| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Serotonin 2 (5-HT2) receptor | Rattus norvegicus | P08909|P14842|P30994 | | 20 nM|4600 nM|3600 nM | | 930 nM|7.8 nM|6 nM|560 nM|2950 nM|977 nM|950 nM | BindingDB |
| Serotonin 2 (5-HT2) receptor | Mus musculus | P35363 | | = 680.0 nM | | = 500.0 nM | NPASS |
| Serotonin 2 (5-HT2) receptor | Homo sapiens | P28223|P28335|P41595 | | | 3162 nM | | BindingDB |
| Serotonin 1f (5-HT1f) receptor | Homo sapiens | P30939 | = 7.9 nM | | | | NPASS |
| Serotonin 1e (5-HT1e) receptor | Homo sapiens | P28566 | | | | = 4.0 nM|= 10.72 nM|= 11.0 nM | NPASS |
| Serotonin 1d (5-HT1d) receptor | Sus scrofa | P79400 | | = 10.0 nM | | | NPASS |
| MAP/microtubule affinity-regulating kinase 4 | Homo sapiens | Q96L34 | | 2990 nM|= 2990.0 nM | | | BindingDB, NPASS |
| Serotonin 1d (5-HT1d) receptor | Homo sapiens | P28221 | | = 3.0 nM | | = 5.5 nM|= 4.8 nM|= 5.06 nM|= 1.7 nM|= 2.0 nM|= 3.0 nM|= 0.5 nM | NPASS |
| Serotonin 1d (5-HT1d) receptor | Cavia porcellus | Q60484 | = 16.0 nM|= 8.5 nM|= 5.2 nM | = 3.0 nM | | | NPASS |
| Serotonin 1b (5-HT1b) receptor | Rattus norvegicus | P28564 | = 26.0 nM | = 5.0 nM|= 4.6 nM|= 4.9 nM | | = 2.512 nM|= 5.4 nM|= 25.0 nM|= 2.5 nM|= 1.1 nM|= 3.467 nM|= 5.0 nM | NPASS |
| Serotonin 1b (5-HT1b) receptor | Homo sapiens | P28222 | = 30.0 nM|= 4.82 nM|= 4.67 nM | = 5.0 nM|= 29.0 nM|= 16.0 nM|= 12.0 nM|= 6.5 nM | | = 4.0 nM|= 7.1 nM|= 6.76 nM|= 5.012 nM|= 4.8 nM|= 1.1 nM|= 18.0 nM|= 14.0 nM | NPASS |
| Serotonin 1a (5-HT1a) receptor | Rattus norvegicus | P19327 | = 10.0 nM|= 323.0 nM | = 5.2 nM|= 3.0 nM|= 2.6 nM | | = 1.585 nM|= 1.7 nM|= 4.31 nM|= 3.0 nM|= 2.1 nM|= 7.3 nM|= 4.786 nM|= 2.0 nM|= 1.862 nM|= 1.6 nM|= 2.6 nM|= 9.0 nM|= 2.3 nM | NPASS |
| Serotonin 1a (5-HT1a) receptor | Mus musculus | Q64264 | | = 5.0 nM | | | NPASS |
| Serotonin 1a (5-HT1a) receptor | Homo sapiens | P08908 | = 8.71 nM|= 3.7 nM|= 43.0 nM|= 10.0 nM|= 0.5 nM|= 1.0 nM|= 0.7 nM|= 229.09 nM|= 150.0 nM|= 147.0 nM|= 3.75 nM|= 39.0 nM|= 3.0 nM|= 27.54 nM|= 169.82 nM|= 15.33 nM|= 69.18 nM|= 97.7 nM|= 5.7 nM|= 19.0 nM|= 5.61 nM|= 56.23 nM|= 18.0 nM|= 1800.0 nM|= 45.3 nM|= 33.11 nM|= 30.9 nM|= 128.82 nM|= 58.88 nM|= 50.12 nM|= 5.8 nM|= 398.11 nM|= 2.03 nM|= 3.4 nM|= 10.96 nM | = 5.6 nM|= 6.0 nM|= 2.0 nM|= 1.2 nM|= 5.2 nM | | = 1.7 nM|= 2.5 nM|= 2.48 nM|= 2.8 nM|= 3.0 nM|= 3.981 nM|= 1.259 nM|= 10000.0 nM|< 50.0 nM|= 0.62 nM|= 0.9 nM|= 9.5 nM|= 2.08 nM|= 1.3 nM|= 1.4 nM|= 1.1 nM|= 5.5 nM|= 1.2 nM|= 3.6 nM|= 0.91 nM|= 4.5 nM | NPASS |
