| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Macrophage migration inhibitory factor | Homo sapiens | P14174 | | = 73600.0 nM | | = 62000.0 nM | NPASS |
| Histamine H4 receptor | Homo sapiens | Q9H3N8 | 12 nM|75 nM|1800 nM|11.6 nM|12.02 nM|9.12 nM|25.12 nM|= 75.0 nM|= 54.95 nM|= 20.89 nM|= 1800.0 nM|= 11.6 nM|= 12.02 nM|= 11.75 nM|= 13.8 nM|= 9.12 nM|= 12.59 nM|= 19.95 nM|= 79.43 nM|= 25.12 nM|= 20.42 nM|= 7.943 nM|= 11.0 nM|= 13.0 nM|= 7.413 nM|= 16.98 nM|= 33.88 nM | | = 5.0 nM|= 16.0 nM | 16 nM|8.1 nM|3442.3 nM|17 nM|2.5 nM|39.8 nM|60 nM|9 nM|13.4 nM|12.02 nM|15.85 nM|= 14.45 nM|= 7.943 nM|= 12.02 nM|= 13.4 nM|= 60.0 nM|= 12.59 nM|= 15.85 nM|= 9.0 nM|= 19.95 nM|= 4.8 nM|= 8.0 nM|= 1.6 nM|= 1.0 nM|= 25.12 nM | BindingDB, NPASS |
| Histamine H4 receptor | Mus musculus | Q91ZY2 | = 5011.87 nM|= 94.0 nM|= 6760.83 nM|= 87.1 nM|= 2344.23 nM | | = 42.0 nM | = 79.43 nM|= 42.0 nM | NPASS |
| Histamine H4 receptor | Rattus norvegicus | Q91ZY1 | = 158.49 nM|= 52480.75 nM|= 295.12 nM|= 3715.35 nM | | = 134.0 nM | = 63.1 nM|= 136.0 nM | NPASS |
| Histamine receptor H4 | Cavia porcellus | | | | | 0.14 nM|104 nM | BindingDB |
| Hrh3 protein | Rattus norvegicus | | | | | 11 nM|100 nM|7.3 nM|62 nM|5.3 nM|25.11 nM|10 nM|158.48 nM|2.51 nM|12 nM|13.2 nM|4.9 nM|2.66 nM | BindingDB |
| Nischarin | Rattus norvegicus | Q4G017 | | | | >10000 nM | BindingDB |
| Trace amine-associated receptor 1 | Homo sapiens | Q96RJ0 | | | | 3107 nM | BindingDB |
| Rattus norvegicus | Rattus norvegicus | | = 62.0 nM|= 4466.84 nM | | | | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM | | | NPASS |
| Solute carrier family 22 member 1 | Rattus norvegicus | Q63089 | | | | 141000 nM|1400000 nM|= 1400000.0 nM|= 141000.0 nM | BindingDB, NPASS |
| Histamine H4 receptor | Cavia porcellus | Q91ZY3 | | | | = 6.0 nM | NPASS |
| Solute carrier family 22 member 2 | Rattus norvegicus | Q9R0W2 | | | | 171000 nM|390000 nM|= 171000.0 nM|= 390000.0 nM | BindingDB, NPASS |
| Solute carrier family 22 member 3 | Homo sapiens | O75751 | | | | 140000 nM|= 140000.0 nM | BindingDB, NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 660.0 nM | | | NPASS |
| Histamine H3 receptor | Rattus norvegicus | Q9QYN8 | 62 nM | | | = 6.31 nM | BindingDB, NPASS |
| Bile salt export pump | Homo sapiens | O95342 | | > 1000000.0 nM | | | NPASS |
