IMPPAT Phytochemical information: 
Serotonin

Serotonin
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Serotonin 2 (5-HT2) receptorRattus norvegicusP08909|P14842|P3099420 nM|4600 nM|3600 nM930 nM|7.8 nM|6 nM|560 nM|2950 nM|977 nM|950 nMBindingDB
Serotonin 2 (5-HT2) receptorMus musculusP35363= 680.0 nM= 500.0 nMNPASS
Serotonin 2 (5-HT2) receptorHomo sapiensP28223|P28335|P415953162 nMBindingDB
Serotonin 1f (5-HT1f) receptorHomo sapiensP30939= 7.9 nMNPASS
Serotonin 1e (5-HT1e) receptorHomo sapiensP28566= 4.0 nM|= 10.72 nM|= 11.0 nMNPASS
Serotonin 1d (5-HT1d) receptorSus scrofaP79400= 10.0 nMNPASS
MAP/microtubule affinity-regulating kinase 4Homo sapiensQ96L342990 nM|= 2990.0 nMBindingDB, NPASS
Serotonin 1d (5-HT1d) receptorHomo sapiensP28221= 3.0 nM= 5.5 nM|= 4.8 nM|= 5.06 nM|= 1.7 nM|= 2.0 nM|= 3.0 nM|= 0.5 nMNPASS
Serotonin 1d (5-HT1d) receptorCavia porcellusQ60484= 16.0 nM|= 8.5 nM|= 5.2 nM= 3.0 nMNPASS
Serotonin 1b (5-HT1b) receptorRattus norvegicusP28564= 26.0 nM= 5.0 nM|= 4.6 nM|= 4.9 nM= 2.512 nM|= 5.4 nM|= 25.0 nM|= 2.5 nM|= 1.1 nM|= 3.467 nM|= 5.0 nMNPASS
Serotonin 1b (5-HT1b) receptorHomo sapiensP28222= 30.0 nM|= 4.82 nM|= 4.67 nM= 5.0 nM|= 29.0 nM|= 16.0 nM|= 12.0 nM|= 6.5 nM= 4.0 nM|= 7.1 nM|= 6.76 nM|= 5.012 nM|= 4.8 nM|= 1.1 nM|= 18.0 nM|= 14.0 nMNPASS
Serotonin 1a (5-HT1a) receptorRattus norvegicusP19327= 10.0 nM|= 323.0 nM= 5.2 nM|= 3.0 nM|= 2.6 nM= 1.585 nM|= 1.7 nM|= 4.31 nM|= 3.0 nM|= 2.1 nM|= 7.3 nM|= 4.786 nM|= 2.0 nM|= 1.862 nM|= 1.6 nM|= 2.6 nM|= 9.0 nM|= 2.3 nMNPASS
Serotonin 1a (5-HT1a) receptorMus musculusQ64264= 5.0 nMNPASS
Serotonin 1a (5-HT1a) receptorHomo sapiensP08908= 8.71 nM|= 3.7 nM|= 43.0 nM|= 10.0 nM|= 0.5 nM|= 1.0 nM|= 0.7 nM|= 229.09 nM|= 150.0 nM|= 147.0 nM|= 3.75 nM|= 39.0 nM|= 3.0 nM|= 27.54 nM|= 169.82 nM|= 15.33 nM|= 69.18 nM|= 97.7 nM|= 5.7 nM|= 19.0 nM|= 5.61 nM|= 56.23 nM|= 18.0 nM|= 1800.0 nM|= 45.3 nM|= 33.11 nM|= 30.9 nM|= 128.82 nM|= 58.88 nM|= 50.12 nM|= 5.8 nM|= 398.11 nM|= 2.03 nM|= 3.4 nM|= 10.96 nM= 5.6 nM|= 6.0 nM|= 2.0 nM|= 1.2 nM|= 5.2 nM= 1.7 nM|= 2.5 nM|= 2.48 nM|= 2.8 nM|= 3.0 nM|= 3.981 nM|= 1.259 nM|= 10000.0 nM|< 50.0 nM|= 0.62 nM|= 0.9 nM|= 9.5 nM|= 2.08 nM|= 1.3 nM|= 1.4 nM|= 1.1 nM|= 5.5 nM|= 1.2 nM|= 3.6 nM|= 0.91 nM|= 4.5 nMNPASS
Serotonin 2 (5-HT2) receptorRattus norvegicusP14842= 4600.0 nM|= 3600.0 nM|= 20.0 nM= 930.0 nM|= 7.8 nM|= 2950.0 nM|= 560.0 nM|= 6.0 nM|= 977.24 nM|= 950.0 nMNPASS
Serotonin 1d (5-HT1d) receptorRattus norvegicusP28565= 5.2 nM= 3.0 nMNPASS