| Serotonin 2 (5-HT2) receptor | Rattus norvegicus | P14842 | | = 4600.0 nM|= 3600.0 nM|= 20.0 nM | | = 930.0 nM|= 7.8 nM|= 2950.0 nM|= 560.0 nM|= 6.0 nM|= 977.24 nM|= 950.0 nM | NPASS |
| Serotonin 1d (5-HT1d) receptor | Rattus norvegicus | P28565 | = 5.2 nM | = 3.0 nM | | | NPASS |
| Serotonin 1 (5-HT1) receptor | Rattus norvegicus | P28565 | | = 5.9 nM|= 20.0 nM | | = 2.0 nM | NPASS |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens | P16083 | | 53900 nM | | | BindingDB |
| Serotonin 2a (5-HT2a) receptor | Homo sapiens | P28223 | = 11.0 nM|= 125.89 nM|= 70.0 nM|= 5.8 nM|= 7.6 nM|= 147.91 nM|= 2.57 nM|= 150.0 nM|= 2.6 nM|= 16.0 nM|= 1.5 nM|= 1.549 nM|= 1.88 nM|= 302.0 nM|= 47.0 nM|= 2.344 nM|= 2.35 nM|= 1.6 nM|= 0.2754 nM|= 0.27 nM|= 0.51 nM|= 0.5129 nM|= 1.1 nM|= 12.1 nM|= 130.0 nM|= 3.0 nM|= 1.32 nM|= 0.23 nM|= 661.0 nM|= 2.951 nM|= 0.631 nM|= 28.0 nM|= 25.12 nM|= 1672.0 nM | = 27.9 nM | | = 14.0 nM|= 510.0 nM|= 398.11 nM|= 8.2 nM|= 120.0 nM|= 160.0 nM|= 130.0 nM|= 150.0 nM|= 320.0 nM|= 690.0 nM|= 323.59 nM|= 11.5 nM|= 17.2 nM | NPASS |
| Macrophage migration inhibitory factor | Homo sapiens | P14174 | | > 400000.0 nM | | | NPASS |
| Melatonin receptor 1A | Homo sapiens | P48039 | | | | > 100000.0 nM | NPASS |
| Melatonin receptor 1B | Homo sapiens | P49286 | | | | > 100000.0 nM | NPASS |
| Melatonin receptor type 1A | Homo sapiens | P48039 | | | | >100000 nM | BindingDB |
| Melatonin receptor type 1A | Ovis aries | P48040 | | | | >10000 nM | BindingDB |
| Melatonin receptor type 1B | Homo sapiens | P49286 | | | | >10000 nM|>100000 nM | BindingDB |
| NG108-15 | Murinae | | = 298.0 nM|= 293.0 nM | | | | NPASS |
| Norepinephrine transporter | Rattus norvegicus | | | | | 1000 nM|3013 nM|>10000 nM | BindingDB |
| Oryctolagus cuniculus | Oryctolagus cuniculus | | = 158.49 nM|= 300.0 nM | | | | NPASS |
| Polyphenol oxidase 2 | Agaricus bisporus | O42713 | | >350000 nM | | | BindingDB |
| Prostaglandin G/H synthase 1 | Homo sapiens | P23219 | | >400000 nM | | | BindingDB |
| Prostaglandin G/H synthase 2 | Homo sapiens | P35354 | | >400000 nM | | | BindingDB |
| Radical scavenging activity | | | > 250000.0 nM | | | | NPASS |
| Rattus norvegicus | Rattus norvegicus | | = 977.24 nM | = 3548.13 nM|= 28183.83 nM|= 369.0 nM | | > 5000.0 nM|= 919.0 nM|= 14092.0 nM|> 3000.0 nM | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM | | | NPASS |
| Serotonin 2a (5-HT2a) receptor | Mus musculus | P35363 | = 0.5248 nM|= 0.53 nM | | | | NPASS |
