| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Sodium-dependent dopamine transporter | Bos taurus | P27922 | | 139 nM|65 nM | | | BindingDB |
| Sodium-dependent serotonin transporter | Rattus norvegicus | P31652 | | 1050 nM|737 nM|1045 nM|207 nM|1059 nM | | 389 nM|304 nM|401 nM|177 nM|413 nM|96 nM|160 nM|95 nM|155 nM|130 nM|293 nM | BindingDB |
| Sodium-dependent serotonin transporter | Homo sapiens | P31645 | 318 nM|416 nM | 318 nM|325 nM|270 nM|413 nM|277 nM | | 601 nM|276 nM|297 nM|155 nM|229 nM|657 nM|632 nM | BindingDB |
| Sodium-dependent noradrenaline transporter | Homo sapiens | P23975 | 385 nM|835 nM | 385 nM|186 nM|192 nM|221 nM | | 830 nM|1115 nM|2420 nM|108 nM|645 nM|2410 nM|10700 nM|2357 nM | BindingDB |
| Transporter | Rattus norvegicus | | | 3300 nM|3520 nM|3530 nM|3825 nM | | 108 nM|186 nM|1900 nM|190 nM|2000 nM|3302 nM | BindingDB |
| Sodium-dependent dopamine transporter | Rattus norvegicus | P23977 | | 297 nM|266 nM|102 nM|1810 nM|843 nM|66 nM|150 nM|15800 nM|89 nM|511 nM|221 nM|580 nM|1450 nM|139 nM | | 690 nM|600 nM|102 nM|104 nM|150 nM|475 nM|478 nM|160 nM|275 nM|555 nM|128 nM|320 nM|280 nM|230 nM|420 nM|301 nM|259 nM|146 nM|270 nM|460 nM|187 nM|423 nM|74 nM | BindingDB |
| Sodium-dependent dopamine transporter | Mus musculus | Q61327 | | 200 nM | | 850 nM | BindingDB |
| Sodium-dependent dopamine transporter | Macaca fascicularis | Q9GJT6 | | 96 nM | | | BindingDB |
| Sodium-dependent dopamine transporter | Homo sapiens | Q01959 | 267 nM|303 nM | 267 nM|301 nM|330 nM|274 nM | | 272 nM|371 nM|743 nM|331 nM|240 nM|68.5 nM|469 nM|419 nM|200 nM|223 nM|270 nM|720 nM|1270 nM|450 nM | BindingDB |
| Sodium channel protein type 1/2/3 subunit alpha | Homo sapiens | P35498|Q99250|Q9NY46 | | 49000 nM | | | BindingDB |
| Sodium-dependent noradrenaline transporter | Bos taurus | P51143 | | | | 197 nM | BindingDB |
| Sigma non-opioid intracellular receptor 1 | Cavia porcellus | Q60492 | | | | >10000 nM | BindingDB |
| Sigma non-opioid intracellular receptor 1 | Rattus norvegicus | Q9R0C9 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 2A | Rattus norvegicus | P14842 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 2C | Rattus norvegicus | P08909 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 3A | Mus musculus | P23979 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 1A | Homo sapiens | P08908 | | | | >10000 nM | BindingDB |
| D(2) dopamine receptor | Homo sapiens | P14416 | | | | >10000 nM | BindingDB |
| Muscarinic acetylcholine receptor M1 | Rattus norvegicus | P08482 | | | | 61397 nM | BindingDB |
| Norepinephrine transporter | Rattus norvegicus | | | | | 367 nM|3830 nM|398 nM|779 nM|119 nM | BindingDB |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens | Q12809 | | 7244 nM|7244.36 nM | | | BindingDB |
| D(1A) dopamine receptor | Homo sapiens | P21728 | | | | >10000 nM | BindingDB |