Serotonin 1 (5-HT1) receptorRattus norvegicusP28565= 5.9 nM|= 20.0 nM= 2.0 nMNPASS
Ribosyldihydronicotinamide dehydrogenase [quinone]Homo sapiensP1608353900 nMBindingDB
Serotonin 2a (5-HT2a) receptorHomo sapiensP28223= 11.0 nM|= 125.89 nM|= 70.0 nM|= 5.8 nM|= 7.6 nM|= 147.91 nM|= 2.57 nM|= 150.0 nM|= 2.6 nM|= 16.0 nM|= 1.5 nM|= 1.549 nM|= 1.88 nM|= 302.0 nM|= 47.0 nM|= 2.344 nM|= 2.35 nM|= 1.6 nM|= 0.2754 nM|= 0.27 nM|= 0.51 nM|= 0.5129 nM|= 1.1 nM|= 12.1 nM|= 130.0 nM|= 3.0 nM|= 1.32 nM|= 0.23 nM|= 661.0 nM|= 2.951 nM|= 0.631 nM|= 28.0 nM|= 25.12 nM|= 1672.0 nM= 27.9 nM= 14.0 nM|= 510.0 nM|= 398.11 nM|= 8.2 nM|= 120.0 nM|= 160.0 nM|= 130.0 nM|= 150.0 nM|= 320.0 nM|= 690.0 nM|= 323.59 nM|= 11.5 nM|= 17.2 nMNPASS
Macrophage migration inhibitory factorHomo sapiensP14174> 400000.0 nMNPASS
Melatonin receptor 1AHomo sapiensP48039> 100000.0 nMNPASS
Melatonin receptor 1BHomo sapiensP49286> 100000.0 nMNPASS
Melatonin receptor type 1AHomo sapiensP48039>100000 nMBindingDB
Melatonin receptor type 1AOvis ariesP48040>10000 nMBindingDB
Melatonin receptor type 1BHomo sapiensP49286>10000 nM|>100000 nMBindingDB
NG108-15Murinae= 298.0 nM|= 293.0 nMNPASS
Norepinephrine transporterRattus norvegicus1000 nM|3013 nM|>10000 nMBindingDB
Oryctolagus cuniculusOryctolagus cuniculus= 158.49 nM|= 300.0 nMNPASS
Polyphenol oxidase 2Agaricus bisporusO42713>350000 nMBindingDB
Prostaglandin G/H synthase 1Homo sapiensP23219>400000 nMBindingDB
Prostaglandin G/H synthase 2Homo sapiensP35354>400000 nMBindingDB
Radical scavenging activity> 250000.0 nMNPASS
Rattus norvegicusRattus norvegicus= 977.24 nM= 3548.13 nM|= 28183.83 nM|= 369.0 nM> 5000.0 nM|= 919.0 nM|= 14092.0 nM|> 3000.0 nMNPASS
SARS-CoV-2Severe acute respiratory syndrome coronavirus 2> 20000.0 nM|> 19952.62 nMNPASS
Serotonin 2a (5-HT2a) receptorMus musculusP35363= 0.5248 nM|= 0.53 nMNPASS
Serotonin 7 (5-HT7) receptorHomo sapiensP34969= 15.0 nM|= 17.0 nM|= 5.754 nM|= 5.8 nM|= 7.0 nM|= 47.86 nM|= 48.0 nM|= 5.7 nM|= 5.37 nM|= 70.0 nM|= 3.66 nM|= 110.0 nM|= 9.333 nM|= 112.2 nM|= 4.5 nM= 0.61 nM|= 2.55 nM|= 1.5 nM|= 0.49 nM|= 0.29 nM|= 0.25 nM|= 0.47 nM= 3.98 nM= 4.0 nM|= 8.1 nM|= 3.162 nM|= 0.22 nM|= 0.13 nM|= 0.11 nM|= 1.4 nM|= 0.8 nM|= 6.0 nM|= 0.17 nM|= 7.943 nM|= 2.12 nM|= 2.1 nMNPASS
Serotonin 2b (5-HT2b) receptorHomo sapiensP41595= 1.5 nM|= 25.12 nM|= 5.8 nM|= 0.5 nM|= 11.0 nM|= 0.86 nM|= 1.1 nM|= 1.072 nM|= 0.92 nM|= 1.445 nM|= 1.46 nM|= 4.5 nM|= 0.8511 nM|= 0.07079 nM|= 2.4 nM|= 1.19 nM|= 1.259 nM= 12.0 nM|= 13.0 nM|= 13.49 nM|= 10.8 nMNPASS