| Serotonin 7 (5-HT7) receptor | Homo sapiens | P34969 | = 15.0 nM|= 17.0 nM|= 5.754 nM|= 5.8 nM|= 7.0 nM|= 47.86 nM|= 48.0 nM|= 5.7 nM|= 5.37 nM|= 70.0 nM|= 3.66 nM|= 110.0 nM|= 9.333 nM|= 112.2 nM|= 4.5 nM | = 0.61 nM|= 2.55 nM|= 1.5 nM|= 0.49 nM|= 0.29 nM|= 0.25 nM|= 0.47 nM | = 3.98 nM | = 4.0 nM|= 8.1 nM|= 3.162 nM|= 0.22 nM|= 0.13 nM|= 0.11 nM|= 1.4 nM|= 0.8 nM|= 6.0 nM|= 0.17 nM|= 7.943 nM|= 2.12 nM|= 2.1 nM | NPASS |
| Serotonin 2b (5-HT2b) receptor | Homo sapiens | P41595 | = 1.5 nM|= 25.12 nM|= 5.8 nM|= 0.5 nM|= 11.0 nM|= 0.86 nM|= 1.1 nM|= 1.072 nM|= 0.92 nM|= 1.445 nM|= 1.46 nM|= 4.5 nM|= 0.8511 nM|= 0.07079 nM|= 2.4 nM|= 1.19 nM|= 1.259 nM | | | = 12.0 nM|= 13.0 nM|= 13.49 nM|= 10.8 nM | NPASS |
| Sodium-dependent dopamine transporter | Rattus norvegicus | P23977 | | | | >10000 nM|2703 nM | BindingDB |
| Sodium-dependent serotonin transporter | Rattus norvegicus | P31652 | | | | 740 nM | BindingDB |
| Solute carrier family 22 member 1 | Rattus norvegicus | Q63089 | | | | 390000 nM|= 390000.0 nM | BindingDB, NPASS |
| Solute carrier family 22 member 2 | Rattus norvegicus | Q9R0W2 | | | | 242000 nM|= 242000.0 nM | BindingDB, NPASS |
| Solute carrier family 22 member 3 | Rattus norvegicus | O88446 | | 97000 nM|= 97000.0 nM | | | BindingDB, NPASS |
| Sortase | Staphylococcus aureus | Q9S446 | | > 100.0 ug.mL-1 | | | NPASS |
| Sodium-dependent dopamine transporter | Homo sapiens | Q01959 | | | | >10000 nM | BindingDB |
| Synaptic vesicular amine transporter | Homo sapiens | Q05940 | | 1430 nM|= 1430.0 nM | | 7690 nM|640000 nM|2290 nM|= 7690.0 nM|= 640000.0 nM|= 2290.0 nM | BindingDB, NPASS |
| Trace amine-associated receptor 1 | Homo sapiens | Q96RJ0 | 35100 nM|= 35100.0 nM | | | | BindingDB, NPASS |
| Tyrosinase | Agaricus bisporus | O42713 | | > 350000.0 nM | | | NPASS |
| Tyrosinase | Mus musculus | P11344 | | 550000 nM|= 550000.0 nM | | | BindingDB, NPASS |
| Vascular endothelial growth factor receptor 2 | Homo sapiens | P35968 | | >50000 nM | | | BindingDB |
| Vascular endothelial growth factor receptor 3 | Homo sapiens | P35916 | | >50000 nM | | | BindingDB |
| Isocitrate lyase | Candida albicans | Q9P8Q7 | | 301000 nM|301300 nM|= 301300.0 nM|= 301000.0 nM|= 53.0 ug.mL-1 | | | BindingDB, NPASS |
| Synaptic vesicular amine transporter | Mus musculus | Q8BRU6 | | 98 nM|= 98.0 nM | | | BindingDB, NPASS |
| Serotonin transporter | Rattus norvegicus | P31652 | | | | = 740.0 nM | NPASS |
| Serotonin receptor 2a and 2c (5HT2A and 5HT2C) | Rattus norvegicus | P14842 | | | | = 10.6 nM|= 6.1 nM|= 600.0 nM | NPASS |
| Serotonin 7 (5-HT7) receptor | Rattus norvegicus | P32305 | | | | = 10.0 nM|= 0.6026 nM|= 7.33 nM | NPASS |
