= 295.0 nM|= 2400.0 nM|= 316.23 nM|= 800.0 nM | = 430.0 nM|= 426.58 nM|= 427.0 nM|= 370.0 nM|= 1.2 nM|= 398.11 nM|= 4.9 nM | | = 9.1 nM|= 2.3 nM|= 1.2 nM|= 2.0 nM|= 2.1 nM|= 4.0 nM|= 1.6 nM|> 10000.0 nM|= 1.5 nM|= 9.46 nM|= 12.59 nM|= 4.9 nM|= 5.5 nM|= 1.05 nM|= 0.6 nM|= 10.0 nM|= 0.045 nM|= 2.2 nM|< 1.0 nM | NPASS |
| Rattus norvegicus | Rattus norvegicus | | = 40.0 nM|= 40000.0 nM | | | | NPASS |
| Neuronal acetylcholine receptor subunit alpha-3/beta-4 | Homo sapiens | P30926|P32297 | 51000 nM|21000 nM|4300 nM|19830 nM | | | 172 nM|320 nM|260 nM|261 nM|1744 nM|5.0 nM|530 nM | BindingDB |
| Acetylcholine receptor subunit alpha | Homo sapiens | P02708 | 180000 nM | 21000 nM | | | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-3/beta-2 | Rat | P04757|P12390 | | | | 47 nM | BindingDB |
| Cytochrome P450 2A6 | Homo sapiens | P11509 | | 2.63e+4 nM|579429 nM|> 400000 nM|= 579428.7 nM | 470000 nM|= 470000.0 nM | 4400 nM|130000 nM|= 4400.0 nM|= 130000.0 nM | BindingDB, NPASS |
| Cytochrome P450 2A5 | Mus musculus | P20852 | | 159956 nM|= 159955.8 nM | | | BindingDB, NPASS |
| Cytochrome P450 1A2 | Homo sapiens | P05177 | | 4100000 nM|= 4100000.0 nM | | | BindingDB, NPASS |
| Cholinergic receptor nicotinic alpha 6 subunit | Gallus gallus | | | | | 131 nM | BindingDB |
| Canalicular multispecific organic anion transporter 2 | Homo sapiens | O15438 | | > 133000.0 nM | | | NPASS |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens | Q92887 | | > 133000.0 nM | | | NPASS |
| Bile salt export pump | Homo sapiens | O95342 | | >135000 nM|>1000000 nM|>133000 nM|> 135000.0 nM|> 1000000.0 nM|> 133000.0 nM | | | BindingDB, NPASS |
| Alpha-bungarotoxin | Buus multicinctus | P60615 | | | | 1700 nM|900 nM | BindingDB |
| Acetylcholinesterase | Musca domestica | Q7YWJ9 | | = 2600000.0 nM | | | NPASS |
| Acetylcholine-binding protein | Lymnaea stagnalis | P58154 | | | 40.7 nM|310 nM|320 nM|316 nM|479 nM|= 478.63 nM|= 320.0 nM|= 316.23 nM | 83 nM|496 nM|63.1 nM|331.13 nM|316.23 nM|100 nM|= 63.1 nM|= 331.13 nM|= 316.23 nM|= 496.0 nM|= 100.0 nM|= 83.18 nM|= 83.0 nM | BindingDB, NPASS |
| Acetylcholine receptor; alpha1/beta1/delta/gamma | Homo sapiens | Q07001 | > 1000.0 nM | > 1000.0 nM | | = 5500.0 nM|= 6270.0 nM|= 1480.0 nM | NPASS |
| Acetylcholine receptor subunit delta | Tetronarce californica | P02718 | 20000 nM | | | | BindingDB |
| Acetylcholine receptor subunit beta-like 2 | Drosophila melanogaster | P25162 | | 4000 nM|= 4000.0 nM | | 2700 nM|= 2700.0 nM | BindingDB, NPASS |
| Acetylcholine receptor subunit alpha/beta/delta/gamma | Tetronarce californica | P02710|P02712|P02714|P02718 | 60000 nM | 4 nM|1 nM | | >10000 nM|6270 nM | BindingDB |