| Histamine H3 receptor | Homo sapiens | Q9Y5N1 | 25 nM|640 nM|77 nM|88 nM|25.1 nM|25.12 nM|12.88 nM|15.85 nM|= 77.0 nM|= 9.772 nM|= 4.074 nM|= 88.0 nM|= 25.1 nM|= 25.12 nM|= 12.88 nM|= 640.0 nM|= 5.012 nM|= 15.85 nM|= 13.0 nM|= 2.512 nM|= 63.1 nM|= 30.0 nM|= 4.0 nM | | = 3.0 nM | 10 nM|>10000 nM|15.2 nM|5.4 nM|2.32 nM|2.61 nM|5.2 nM|11.75 nM|6.31 nM|= 9.333 nM|= 33.88 nM|= 5.2 nM|= 10.0 nM|= 11.75 nM|= 6.31 nM|= 16.0 nM|= 12.8 nM|= 12.59 nM|= 2.512 nM|= 501.19 nM|= 389.05 nM|= 25.12 nM|= 1174.9 nM|= 25.7 nM|= 588.84 nM | BindingDB, NPASS |
| Histamine H3 receptor | Mus musculus | P58406 | | | | 68 nM|= 68.0 nM | BindingDB, NPASS |
| 5-hydroxytryptamine receptor 7 | Rattus norvegicus | P32305 | | | | 1000 nM|>10000 nM | BindingDB |
| Cavia porcellus | Cavia porcellus | | = 980.0 nM|= 240.0 nM|= 1000.0 nM|= 140.0 nM|= 199.53 nM|= 2238.72 nM|= 316.23 nM | | = 0.8511 nM | | NPASS |
| D(1A) dopamine receptor | Rattus norvegicus | P18901 | | | | >10000 nM | BindingDB |
| D(2) dopamine receptor | Rattus norvegicus | P61169 | | | | >10000 nM | BindingDB |
| Glutaminyl-peptide cyclotransferase | Homo sapiens | Q16769 | | | | 850000 nM | BindingDB |
| 5-hydroxytryptamine receptor 7 | Homo sapiens | P34969 | | | | >10000 nM | BindingDB |
| Histamine H1 receptor | Homo sapiens | P35367 | 191 nM|13 nM|45 nM|190 nM|190.55 nM|= 13.0 nM|= 45.0 nM|= 190.0 nM|= 190.55 nM|= 199.53 nM | 158 nM|= 158.49 nM|~ 1000.0 nM | = 4.5 nM | >10000 nM|1258.92 nM|1258.93 nM|2060 nM|7010 nM|190 nM|79432.82 nM|= 15848931924611.11 nM|= 79432.82 nM|= 1000000.0 nM|= 39810.72 nM|= 19952.62 nM|= 31622.78 nM|= 12589.25 nM|= 6000.0 nM|= 2398.83 nM | BindingDB, NPASS |
| Histamine H1 receptor | Rattus norvegicus | P31390 | = 4466.84 nM | | = 10.0 nM | >10000 nM | BindingDB, NPASS |
| Histamine H2 receptor | Cavia porcellus | P47747 | 1000 nM|1200 nM|1202.26 nM|= 1000.0 nM|= 1200.0 nM|= 1202.26 nM|= 691.83 nM|= 251.19 nM | | 69183 nM|= 69183.1 nM | >10000 nM|1200 nM | BindingDB, NPASS |
| Histamine H2 receptor | Homo sapiens | P25021 | 1202 nM|463 nM|650 nM|1200 nM|1258.93 nM|1202.26 nM|= 463.0 nM|= 650.0 nM|= 1200.0 nM|= 1202.26 nM|= 1258.93 nM|= 1584.89 nM|= 1412.54 nM|= 3801.89 nM|= 5495.41 nM|= 114.82 nM|= 977.24 nM | | = 12.2 nM | >10000 nM|1200 nM|= 50118.72 nM|= 5000.0 nM|= 295.12 nM|= 263.03 nM | BindingDB, NPASS |
| Histamine H2 receptor | Rattus norvegicus | P25102 | | | 117490 nM|= 117489.76 nM | 17 nM | BindingDB, NPASS |
| Histamine H3 receptor | Cavia porcellus | Q9JI35 | | | | 100 nM|= 0.1445 nM|= 10.47 nM | BindingDB, NPASS |
| Histamine H1 receptor | Cavia porcellus | P31389 | = 870963589956083.2 nM|= 199.53 nM|= 162.18 nM | | = 0.8511 nM|= 0.7762 nM|= 1.0 nM|= 10.0 nM | 3162.27 nM|>10000 nM|9900 nM|4650 nM|4600 nM | BindingDB, NPASS |