| Serotonin 2b (5-HT2b) receptor | Rattus norvegicus | P30994 | = 3.5 nM|= 4.19 nM | | | | NPASS |
| Serotonin 2c (5-HT2c) receptor | Homo sapiens | P28335 | = 1.7 nM|= 25.12 nM|= 24.0 nM|= 0.09 nM|= 25.0 nM|= 1.63 nM|= 43.65 nM|= 0.871 nM|= 44.0 nM|= 0.87 nM|= 0.4 nM|= 0.3467 nM|= 0.21 nM|= 190.55 nM|= 0.182 nM|= 0.17 nM|= 15.14 nM|= 15.0 nM|= 0.1905 nM|= 0.19 nM|= 0.41 nM|= 0.166 nM|= 0.1349 nM|= 0.14 nM|= 21.88 nM|= 21.0 nM|= 0.12 nM|= 1.202 nM|= 0.1259 nM|= 1.2 nM | = 81.0 nM|= 1.25 nM | | = 35.0 nM|= 6.9 nM|= 50.12 nM|= 8.3 nM|= 130.0 nM|= 20.0 nM|= 445.0 nM|= 214.0 nM|= 79.43 nM|= 79.0 nM | NPASS |
| Serotonin 2c (5-HT2c) receptor | Rattus norvegicus | P08909 | = 2.8 nM | = 81.0 nM|= 42.0 nM | | = 31.62 nM|= 23.0 nM|= 10.0 nM | NPASS |
| Serotonin 3 (5-HT3) receptor | Homo sapiens | Q8WXA8 | | | | = 144.54 nM|= 120.0 nM | NPASS |
| Serotonin 3 (5-HT3) receptor | Rattus norvegicus | Q9JJ16 | | = 727.0 nM | | = 398.11 nM|= 320.0 nM|= 66.0 nM|= 120.0 nM|= 87.0 nM|= 390.0 nM | NPASS |
| Serotonin 3 receptor (5HT3) | Mus musculus | P23979 | | | | = 361.0 nM | NPASS |
| Serotonin 3a (5-HT3a) receptor | Homo sapiens | P46098 | = 500.0 nM|= 457.09 nM|= 178.0 nM|= 141.0 nM | | | | NPASS |
| Serotonin 3a (5-HT3a) receptor | Mus musculus | P23979 | = 3400.0 nM|= 24000.0 nM|= 3300.0 nM|= 170000.0 nM|= 37000.0 nM|= 20900.0 nM|= 17200.0 nM|= 9600.0 nM|= 90000.0 nM|= 4400.0 nM|= 210000.0 nM|= 140000.0 nM|= 49000.0 nM|= 7100.0 nM|= 980.0 nM|= 51000.0 nM|= 11000.0 nM|= 6200.0 nM|= 5100.0 nM|= 2900.0 nM|= 27000.0 nM|= 1300.0 nM|= 1320.0 nM|= 63000.0 nM|= 42000.0 nM|= 15000.0 nM | | | | NPASS |
| Serotonin 3a (5-HT3a) receptor | Rattus norvegicus | P35563 | = 12000.0 nM | | | | NPASS |
| Serotonin 4 (5-HT4) receptor | Cavia porcellus | O70528 | = 5.0 nM|= 10.0 nM | | | = 100.0 nM|= 230.0 nM | NPASS |
| Serotonin 4 (5-HT4) receptor | Homo sapiens | Q13639 | = 100.0 nM|= 12.0 nM | = 323.0 nM | | = 1049.0 nM|= 500.0 nM|= 29.51 nM|= 109.65 nM|= 246.0 nM | NPASS |
| Serotonin 4 (5-HT4) receptor | Rattus norvegicus | Q62758 | = 6.31 nM|= 17.1 nM | = 3.7 nM|= 147.0 nM | | = 187.0 nM|= 37.4 nM | NPASS |
| Serotonin 5a (5-HT5a) receptor | Homo sapiens | P47898 | | = 79.0 nM|= 180.0 nM|= 184.0 nM|= 280.0 nM|= 160.0 nM|= 260.0 nM | | = 250.0 nM|= 126.0 nM|= 110.0 nM|= 170.0 nM|= 82.0 nM|= 130.0 nM | NPASS |
| Serotonin 5a (5-HT5a) receptor | Mus musculus | P30966 | | | | = 150.0 nM | NPASS |