| Acetylcholine receptor subunit alpha/beta/delta/gamma | Homo sapiens | P02708|P07510|P11230|Q07001 | | | | 5500 nM | BindingDB |
| Acetylcholine receptor subunit alpha/Neuronal acetylcholine receptor subunit beta-4 | Homo sapiens | P02708|P30926 | 10000 nM | | | | BindingDB |
| Acetylcholine receptor subunit alpha | Rattus norvegicus | P25108 | | | | >10000 nM | BindingDB |
| Acetylcholine receptor protein delta chain | Torpedo californica | P02718 | = 160000.0 nM | | | | NPASS |
| Acetylcholine receptor protein alpha chain | Torpedo californica | P02710 | | = 23100.0 nM | | | NPASS |
| Acetylcholine receptor protein alpha chain | Homo sapiens | P02708 | = 180000.0 nM | = 21000.0 nM | | | NPASS |
| Acetylcholine receptor | Torpedo californica | P02714 | = 60000.0 nM | = 4.0 nM|= 1.0 nM | | > 10000.0 nM|= 6270.0 nM | NPASS |
| ATP-binding cassette sub-family C member 4 | Homo sapiens | O15439 | | >133000 nM | | | BindingDB |
| ATP-binding cassette sub-family C member 3 | Homo sapiens | O15438 | | >133000 nM | | | BindingDB |
| ATP-binding cassette sub-family C member 2 | Homo sapiens | Q92887 | | >133000 nM | | | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-3/beta-2 | Rattus norvegicus | P04757|P12390 | | | | 1 nM|43 nM|47 nM | BindingDB |
| Cytochrome P450 3A4 | Homo sapiens | P08684 | | 1.424e+5 nM | | | BindingDB |
| HERG | Homo sapiens | Q12809 | | = 245470.89 nM|= 244300.0 nM|= 244299.74 nM | | | NPASS |
| Cytochrome P450 2A13 | Homo sapiens | Q16696 | | | 54000 nM|= 54000.0 nM | 72000 nM|= 72000.0 nM | BindingDB, NPASS |
| IMR-32 | Homo sapiens | | = 21000.0 nM | | | | NPASS |
| Neuronal acetylcholine receptor subunit alpha-3/beta-2 | Homo sapiens | P17787|P32297 | 132000 nM | 3.8 nM | | 47 nM|29 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-3 | Rattus norvegicus | P04757 | | | | 475 nM|100 nM|290 nM|47 nM|440 nM|600 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-3 | Homo sapiens | P32297 | 9400 nM | 45 nM|= 45.0 nM | | >10000 nM|14 nM|187 nM|220 nM|= 220.0 nM | BindingDB, NPASS |
| Neuronal acetylcholine receptor subunit alpha-2/beta-4 | Rattus norvegicus | P12389|P12392 | | | | 112 nM|110 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-2/beta-4 | Rat | P12389|P12392 | | | | 110 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-2/beta-4 | Homo sapiens | P30926|Q15822 | | | | 103 nM|70 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-2/beta-2 | Rattus norvegicus | P12389|P12390 | | | | 15 nM|12 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-2/beta-2 | Rat | P12389|P12390 | | | | 12 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-2/beta-2 | Homo sapiens | P17787|Q15822 | | | | 5.5 nM | BindingDB |
| High affinity choline transporter 1 | Mus musculus | Q8BGY9 | | | | 520115.74 nM | BindingDB |
