IMPPAT Phytochemical information: 
Cocaine

Cocaine
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Sodium-dependent dopamine transporterBos taurusP27922139 nM|65 nMBindingDB
Sodium-dependent serotonin transporterRattus norvegicusP316521050 nM|737 nM|1045 nM|207 nM|1059 nM389 nM|304 nM|401 nM|177 nM|413 nM|96 nM|160 nM|95 nM|155 nM|130 nM|293 nMBindingDB
Sodium-dependent serotonin transporterHomo sapiensP31645318 nM|416 nM318 nM|325 nM|270 nM|413 nM|277 nM601 nM|276 nM|297 nM|155 nM|229 nM|657 nM|632 nMBindingDB
Sodium-dependent noradrenaline transporterHomo sapiensP23975385 nM|835 nM385 nM|186 nM|192 nM|221 nM830 nM|1115 nM|2420 nM|108 nM|645 nM|2410 nM|10700 nM|2357 nMBindingDB
TransporterRattus norvegicus3300 nM|3520 nM|3530 nM|3825 nM108 nM|186 nM|1900 nM|190 nM|2000 nM|3302 nMBindingDB
Sodium-dependent dopamine transporterRattus norvegicusP23977297 nM|266 nM|102 nM|1810 nM|843 nM|66 nM|150 nM|15800 nM|89 nM|511 nM|221 nM|580 nM|1450 nM|139 nM690 nM|600 nM|102 nM|104 nM|150 nM|475 nM|478 nM|160 nM|275 nM|555 nM|128 nM|320 nM|280 nM|230 nM|420 nM|301 nM|259 nM|146 nM|270 nM|460 nM|187 nM|423 nM|74 nMBindingDB
Sodium-dependent dopamine transporterMus musculusQ61327200 nM850 nMBindingDB
Sodium-dependent dopamine transporterMacaca fascicularisQ9GJT696 nMBindingDB
Sodium-dependent dopamine transporterHomo sapiensQ01959267 nM|303 nM267 nM|301 nM|330 nM|274 nM272 nM|371 nM|743 nM|331 nM|240 nM|68.5 nM|469 nM|419 nM|200 nM|223 nM|270 nM|720 nM|1270 nM|450 nMBindingDB
Sodium channel protein type 1/2/3 subunit alphaHomo sapiensP35498|Q99250|Q9NY4649000 nMBindingDB
Sodium-dependent noradrenaline transporterBos taurusP51143197 nMBindingDB
Sigma non-opioid intracellular receptor 1Cavia porcellusQ60492>10000 nMBindingDB
Sigma non-opioid intracellular receptor 1Rattus norvegicusQ9R0C9>10000 nMBindingDB
5-hydroxytryptamine receptor 2ARattus norvegicusP14842>10000 nMBindingDB
5-hydroxytryptamine receptor 2CRattus norvegicusP08909>10000 nMBindingDB
5-hydroxytryptamine receptor 3AMus musculusP23979>10000 nMBindingDB
5-hydroxytryptamine receptor 1AHomo sapiensP08908>10000 nMBindingDB
D(2) dopamine receptorHomo sapiensP14416>10000 nMBindingDB
Muscarinic acetylcholine receptor M1Rattus norvegicusP0848261397 nMBindingDB
Norepinephrine transporterRattus norvegicus367 nM|3830 nM|398 nM|779 nM|119 nMBindingDB
Potassium voltage-gated channel subfamily H member 2Homo sapiensQ128097244 nM|7244.36 nMBindingDB
D(1A) dopamine receptorHomo sapiensP21728>10000 nMBindingDB