| Serotonin 6 (5-HT6) receptor | Homo sapiens | P50406 | = 43.6 nM|= 42.1 nM | = 200.0 nM|= 262.0 nM|= 27.5 nM|= 180.0 nM|= 100.0 nM|= 120.0 nM|= 130.0 nM | | = 65.0 nM|= 78.0 nM|= 75.0 nM|= 125.89 nM|= 100.0 nM|= 93.0 nM|= 84.0 nM|= 70.0 nM|= 50.0 nM|= 33.0 nM|= 61.0 nM | NPASS |
| Serotonin 2a (5-HT2a) receptor | Rattus norvegicus | P14842 | = 351.0 nM|= 55.8 nM|= 57.9 nM | = 0.9 nM|= 2350.0 nM|= 0.94 nM|= 13000.0 nM|= 30600.0 nM|= 600.0 nM | | = 1258.93 nM|= 0.3 nM|= 1258.0 nM|= 10.6 nM|= 600.0 nM | NPASS |
| Insulin-like growth factor 1 receptor | Homo sapiens | P08069 | | >50000 nM | | | BindingDB |
| D(1A) dopamine receptor | Rattus norvegicus | P18901 | | | | 5000 nM | BindingDB |
| Dopamine receptor D4 | Canis lupus familiaris | | | | | 4180 nM | BindingDB |
| 5-hydroxytryptamine receptor 1F | Mus musculus | Q02284 | | | | 125.89 nM | BindingDB |
| 5-hydroxytryptamine receptor 1F | Rattus norvegicus | P30940 | | | | 67.6 nM | BindingDB |
| 5-hydroxytryptamine receptor 2A | Homo sapiens | P28223 | 11 nM|1.9 nM|302 nM|5.8 nM|47 nM|2.3 nM|2.4 nM|70 nM|7.6 nM|2.6 nM|150 nM|1.6 nM|126 nM|0.275423 nM|0.270000 nM|0.510000 nM|0.512861 nM|1.1 nM|12 nM|130 nM|661 nM|1672 nM | 28 nM | | 63.09 nM|12.02 nM|602.55 nM|7.77 nM|218.77 nM|30.90 nM|341 nM|21 nM|16.22 nM|20.0 nM|510 nM|320 nM|160 nM|150 nM|120 nM|14 nM|8.2 nM|690 nM|8.20 nM|130 nM|12 nM|398 nM|17 nM | BindingDB |
| 5-hydroxytryptamine receptor 2A | Mus musculus | P35363 | 0.524807 nM|0.530000 nM | | | | BindingDB |
| 5-hydroxytryptamine receptor 2A/2B/2C | Mus musculus | P34968|P35363|Q02152 | | 680 nM | | 500 nM | BindingDB |
| 5-hydroxytryptamine receptor 2B | Bos taurus | | | | | 750 nM | BindingDB |
| 5-hydroxytryptamine receptor 1F | Homo sapiens | P30939 | 7.9 nM | | | 10 nM|>10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 2B | Homo sapiens | P41595 | 1.5 nM|0.920000 nM|0.5 nM|11 nM|1.4 nM|5.8 nM|0.86 nM|4.5 nM|25 nM|0.860000 nM|0.851138 nM|0.070795 nM | | | 0.79 nM|9.8 nM|9.46 nM|1.17 nM|2.09 nM|4 nM|1 nM|19 nM|13.49 nM|12 nM|13 nM|11 nM | BindingDB |
| 5-hydroxytryptamine receptor 2B | Rattus norvegicus | P30994 | 3.5 nM|4.2 nM | | | 10 nM|28.18 nM|10.23 nM|10.2 nM|11.3 nM | BindingDB |
| 5-hydroxytryptamine receptor 2C | Homo sapiens | P28335 | 1.7 nM|0.210000 nM|191 nM|0.09 nM|25 nM|15 nM|0.170000 nM|0.181970 nM|24 nM|1.63 nM|0.870000 nM|44 nM|0.190546 nM|0.190000 nM|0.410000 nM|0.165959 nM|0.134896 nM|0.140000 nM|22 nM|21 nM | 278 nM|81 nM|1.3 nM | | 656 nM|15.5 nM|56.23 nM|5.75 nM|2.9 nM|18.20 nM|2.4 nM|130 nM|6.9 nM|8.3 nM|20 nM|35 nM|8.30 nM|214 nM|445 nM|79 nM|50 nM | BindingDB |