Sodium-dependent dopamine transporterRattus norvegicusP23977>10000 nM|2703 nMBindingDB
Sodium-dependent serotonin transporterRattus norvegicusP31652740 nMBindingDB
Solute carrier family 22 member 1Rattus norvegicusQ63089390000 nM|= 390000.0 nMBindingDB, NPASS
Solute carrier family 22 member 2Rattus norvegicusQ9R0W2242000 nM|= 242000.0 nMBindingDB, NPASS
Solute carrier family 22 member 3Rattus norvegicusO8844697000 nM|= 97000.0 nMBindingDB, NPASS
SortaseStaphylococcus aureusQ9S446> 100.0 ug.mL-1NPASS
Sodium-dependent dopamine transporterHomo sapiensQ01959>10000 nMBindingDB
Synaptic vesicular amine transporterHomo sapiensQ059401430 nM|= 1430.0 nM7690 nM|640000 nM|2290 nM|= 7690.0 nM|= 640000.0 nM|= 2290.0 nMBindingDB, NPASS
Trace amine-associated receptor 1Homo sapiensQ96RJ035100 nM|= 35100.0 nMBindingDB, NPASS
TyrosinaseAgaricus bisporusO42713> 350000.0 nMNPASS
TyrosinaseMus musculusP11344550000 nM|= 550000.0 nMBindingDB, NPASS
Vascular endothelial growth factor receptor 2Homo sapiensP35968>50000 nMBindingDB
Vascular endothelial growth factor receptor 3Homo sapiensP35916>50000 nMBindingDB
Isocitrate lyaseCandida albicansQ9P8Q7301000 nM|301300 nM|= 301300.0 nM|= 301000.0 nM|= 53.0 ug.mL-1BindingDB, NPASS
Synaptic vesicular amine transporterMus musculusQ8BRU698 nM|= 98.0 nMBindingDB, NPASS
Serotonin transporterRattus norvegicusP31652= 740.0 nMNPASS
Serotonin receptor 2a and 2c (5HT2A and 5HT2C)Rattus norvegicusP14842= 10.6 nM|= 6.1 nM|= 600.0 nMNPASS
Serotonin 7 (5-HT7) receptorRattus norvegicusP32305= 10.0 nM|= 0.6026 nM|= 7.33 nMNPASS
Serotonin 2b (5-HT2b) receptorRattus norvegicusP30994= 3.5 nM|= 4.19 nMNPASS
Serotonin 2c (5-HT2c) receptorHomo sapiensP28335= 1.7 nM|= 25.12 nM|= 24.0 nM|= 0.09 nM|= 25.0 nM|= 1.63 nM|= 43.65 nM|= 0.871 nM|= 44.0 nM|= 0.87 nM|= 0.4 nM|= 0.3467 nM|= 0.21 nM|= 190.55 nM|= 0.182 nM|= 0.17 nM|= 15.14 nM|= 15.0 nM|= 0.1905 nM|= 0.19 nM|= 0.41 nM|= 0.166 nM|= 0.1349 nM|= 0.14 nM|= 21.88 nM|= 21.0 nM|= 0.12 nM|= 1.202 nM|= 0.1259 nM|= 1.2 nM= 81.0 nM|= 1.25 nM= 35.0 nM|= 6.9 nM|= 50.12 nM|= 8.3 nM|= 130.0 nM|= 20.0 nM|= 445.0 nM|= 214.0 nM|= 79.43 nM|= 79.0 nMNPASS
Serotonin 2c (5-HT2c) receptorRattus norvegicusP08909= 2.8 nM= 81.0 nM|= 42.0 nM= 31.62 nM|= 23.0 nM|= 10.0 nMNPASS
Serotonin 3 (5-HT3) receptorHomo sapiensQ8WXA8= 144.54 nM|= 120.0 nMNPASS
