| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM | | | NPASS |
| Matrix protein 2 | InflueA virus (strain A/Udorn/307/1972 H3N2) | P0DOF8 | 660 nM | 16000 nM|4700 nM|12500 nM|16100 nM | 2170 nM|9000 nM|210000 nM|12000 nM | | BindingDB |
| Matrix protein 2 [1-96] | InflueA virus (strain A/Udorn/1972 H3N2) | P0DOF5 | | 16000 nM|199900 nM | | | BindingDB |
| Multidrug and toxin extrusion protein 1 | Homo sapiens | Q96FL8 | | 37800 nM|= 37800.0 nM | | | BindingDB, NPASS |
| NON-PROTEIN TARGET | | | > 500000.0 nM|> 100000.0 nM|= 64200.0 nM|= 240000.0 nM|= 1400.0 nM|= 500.0 nM|= 450.0 nM|> 10000.0 nM|= 140.0 nM|= 2000.0 nM|= 1800.0 nM|= 40.0 nM | = 10780.0 nM|> 198340.0 nM|= 214870.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 5670.0 nM | | | NPASS |
| Sigma non-opioid intracellular receptor 1 | Homo sapiens | Q99720 | | | | 20 nM | BindingDB |
| Trypanosoma brucei rhodesiense | Trypanosoma brucei rhodesiense | | | = 52760.0 nM | | | NPASS |
| Solute carrier family 22 member 1 | Homo sapiens | O15245 | | = 39600.0 nM | | | NPASS |
| Solute carrier family 22 member 1 | Rattus norvegicus | Q63089 | | 280000 nM|500000 nM|76300 nM|= 76300.0 nM|= 280000.0 nM|= 500000.0 nM | | | BindingDB, NPASS |
| Solute carrier family 22 member 2 | Homo sapiens | O15244 | | 23000 nM|= 23000.0 nM|= 45900.0 nM | | | BindingDB, NPASS |
| Solute carrier family 22 member 2 | Rattus norvegicus | Q9R0W2 | | 210000 nM|290000 nM|270900 nM|= 270900.0 nM|= 210000.0 nM|= 290000.0 nM | | | BindingDB, NPASS |
| Trypanosoma brucei | Trypanosoma brucei | | | > 130000.0 nM|> 132000.0 nM | | | NPASS |
| Matrix protein 2 | InflueA virus (strain A/Chicken/Weybridge H7N7) | P05778 | | | 320 nM | | BindingDB |
| Trypanosoma cruzi | Trypanosoma cruzi | | | = 371300.0 nM | | | NPASS |
| Sigma opioid receptor | Homo sapiens | Q99720 | | | | = 20.25 nM | NPASS |
| Matrix protein 2 | InflueA virus | P06821 | | = 16000.0 nM|= 199900.0 nM | = 320.0 nM|= 2170.0 nM | | NPASS |
| Influenza virus A matrix protein M2 | InflueA virus (A/Udorn/307/1972(H3N2)) | P0DOF8 | = 660.0 nM | > 500000.0 nM|= 16000.0 nM|= 16100.0 nM|= 4700.0 nM|= 12500.0 nM | = 12000.0 nM|= 2170.0 nM|= 210000.0 nM|= 9000.0 nM | | NPASS |
| Leishmania donovani | Leishmadonovani | | | > 595030.0 nM|> 198340.0 nM | | | NPASS |
| Epithelial cells | | | > 1333000.0 nM | | | | NPASS |
| Glutamate NMDA receptor | Rattus norvegicus | Q9R1M7 | | = 92000.0 nM|= 358000.0 nM | | | NPASS |
| MDCK | Canis lupus familiaris | | = 1100.0 nM | = 660900.0 nM|> 1321800.0 nM|= 56.0 ug.mL-1 | | | NPASS |