| 5-hydroxytryptamine receptor 2C | Rattus norvegicus | P08909 | 2.8 nM | 81 nM|42 nM | 32 nM | 0.7 nM|22.9 nM|87.09 nM|44 nM|11 nM|159 nM|12.2 nM|10 nM|23 nM | BindingDB |
| 5-hydroxytryptamine receptor 3A | Cavia porcellus | O70212 | | | | >10000 nM|495 nM | BindingDB |
| 5-hydroxytryptamine receptor 3A | Homo sapiens | P46098 | 141 nM|178 nM|457 nM | | | | BindingDB |
| 5-hydroxytryptamine receptor 3A | Mus musculus | P23979 | 3400 nM | | | 269.15 nM|292 nM|361 nM | BindingDB |
| 5-hydroxytryptamine receptor 2B | Mus musculus | Q02152 | | | | 1258.92 nM | BindingDB |
| 5-hydroxytryptamine receptor 1E | Rattus norvegicus | | | | | 7 nM | BindingDB |
| 5-hydroxytryptamine receptor 1E | Homo sapiens | P28566 | | | | 11 nM|3.5 nM|10.96 nM|7.24 nM|6.16 nM|2.3 nM|4 nM | BindingDB |
| 5-hydroxytryptamine receptor 1D | Sus scrofa | P79400 | | 10 nM|10.0 nM | | | BindingDB |
| Epidermal growth factor receptor | Homo sapiens | P00533 | | >50000 nM | | | BindingDB |
| 5-hydroxytryptamine 1D receptor | Bos taurus | | | | | 4 nM|1.9 nM | BindingDB |
| 5-hydroxytryptamine receptor 1A | Homo sapiens | P08908 | 10 nM|1 nM|3.0 nM|1.000 nM|0.700000 nM|28 nM|170 nM|43 nM|15 nM|3.7 nM|150 nM|69 nM|147 nM|3.8 nM|98 nM|5.7 nM|19 nM|8.7 nM|229 nM|5.6 nM|5.61 nM|18 nM|1800 nM|45 nM|33 nM|31 nM|129 nM|59 nM|50 nM|5.8 nM|2.0 nM | 5.2 nM|6 nM|2 nM|5.6 nM|1.2 nM | 3.2 nM | 0.26 nM|1.25 nM|12.58 nM|0.79 nM|3.98 nM|102.32 nM|102.3 nM|1.3 nM|3 nM|2.8 nM|1.7 nM|2.48 nM|2.5 nM|2.1 nM|0.62 nM|10 nM|10000 nM|0.900000 nM|1.4 nM|4.0 nM|5.5 nM|1.2 nM|3.6 nM|3.0 nM|0.910000 nM|4.5 nM | BindingDB |
| 5-hydroxytryptamine receptor 1A | Human | P08908 | | | | 1.2 nM|10.0 nM | BindingDB |
| 5-hydroxytryptamine receptor 1A | Mus musculus | Q64264 | | 5 nM | | | BindingDB |
| 5-hydroxytryptamine receptor 1A | Rattus norvegicus | P19327 | 10 nM|323 nM | 5.2 nM|3 nM|2.6 nM | | 46.77 nM|134 nM|4.2 nM|0.12 nM|90 nM|2 nM|1.7 nM|3 nM|1.6 nM|4.3 nM|2.1 nM|7.3 nM|2.6 nM|4.8 nM|1.9 nM|2.3 nM | BindingDB |
| 5-hydroxytryptamine receptor 1A/1B/1D/1F | Rattus norvegicus | P19327|P28564|P28565|P30940 | | 20 nM | | 2 nM | BindingDB |
| 5-hydroxytryptamine receptor 1B | Cavia porcellus | O08892 | | | | 2.51 nM | BindingDB |
| 5-hydroxytryptamine receptor 1B | Homo sapiens | P28222 | 30 nM|4.82 nM|4.7 nM | 5 nM | | 0.59 nM|3.9 nM|4.26 nM|1.09 nM|3.98 nM|0.57 nM|15.84 nM|7.94 nM|38 nM|9 nM|4.07 nM|6.8 nM|4 nM|1.1 nM|7.1 nM|4.8 nM|14 nM|5.0 nM | BindingDB |
| 5-hydroxytryptamine receptor 1B | Mus musculus | P28334 | | | | 39.81 nM | BindingDB |