| Neuronal acetylcholine receptor subunit alpha-2 | Homo sapiens | Q15822 | | | | 9900 nM | BindingDB |
| Neuronal acetylcholine receptor protein alpha-9 subunit | Rattus norvegicus | P43144 | | = 2.4 nM | = 5.0 nM | | NPASS |
| Neuronal acetylcholine receptor protein alpha-7 subunit | Rattus norvegicus | Q05941 | = 54000.0 nM|= 43000000.0 nM|= 13000.0 nM|= 1500.0 nM|= 1071.52 nM|= 23000.0 nM|= 109647.82 nM|= 108700.0 nM|= 47000.0 nM | = 16.0 nM | | = 4000.0 nM|= 770.0 nM|= 450.0 nM|= 340.0 nM|= 480.0 nM|= 130.0 nM|= 460.0 nM|= 6290.0 nM|= 1748.0 nM|= 750.0 nM|= 234.0 nM|= 1500.0 nM|= 670.0 nM|= 176.0 nM|= 16000.0 nM|= 15848.93 nM|= 469.0 nM|= 1400.0 nM|= 517.0 nM|= 230.0 nM|= 520.0 nM|= 610.0 nM|= 15000.0 nM|= 250.0 nM|= 400.0 nM | NPASS |
| Neuronal acetylcholine receptor subunit alpha-2 | Rattus norvegicus | P12389 | | | | 3.6 nM|83 nM|12 nM|110 nM | BindingDB |
| Neuronal acetylcholine receptor protein alpha-7 subunit | Homo sapiens | P36544 | = 83000.0 nM|= 38000.0 nM|= 113000.0 nM|= 1584.89 nM|= 91000.0 nM|= 4710.0 nM | = 21000.0 nM|= 7600.0 nM | = 1.06 nM | = 1610.0 nM|= 620.0 nM|= 7200.0 nM|= 6300.0 nM|= 630.0 nM|= 24000.0 nM|= 25118.86 nM|= 12000.0 nM|= 10000.0 nM|= 1000.0 nM|= 2110.0 nM|= 1023.29 nM|= 3000.0 nM|= 3800.0 nM|= 6290.0 nM | NPASS |
| K177cell line | | | = 5000.0 nM | | | | NPASS |
| Neuronal acetylcholine receptor protein alpha-7 subunit | Mus musculus | P49582 | | | | = 480.0 nM|= 244.0 nM | NPASS |
| Multidrug resistance-associated protein 4 | Homo sapiens | O15439 | | > 133000.0 nM | | | NPASS |
| Mus musculus | Mus musculus | | | | = 1.41 nM | | NPASS |
| Muscarinic acetylcholine receptor | Rattus norvegicus | P10980 | | = 32000.0 nM|= 360000.0 nM|= 28000.0 nM | | > 5000.0 nM|> 10000.0 nM | NPASS |
| Lycopene cyclase | Pantoea ananas | P21687 | | = 4800.0 nM | | | NPASS |
| Muscle-type nicotinic acetylcholine receptor | Homo sapiens | Q04844 | = 65000.0 nM | | | | NPASS |
| NON-PROTEIN TARGET | | | = 941600.0 nM|= 1963000.0 nM | = 5800.0 nM|= 6200.0 nM|= 3700.0 nM|= 3600.0 nM | | | NPASS |
| Neuronal acetylcholine receptor | Rattus norvegicus | Q05941 | = 20000.0 nM | = 6.6 nM|= 7.0 nM|= 3.0 nM|= 4.0 nM | = 4.9e-06 nM|= 0.01 nM|= 430.0 nM|= 11000.0 nM|= 43000000.0 nM|= 0.022 nM|= 10.0 nM|= 5.2 nM|= 45000.0 nM | = 8.4 nM|= 2.4 nM|= 1.15 nM|= 1.1 nM|= 13.0 nM|= 27.0 nM|= 1.3 nM|= 1.0 nM | NPASS |
| Neuronal acetylcholine receptor protein alpha-2 subunit | Rattus norvegicus | P12389 | | | | = 12.0 nM | NPASS |
| Neuronal acetylcholine receptor protein alpha-4 subunit | Mus musculus | O70174 | | = 7.0 nM | | | NPASS |
| Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 | Rattus norvegicus | P08482|P08483|P08485|P08911|P10980 | | 360000 nM|28000 nM|32000 nM | | >5000 nM | BindingDB |