IMPPAT Phytochemical information: 
Pilocarpine

Pilocarpine
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Muscarinic acetylcholine receptor M1/M2/M3/M4/M5Rattus norvegicusP08482|P08483|P08485|P08911|P1098080 nM|7600 nM|68 nM1010 nM|83 nM|1110 nM|3670 nMBindingDB
SARS-CoV-2Severe acute respiratory syndrome coronavirus 2> 19952.62 nM|> 20000.0 nMNPASS
Muscarinic acetylcholine receptor M5Homo sapiensP08912= 630.96 nM10233 nM|= 10232.93 nMBindingDB, NPASS
Muscarinic acetylcholine receptor M4Homo sapiensP08173= 3311.31 nMNPASS
Muscarinic acetylcholine receptor M3Homo sapiensP20309= 1445.44 nMNPASS
Muscarinic acetylcholine receptor M2Rattus norvegicusP109808800 nM|= 8800.0 nM= 10000.0 nM>10000 nM|7000 nM|9800 nM|= 9800.0 nMBindingDB, NPASS
Muscarinic acetylcholine receptor M2Homo sapiensP0817263000 nM|= 1000.0 nM|= 63000.0 nM12023 nM|= 12022.64 nMBindingDB, NPASS
Muscarinic acetylcholine receptor M1Mus musculusP126576900 nM|= 6900.0 nMBindingDB, NPASS
Muscarinic acetylcholine receptor M1Homo sapiensP1122918 nM|832 nM|8792 nM|= 17.5 nM|= 831.76 nM|= 8792.0 nM|= 812.83 nM2692 nM|= 2691.53 nM12 nM|7943 nM|6607 nM|= 6606.93 nM|= 7943.28 nMBindingDB, NPASS
Muscarinic acetylcholine receptor DM1Drosophila melanogasterP163952800 nM|2980 nM|= 2980.0 nM|= 2800.0 nMBindingDB, NPASS
Muscarinic acetylcholine receptorRattus norvegicusP08482|P08483|P08485|P08911|P10980= 7600.0 nM|= 80.0 nM|= 68.0 nM= 3670.0 nM|= 1010.0 nM|= 1110.0 nM|= 82.9 nMNPASS
Cytochrome P450 2A6Homo sapiensP115093600 nM|= 3600.0 nM3000 nM|= 3000.0 nMBindingDB, NPASS
Cytochrome P450 2A13Homo sapiensQ166963000 nM|= 3000.0 nM1400 nM|= 1400.0 nMBindingDB, NPASS
Muscarinic acetylcholine receptor M1Rattus norvegicusP084824430 nM|960 nM|= 960.0 nM|= 4430.0 nM9930 nM|3100 nM|= 3100.0 nMBindingDB, NPASS