| 5-hydroxytryptamine receptor 1B | Rattus norvegicus | P28564 | 26 nM | 5 nM|4.9 nM|4.6 nM | | 14 nM|15.84 nM|5.24 nM|3.01 nM|0.57 nM|3 nM|2.6 nM|5 nM|5.4 nM|3.5 nM|25 nM|2.5 nM|1.1 nM | BindingDB |
| 5-hydroxytryptamine receptor 1D | Canis lupus familiaris | P11614 | | | | 5.01 nM|15.84 nM | BindingDB |
| 5-hydroxytryptamine receptor 1D | Cavia porcellus | Q60484 | 8.5 nM|16 nM|5.2 nM | 3 nM | | | BindingDB |
| 5-hydroxytryptamine receptor 1D | Homo sapiens | P28221 | | 3 nM | 13 nM | 4.3 nM|8.9 nM|2.1 nM|8.91 nM|2.08 nM|3.89 nM|3.98 nM|3.4 nM|3.38 nM|3 nM|5.5 nM|1.7 nM|5.06 nM|5.1 nM|2 nM|0.500000 nM|4.8 nM | BindingDB |
| 5-hydroxytryptamine receptor 1D | Rattus norvegicus | P28565 | 5.2 nM | 3 nM | | 2.51 nM|18 nM | BindingDB |
| 5-hydroxytryptamine receptor 3A | Rattus norvegicus | P35563 | 12000 nM | | | | BindingDB |
| 5-hydroxytryptamine receptor 3A/3B | Rattus norvegicus | P35563|Q9JJ16 | | 727 nM | | 87 nM|320 nM|390 nM|66 nM|120 nM | BindingDB |
| 5-hydroxytryptamine receptor 2A | Rattus norvegicus | P14842 | 58 nM|55.8 nM|351 nM | 0.940000 nM|2350 nM|0.9 nM|13000 nM|30600 nM|600 nM | | 3 nM|270 nM|83 nM|125.89 nM|5.75 nM|1.99 nM|478.63 nM|707.94 nM|251.18 nM|2955 nM|120.22 nM|96 nM|1258 nM|11 nM|600 nM|0.3 nM | BindingDB |
| 5-hydroxytryptamine receptor 4 | Homo sapiens | Q13639 | 12 nM|100 nM | 323 nM | | 1049 nM|316.22 nM|56.23 nM|1151 nM|481.9 nM|330 nM|251.18 nM|158.5 nM|100 nM|500 nM|29.51 nM|109.65 nM|246 nM | BindingDB |
| Canis familiaris | Canis lupus familiaris | | = 210.0 nM | | | | NPASS |
| Cyclooxygenase-1 | Homo sapiens | P23219 | | > 400000.0 nM | | | NPASS |
| Cyclooxygenase-2 | Homo sapiens | P35354 | | > 400000.0 nM | | | NPASS |
| D(1A) dopamine receptor | Homo sapiens | P21728 | | | 9690 nM | >10000 nM | BindingDB |
| D(1B) dopamine receptor | Homo sapiens | P21918 | | | | 3000 nM | BindingDB |
| D(2) dopamine receptor | Canis lupus familiaris | Q9GJU1 | | | | >10000 nM | BindingDB |
| B16 | Mus musculus | | | > 30000.0 nM | | | NPASS |
| D(2) dopamine receptor | Homo sapiens | P14416 | | 0.000 nM | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 4 | Cavia porcellus | O70528 | 5 nM|10 nM | | | 79.43 nM|50.11 nM|39.81 nM|230 nM|100 nM | BindingDB |
| D(3) dopamine receptor | Rattus norvegicus | P19020 | | | | 2338 nM | BindingDB |
| Dopamine D1 receptor | Homo sapiens | P21728 | | | = 9690.0 nM | | NPASS |
| Dopamine D2 receptor | Homo sapiens | P14416 | | = 0.0003 nM | | | NPASS |
| Dopamine D3 receptor | Homo sapiens | P35462 | = 523.0 nM | | | | NPASS |
