| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 | Rattus norvegicus | P08482|P08483|P08485|P08911|P10980 | | 80 nM|7600 nM|68 nM | | 1010 nM|83 nM|1110 nM|3670 nM | BindingDB |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 19952.62 nM|> 20000.0 nM | | | NPASS |
| Muscarinic acetylcholine receptor M5 | Homo sapiens | P08912 | = 630.96 nM | | | 10233 nM|= 10232.93 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M4 | Homo sapiens | P08173 | = 3311.31 nM | | | | NPASS |
| Muscarinic acetylcholine receptor M3 | Homo sapiens | P20309 | = 1445.44 nM | | | | NPASS |
| Muscarinic acetylcholine receptor M2 | Rattus norvegicus | P10980 | | 8800 nM|= 8800.0 nM | = 10000.0 nM | >10000 nM|7000 nM|9800 nM|= 9800.0 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M2 | Homo sapiens | P08172 | 63000 nM|= 1000.0 nM|= 63000.0 nM | | | 12023 nM|= 12022.64 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M1 | Mus musculus | P12657 | 6900 nM|= 6900.0 nM | | | | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M1 | Homo sapiens | P11229 | 18 nM|832 nM|8792 nM|= 17.5 nM|= 831.76 nM|= 8792.0 nM|= 812.83 nM | | 2692 nM|= 2691.53 nM | 12 nM|7943 nM|6607 nM|= 6606.93 nM|= 7943.28 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor DM1 | Drosophila melanogaster | P16395 | | | | 2800 nM|2980 nM|= 2980.0 nM|= 2800.0 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor | Rattus norvegicus | P08482|P08483|P08485|P08911|P10980 | | = 7600.0 nM|= 80.0 nM|= 68.0 nM | | = 3670.0 nM|= 1010.0 nM|= 1110.0 nM|= 82.9 nM | NPASS |
| Cytochrome P450 2A6 | Homo sapiens | P11509 | | | 3600 nM|= 3600.0 nM | 3000 nM|= 3000.0 nM | BindingDB, NPASS |
| Cytochrome P450 2A13 | Homo sapiens | Q16696 | | | 3000 nM|= 3000.0 nM | 1400 nM|= 1400.0 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M1 | Rattus norvegicus | P08482 | | 4430 nM|960 nM|= 960.0 nM|= 4430.0 nM | | 9930 nM|3100 nM|= 3100.0 nM | BindingDB, NPASS |