| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Histamine H3 receptor | Homo sapiens | Q9Y5N1 | | | | 0.500000 nM | BindingDB |
| Melatonin receptor | Oryctolagus cuniculus | | | | | 6.3 nM|0.37 nM | BindingDB |
| Melatonin receptor type 1A | Homo sapiens | P48039 | 1.92 nM|2.24 nM|0.098000 nM|1.5 nM|0.026 nM|2.2 nM|1.000000 nM|0.110000 nM|0.022000 nM | 0.600000 nM|0.2 nM|0.110 nM|0.200000 nM|1 nM | | 1.48 nM|0.88 nM|0.08 nM|0.56 nM|0.66 nM|0.29 nM|0.2 nM|0.120000 nM|0.12 nM|0.0823 nM|0.14 nM|0.140000 nM|0.400000 nM|0.530000 nM|0.3 nM|0.39 nM|0.091000 nM|0.525 nM|0.250000 nM|0.230000 nM|0.130000 nM|0.200000 nM|0.296 nM|0.25 nM|0.24 nM|0.22 nM|0.660 nM|0.37 nM|0.304 nM|0.331 nM|0.263 nM|0.296000 nM|0.204174 nM|0.288403 nM|0.165959 nM|0.263027 nM|0.141254 nM|0.880000 nM|0.460000 nM|0.660000 nM|0.270000 nM|0.180000 nM|0.240000 nM | BindingDB |
| Melatonin receptor type 1A | Ovis aries | P48040 | | | | 0.24 nM | BindingDB |
| Melatonin receptor type 1A | Sus scrofa | O02781 | | | | 0.25 nM|0.24 nM | BindingDB |
| Melatonin receptor type 1A/1B | Homo sapiens | P48039|P49286 | | 0.017000 nM|0.157000 nM|3.1 nM|2.2 nM|15 nM|3.0 nM|13 nM | 0.091500 nM | 0.082300 nM|0.140000 nM|0.410000 nM|0.091500 nM|1.1 nM|0.610000 nM | BindingDB |
| Melatonin receptor type 1B | Homo sapiens | P49286 | 0.47 nM|0.49 nM|0.069000 nM|0.42 nM|0.82 nM|25 nM|0.070000 nM|0.850000 nM | 0.300000 nM|0.53 nM|0.530000 nM | | 1.11 nM|0.23 nM|0.18 nM|0.38 nM|0.19 nM|0.48 nM|0.33 nM|0.25 nM|0.12 nM|0.53 nM|0.310000 nM|0.31 nM|0.195 nM|0.41 nM|0.410000 nM|0.300000 nM|0.320000 nM|0.7 nM|0.35 nM|0.150000 nM|0.3 nM|0.741 nM|0.340000 nM|0.520000 nM|0.230000 nM|0.290000 nM|0.429 nM|0.34 nM|0.21 nM|0.617 nM|0.339 nM|0.500000 nM|0.429000 nM|0.288403 nM|0.281838 nM|0.295121 nM|0.338844 nM|0.239883 nM|0.950000 nM|0.301995 nM|0.330000 nM|0.180000 nM|0.130000 nM|0.120000 nM|0.210000 nM | BindingDB |
| Cytochrome P450 1B1 | Homo sapiens | Q16678 | | | | 14000 nM | BindingDB |
| Melatonin receptor type 1B | Gallus gallus | P51050 | | | | 1.21 nM|1.2 nM|0.700000 nM | BindingDB |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens | P16083 | | 11300 nM|65 nM|6600 nM|64.57 nM | | 57 nM|28 nM | BindingDB |
| Melatonin receptor type 1C | Gallus gallus | P49288 | 23 nM | | | 0.590000 nM|0.670000 nM|0.176000 nM|1.1 nM|0.460000 nM|0.676083 nM|0.700000 nM | BindingDB |
| Melatonin receptor type 1C | Xenopus laevis | P49219 | 0.079433 nM | | | 1.87 nM|1.86 nM | BindingDB |
| Myeloperoxidase | Homo sapiens | P05164 | | 3000 nM | | | BindingDB |
| Melatonin receptor type 1A/1B/1C | Gallus gallus | P49285|P49288|P51050 | | | | 0.570000 nM | BindingDB |
| Cytochrome P450 1A2 | Homo sapiens | P05177 | | | | 12000 nM | BindingDB |
| 5-hydroxytryptamine receptor 5A | Rattus norvegicus | P35364 | | | | 1000 nM | BindingDB |
| Carboxylic ester hydrolase | Equus caballus | | | >100 nM | | | BindingDB |
| Cytochrome P450 1A1 | Homo sapiens | P04798 | | | | 59000 nM | BindingDB |
| 5-hydroxytryptamine receptor 2A | Homo sapiens | P28223 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 2A | Rattus norvegicus | P14842 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 2C | Homo sapiens | P28335 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 2C | Sus scrofa | | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 5B | Rattus norvegicus | P35365 | | | | 1000 nM | BindingDB |
| 5-hydroxytryptamine receptor 2B | Homo sapiens | P41595 | | | | >10000 nM|5754.40 nM | BindingDB |
| ATP-binding cassette sub-family C member 2 | Homo sapiens | Q92887 | | >133000 nM | | | BindingDB |
| ATP-binding cassette sub-family C member 3 | Homo sapiens | O15438 | | >133000 nM | | | BindingDB |
| ATP-binding cassette sub-family C member 4 | Homo sapiens | O15439 | | >133000 nM | | | BindingDB |
| Acetylcholinesterase | Bos taurus | P23795 | | >100 nM | | | BindingDB |
| Bile salt export pump | Homo sapiens | O95342 | | >133000 nM | | | BindingDB |
| 5-hydroxytryptamine receptor 7 | Rattus norvegicus | P32305 | | | | 1000 nM | BindingDB |