Serotonin 3 (5-HT3) receptorRattus norvegicusQ9JJ16= 727.0 nM= 398.11 nM|= 320.0 nM|= 66.0 nM|= 120.0 nM|= 87.0 nM|= 390.0 nMNPASS
Serotonin 3 receptor (5HT3)Mus musculusP23979= 361.0 nMNPASS
Serotonin 3a (5-HT3a) receptorHomo sapiensP46098= 500.0 nM|= 457.09 nM|= 178.0 nM|= 141.0 nMNPASS
Serotonin 3a (5-HT3a) receptorMus musculusP23979= 3400.0 nM|= 24000.0 nM|= 3300.0 nM|= 170000.0 nM|= 37000.0 nM|= 20900.0 nM|= 17200.0 nM|= 9600.0 nM|= 90000.0 nM|= 4400.0 nM|= 210000.0 nM|= 140000.0 nM|= 49000.0 nM|= 7100.0 nM|= 980.0 nM|= 51000.0 nM|= 11000.0 nM|= 6200.0 nM|= 5100.0 nM|= 2900.0 nM|= 27000.0 nM|= 1300.0 nM|= 1320.0 nM|= 63000.0 nM|= 42000.0 nM|= 15000.0 nMNPASS
Serotonin 3a (5-HT3a) receptorRattus norvegicusP35563= 12000.0 nMNPASS
Serotonin 4 (5-HT4) receptorCavia porcellusO70528= 5.0 nM|= 10.0 nM= 100.0 nM|= 230.0 nMNPASS
Serotonin 4 (5-HT4) receptorHomo sapiensQ13639= 100.0 nM|= 12.0 nM= 323.0 nM= 1049.0 nM|= 500.0 nM|= 29.51 nM|= 109.65 nM|= 246.0 nMNPASS
Serotonin 4 (5-HT4) receptorRattus norvegicusQ62758= 6.31 nM|= 17.1 nM= 3.7 nM|= 147.0 nM= 187.0 nM|= 37.4 nMNPASS
Serotonin 5a (5-HT5a) receptorHomo sapiensP47898= 79.0 nM|= 180.0 nM|= 184.0 nM|= 280.0 nM|= 160.0 nM|= 260.0 nM= 250.0 nM|= 126.0 nM|= 110.0 nM|= 170.0 nM|= 82.0 nM|= 130.0 nMNPASS
Serotonin 5a (5-HT5a) receptorMus musculusP30966= 150.0 nMNPASS
Serotonin 6 (5-HT6) receptorHomo sapiensP50406= 43.6 nM|= 42.1 nM= 200.0 nM|= 262.0 nM|= 27.5 nM|= 180.0 nM|= 100.0 nM|= 120.0 nM|= 130.0 nM= 65.0 nM|= 78.0 nM|= 75.0 nM|= 125.89 nM|= 100.0 nM|= 93.0 nM|= 84.0 nM|= 70.0 nM|= 50.0 nM|= 33.0 nM|= 61.0 nMNPASS
Serotonin 2a (5-HT2a) receptorRattus norvegicusP14842= 351.0 nM|= 55.8 nM|= 57.9 nM= 0.9 nM|= 2350.0 nM|= 0.94 nM|= 13000.0 nM|= 30600.0 nM|= 600.0 nM= 1258.93 nM|= 0.3 nM|= 1258.0 nM|= 10.6 nM|= 600.0 nMNPASS
Insulin-like growth factor 1 receptorHomo sapiensP08069>50000 nMBindingDB
D(1A) dopamine receptorRattus norvegicusP189015000 nMBindingDB
Dopamine receptor D4Canis lupus familiaris4180 nMBindingDB
5-hydroxytryptamine receptor 1FMus musculusQ02284125.89 nMBindingDB
5-hydroxytryptamine receptor 1FRattus norvegicusP3094067.6 nMBindingDB
5-hydroxytryptamine receptor 2AHomo sapiensP2822311 nM|1.9 nM|302 nM|5.8 nM|47 nM|2.3 nM|2.4 nM|70 nM|7.6 nM|2.6 nM|150 nM|1.6 nM|126 nM|0.275423 nM|0.270000 nM|0.510000 nM|0.512861 nM|1.1 nM|12 nM|130 nM|661 nM|1672 nM28 nM63.09 nM|12.02 nM|602.55 nM|7.77 nM|218.77 nM|30.90 nM|341 nM|21 nM|16.22 nM|20.0 nM|510 nM|320 nM|160 nM|150 nM|120 nM|14 nM|8.2 nM|690 nM|8.20 nM|130 nM|12 nM|398 nM|17 nMBindingDB