| Dopamine D3 receptor | Rattus norvegicus | P19020 | | | | = 2338.0 nM | NPASS |
| D(2) dopamine receptor | Rattus norvegicus | P61169 | | | | >10000 nM|1655 nM|7950 nM | BindingDB |
| Alpha-glucosidase MAL62 | Saccharomyces cerevisiae | P07265 | | >300000 nM|> 300000.0 nM | | | BindingDB, NPASS |
| D(3) dopamine receptor | Homo sapiens | P35462 | 523 nM | | | | BindingDB |
| Alpha-1A adrenergic receptor | Rattus norvegicus | P43140 | | | | 18000 nM|23000 nM | BindingDB |
| 5-hydroxytryptamine receptor 4 | Mus musculus | P97288 | | | | 79.43 nM|56.23 nM | BindingDB |
| Alpha-2C adrenergic receptor | Rattus norvegicus | P22086 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 4 | Rattus norvegicus | Q62758 | 17 nM|6.3 nM | 3.7 nM|147 nM | | 145 nM|200 nM|6.3 nM|7.94 nM|125.89 nM|199.52 nM|158.48 nM|38.9 nM|37 nM|187 nM | BindingDB |
| 5-hydroxytryptamine receptor 5A | Homo sapiens | P47898 | | 180 nM|260 nM|79 nM | | 126 nM|130 nM|250 nM|170 nM | BindingDB |
| 5-hydroxytryptamine receptor 5A | Rattus norvegicus | P35364 | | | | 1333 nM|239.88 nM | BindingDB |
| 5-hydroxytryptamine receptor 5B | Mus musculus | P31387 | | | | 251.18 nM | BindingDB |
| 5-hydroxytryptamine receptor 5B | Rattus norvegicus | P35365 | | | | 239 nM|1318.25 nM|7.76 nM|7.8 nM | BindingDB |
| 5-hydroxytryptamine receptor 6 | Homo sapiens | P50406 | 44 nM|42 nM | 120 nM|27.5 nM|130 nM | | 56 nM|65 nM|33 nM|75 nM|78 nM|61 nM|100 nM|84 nM|126 nM|70 nM | BindingDB |
| 5-hydroxytryptamine receptor 5A | Mus musculus | P30966 | | | | 251.18 nM|1100 nM|150 nM | BindingDB |
| 5-hydroxytryptamine receptor 6 | Rattus norvegicus | P31388 | | | | 151 nM|56 nM|151.35 nM|56.23 nM|12.58 nM|234.42 nM|79.43 nM | BindingDB |
| 5-hydroxytryptamine receptor 7 | Rattus norvegicus | P32305 | | | | 1.81 nM|4.89 nM|1.51 nM|25.11 nM|0.6 nM|1.83 nM|1.52 nM|5 nM|2.00 nM|0.63 nM|7.94 nM|0.13 nM|7.33 nM|10 nM|0.602560 nM | BindingDB |
| 5-hydroxytryptamine receptor 7 | Cavia porcellus | P50407 | | | | 1 nM|1.34 nM|0.25 nM|0.10 nM | BindingDB |
| 5-hydroxytryptamine receptor 7 | Homo sapiens | P34969 | 17 nM|15 nM|5.8 nM|48 nM|7.0 nM|5.4 nM|5.7 nM|70 nM|3.7 nM|9.3 nM|9.33 nM|112 nM|110 nM | 0.250 nM|2.55 nM|0.470000 nM | 4.0 nM | 8.12 nM|8.1 nM|7.94 nM|0.40 nM|0.38 nM|6.31 nM|1.4 nM|0.800000 nM|4 nM|6.0 nM|0.170000 nM|0.13 nM|3.2 nM|7.9 nM|2.1 nM | BindingDB |
| 5-hydroxytryptamine receptor 6 | Mus musculus | Q9R1C8 | | | | 39.81 nM|5.01 nM|95.50 nM | BindingDB |
| 5-hydroxytryptamine receptor 7 | Mus musculus | P32304 | | | | 5.01 nM | BindingDB |