5-hydroxytryptamine receptor 2AMus musculusP353630.524807 nM|0.530000 nMBindingDB
5-hydroxytryptamine receptor 2A/2B/2CMus musculusP34968|P35363|Q02152680 nM500 nMBindingDB
5-hydroxytryptamine receptor 2BBos taurus750 nMBindingDB
5-hydroxytryptamine receptor 1FHomo sapiensP309397.9 nM10 nM|>10000 nMBindingDB
5-hydroxytryptamine receptor 2BHomo sapiensP415951.5 nM|0.920000 nM|0.5 nM|11 nM|1.4 nM|5.8 nM|0.86 nM|4.5 nM|25 nM|0.860000 nM|0.851138 nM|0.070795 nM0.79 nM|9.8 nM|9.46 nM|1.17 nM|2.09 nM|4 nM|1 nM|19 nM|13.49 nM|12 nM|13 nM|11 nMBindingDB
5-hydroxytryptamine receptor 2BRattus norvegicusP309943.5 nM|4.2 nM10 nM|28.18 nM|10.23 nM|10.2 nM|11.3 nMBindingDB
5-hydroxytryptamine receptor 2CHomo sapiensP283351.7 nM|0.210000 nM|191 nM|0.09 nM|25 nM|15 nM|0.170000 nM|0.181970 nM|24 nM|1.63 nM|0.870000 nM|44 nM|0.190546 nM|0.190000 nM|0.410000 nM|0.165959 nM|0.134896 nM|0.140000 nM|22 nM|21 nM278 nM|81 nM|1.3 nM656 nM|15.5 nM|56.23 nM|5.75 nM|2.9 nM|18.20 nM|2.4 nM|130 nM|6.9 nM|8.3 nM|20 nM|35 nM|8.30 nM|214 nM|445 nM|79 nM|50 nMBindingDB
5-hydroxytryptamine receptor 2CRattus norvegicusP089092.8 nM81 nM|42 nM32 nM0.7 nM|22.9 nM|87.09 nM|44 nM|11 nM|159 nM|12.2 nM|10 nM|23 nMBindingDB
5-hydroxytryptamine receptor 3ACavia porcellusO70212>10000 nM|495 nMBindingDB
5-hydroxytryptamine receptor 3AHomo sapiensP46098141 nM|178 nM|457 nMBindingDB
5-hydroxytryptamine receptor 3AMus musculusP239793400 nM269.15 nM|292 nM|361 nMBindingDB
5-hydroxytryptamine receptor 2BMus musculusQ021521258.92 nMBindingDB
5-hydroxytryptamine receptor 1ERattus norvegicus7 nMBindingDB
5-hydroxytryptamine receptor 1EHomo sapiensP2856611 nM|3.5 nM|10.96 nM|7.24 nM|6.16 nM|2.3 nM|4 nMBindingDB
5-hydroxytryptamine receptor 1DSus scrofaP7940010 nM|10.0 nMBindingDB
Epidermal growth factor receptorHomo sapiensP00533>50000 nMBindingDB
5-hydroxytryptamine 1D receptorBos taurus4 nM|1.9 nMBindingDB
5-hydroxytryptamine receptor 1AHomo sapiensP0890810 nM|1 nM|3.0 nM|1.000 nM|0.700000 nM|28 nM|170 nM|43 nM|15 nM|3.7 nM|150 nM|69 nM|147 nM|3.8 nM|98 nM|5.7 nM|19 nM|8.7 nM|229 nM|5.6 nM|5.61 nM|18 nM|1800 nM|45 nM|33 nM|31 nM|129 nM|59 nM|50 nM|5.8 nM|2.0 nM5.2 nM|6 nM|2 nM|5.6 nM|1.2 nM3.2 nM0.26 nM|1.25 nM|12.58 nM|0.79 nM|3.98 nM|102.32 nM|102.3 nM|1.3 nM|3 nM|2.8 nM|1.7 nM|2.48 nM|2.5 nM|2.1 nM|0.62 nM|10 nM|10000 nM|0.900000 nM|1.4 nM|4.0 nM|5.5 nM|1.2 nM|3.6 nM|3.0 nM|0.910000 nM|4.5 nMBindingDB
5-hydroxytryptamine receptor 1AHumanP089081.2 nM|10.0 nMBindingDB
5-hydroxytryptamine receptor 1AMus musculusQ642645 nMBindingDB
5-hydroxytryptamine receptor 1ARattus norvegicusP1932710 nM|323 nM5.2 nM|3 nM|2.6 nM46.77 nM|134 nM|4.2 nM|0.12 nM|90 nM|2 nM|1.7 nM|3 nM|1.6 nM|4.3 nM|2.1 nM|7.3 nM|2.6 nM|4.8 nM|1.9 nM|2.3 nMBindingDB
5-hydroxytryptamine receptor 1A/1B/1D/1FRattus norvegicusP19327|P28564|P28565|P3094020 nM2 nMBindingDB
5-hydroxytryptamine receptor 1BCavia porcellusO088922.51 nMBindingDB
5-hydroxytryptamine receptor 1BHomo sapiensP2822230 nM|4.82 nM|4.7 nM5 nM0.59 nM|3.9 nM|4.26 nM|1.09 nM|3.98 nM|0.57 nM|15.84 nM|7.94 nM|38 nM|9 nM|4.07 nM|6.8 nM|4 nM|1.1 nM|7.1 nM|4.8 nM|14 nM|5.0 nMBindingDB
5-hydroxytryptamine receptor 1BMus musculusP2833439.81 nMBindingDB
5-hydroxytryptamine receptor 1BRattus norvegicusP2856426 nM5 nM|4.9 nM|4.6 nM14 nM|15.84 nM|5.24 nM|3.01 nM|0.57 nM|3 nM|2.6 nM|5 nM|5.4 nM|3.5 nM|25 nM|2.5 nM|1.1 nMBindingDB
5-hydroxytryptamine receptor 1DCanis lupus familiarisP116145.01 nM|15.84 nMBindingDB
5-hydroxytryptamine receptor 1DCavia porcellusQ604848.5 nM|16 nM|5.2 nM3 nMBindingDB
5-hydroxytryptamine receptor 1DHomo sapiensP282213 nM13 nM4.3 nM|8.9 nM|2.1 nM|8.91 nM|2.08 nM|3.89 nM|3.98 nM|3.4 nM|3.38 nM|3 nM|5.5 nM|1.7 nM|5.06 nM|5.1 nM|2 nM|0.500000 nM|4.8 nMBindingDB
5-hydroxytryptamine receptor 1DRattus norvegicusP285655.2 nM3 nM2.51 nM|18 nMBindingDB
5-hydroxytryptamine receptor 3ARattus norvegicusP3556312000 nMBindingDB
5-hydroxytryptamine receptor 3A/3BRattus norvegicusP35563|Q9JJ16727 nM87 nM|320 nM|390 nM|66 nM|120 nMBindingDB
5-hydroxytryptamine receptor 2ARattus norvegicusP1484258 nM|55.8 nM|351 nM0.940000 nM|2350 nM|0.9 nM|13000 nM|30600 nM|600 nM3 nM|270 nM|83 nM|125.89 nM|5.75 nM|1.99 nM|478.63 nM|707.94 nM|251.18 nM|2955 nM|120.22 nM|96 nM|1258 nM|11 nM|600 nM|0.3 nMBindingDB
5-hydroxytryptamine receptor 4Homo sapiensQ1363912 nM|100 nM323 nM1049 nM|316.22 nM|56.23 nM|1151 nM|481.9 nM|330 nM|251.18 nM|158.5 nM|100 nM|500 nM|29.51 nM|109.65 nM|246 nMBindingDB
Canis familiarisCanis lupus familiaris= 210.0 nMNPASS
Cyclooxygenase-1Homo sapiensP23219> 400000.0 nMNPASS
Cyclooxygenase-2Homo sapiensP35354> 400000.0 nMNPASS
D(1A) dopamine receptorHomo sapiensP217289690 nM>10000 nMBindingDB
D(1B) dopamine receptorHomo sapiensP219183000 nMBindingDB
D(2) dopamine receptorCanis lupus familiarisQ9GJU1>10000 nMBindingDB
B16Mus musculus> 30000.0 nMNPASS
D(2) dopamine receptorHomo sapiensP144160.000 nM>10000 nMBindingDB
5-hydroxytryptamine receptor 4Cavia porcellusO705285 nM|10 nM79.43 nM|50.11 nM|39.81 nM|230 nM|100 nMBindingDB
D(3) dopamine receptorRattus norvegicusP190202338 nMBindingDB
Dopamine D1 receptorHomo sapiensP21728= 9690.0 nMNPASS
Dopamine D2 receptorHomo sapiensP14416= 0.0003 nMNPASS
Dopamine D3 receptorHomo sapiensP35462= 523.0 nMNPASS
Dopamine D3 receptorRattus norvegicusP19020= 2338.0 nMNPASS
D(2) dopamine receptorRattus norvegicusP61169>10000 nM|1655 nM|7950 nMBindingDB
Alpha-glucosidase MAL62Saccharomyces cerevisiaeP07265>300000 nM|> 300000.0 nMBindingDB, NPASS
D(3) dopamine receptorHomo sapiensP35462523 nMBindingDB
Alpha-1A adrenergic receptorRattus norvegicusP4314018000 nM|23000 nMBindingDB
5-hydroxytryptamine receptor 4Mus musculusP9728879.43 nM|56.23 nMBindingDB
Alpha-2C adrenergic receptorRattus norvegicusP22086>10000 nMBindingDB
5-hydroxytryptamine receptor 4Rattus norvegicusQ6275817 nM|6.3 nM3.7 nM|147 nM145 nM|200 nM|6.3 nM|7.94 nM|125.89 nM|199.52 nM|158.48 nM|38.9 nM|37 nM|187 nMBindingDB
5-hydroxytryptamine receptor 5AHomo sapiensP47898180 nM|260 nM|79 nM126 nM|130 nM|250 nM|170 nMBindingDB
5-hydroxytryptamine receptor 5ARattus norvegicusP353641333 nM|239.88 nMBindingDB
5-hydroxytryptamine receptor 5BMus musculusP31387251.18 nMBindingDB
5-hydroxytryptamine receptor 5BRattus norvegicusP35365239 nM|1318.25 nM|7.76 nM|7.8 nMBindingDB
5-hydroxytryptamine receptor 6Homo sapiensP5040644 nM|42 nM120 nM|27.5 nM|130 nM56 nM|65 nM|33 nM|75 nM|78 nM|61 nM|100 nM|84 nM|126 nM|70 nMBindingDB
5-hydroxytryptamine receptor 5AMus musculusP30966251.18 nM|1100 nM|150 nMBindingDB
5-hydroxytryptamine receptor 6Rattus norvegicusP31388151 nM|56 nM|151.35 nM|56.23 nM|12.58 nM|234.42 nM|79.43 nMBindingDB
5-hydroxytryptamine receptor 7Rattus norvegicusP323051.81 nM|4.89 nM|1.51 nM|25.11 nM|0.6 nM|1.83 nM|1.52 nM|5 nM|2.00 nM|0.63 nM|7.94 nM|0.13 nM|7.33 nM|10 nM|0.602560 nMBindingDB
5-hydroxytryptamine receptor 7Cavia porcellusP504071 nM|1.34 nM|0.25 nM|0.10 nMBindingDB
5-hydroxytryptamine receptor 7Homo sapiensP3496917 nM|15 nM|5.8 nM|48 nM|7.0 nM|5.4 nM|5.7 nM|70 nM|3.7 nM|9.3 nM|9.33 nM|112 nM|110 nM0.250 nM|2.55 nM|0.470000 nM4.0 nM8.12 nM|8.1 nM|7.94 nM|0.40 nM|0.38 nM|6.31 nM|1.4 nM|0.800000 nM|4 nM|6.0 nM|0.170000 nM|0.13 nM|3.2 nM|7.9 nM|2.1 nMBindingDB
5-hydroxytryptamine receptor 6Mus musculusQ9R1C839.81 nM|5.01 nM|95.50 nMBindingDB
5-hydroxytryptamine receptor 7Mus musculusP323045.01 nMBindingDB