| Glutamate NMDA receptor; Grin1/Grin2a | Rattus norvegicus | P35439|Q00959 | | = 40000.0 nM | | | NPASS |
| Glutamate [NMDA] receptor | Homo sapiens | | | | | = 10500.0 nM | NPASS |
| Glutamate receptor ionotropic, NMDA 1 | Rattus norvegicus | P35439 | | | | >10000 nM | BindingDB |
| Glutamate receptor ionotropic, NMDA 1/2A | Homo sapiens | Q05586|Q12879 | | | | 10000 nM | BindingDB |
| Glutamate NMDA receptor; GRIN1/GRIN2A | Homo sapiens | Q12879 | | | | = 10000.0 nM | NPASS |
| Influenza A virus | InflueA virus | | = 1980.0 nM|= 0.054 ug.mL-1|> 100000.0 nM|= 2000.0 nM|= 800.0 nM|= 400.0 nM|= 20000.0 nM|= 19000.0 nM|= 7000.0 nM|= 9200.0 nM|= 87.0 ug.mL-1|= 101.0 ug.mL-1|= 115.0 ug.mL-1|= 117.0 ug.mL-1|= 18.0 ug.mL-1|= 44.0 ug.mL-1|= 0.3 ug.mL-1|= 0.2 ug.mL-1|= 4100.0 nM|= 154000.0 nM|= 5000.0 nM|= 89000.0 nM|= 2300.0 nM|= 61000.0 nM|= 11000.0 nM|= 5100.0 nM|= 3400.0 nM|= 450.0 nM|= 208000.0 nM|= 224000.0 nM|= 65500.0 nM|= 22500.0 nM|= 1900.0 nM|= 600.0 nM|= 300.0 nM|= 17000.0 nM|= 140000.0 nM|= 840.0 nM|= 820.0 nM|= 24000.0 nM|= 340.0 nM|= 2770.0 nM|> 500000.0 nM|> 200000.0 nM|= 4280.0 nM|> 20510.0 nM|= 2200.0 nM|= 1400.0 nM|= 1800.0 nM|= 1000.0 nM|= 480.0 nM|= 780.0 nM|= 230.0 nM|= 22600.0 nM|= 430.0 nM|> 532700.0 nM|= 6400.0 nM | = 1250.0 nM|= 15.0 ug.mL-1|= 50000.0 nM|= 0.92 ug.mL-1|= 5960.0 nM|= 21110.0 nM|= 2380.0 nM|= 2220.0 nM|> 50000.0 nM|= 3840.0 nM|= 820.0 nM|> 200000.0 nM|> 100000.0 nM|= 337200.0 nM|= 13000.0 nM|= 64000.0 nM|= 480.0 nM|= 330.0 nM | | | NPASS |
| Influenza A virus (A/PR/8/34(H1N1)) | InflueA virus (A/Puerto Rico/8/1934(H1N1)) | | = 77000.0 nM|= 45000.0 nM|= 35000.0 nM|= 7600.0 nM|= 53000.0 nM|= 212000.0 nM|= 75000.0 nM|= 58000.0 nM|= 38000.0 nM|= 34000.0 nM|= 24000.0 nM|= 30000.0 nM|= 111000.0 nM|> 10000.0 nM|> 80000.0 nM|= 224000.0 nM|= 453000.0 nM|> 20000.0 nM|= 44000.0 nM|= 47000.0 nM|= 85000.0 nM|= 178000.0 nM|> 100000.0 nM|= 26000.0 nM|> 500000.0 nM | = 64200.0 nM|= 64000.0 nM | | | NPASS |
| Influenza A virus (H5N1) | InflueA virus (H5N1) | | | = 3840.0 nM | | | NPASS |
| Influenza A virus H3N2 | InflueA virus H3N2 | | = 100000.0 nM|= 75300.0 nM|= 2700.0 nM|= 1500.0 nM|= 1600.0 nM|= 2000.0 nM|= 30.0 nM|= 200.0 nM|= 3800.0 nM|= 1200.0 nM | = 630.0 nM|= 500.0 nM | | | NPASS |
| Influenza B virus | InflueB virus | | > 100000.0 nM|> 500000.0 nM|> 200.0 ug.mL-1|> 200000.0 nM|= 143840.0 nM|> 400000.0 nM | = 50000.0 nM | | | NPASS |
| Influenza B virus (B/Lee/40) | InflueB virus (B/Lee/40) | | > 100000.0 nM | | | | NPASS |
| HeLa | Homo sapiens | | | > 660900.0 nM | | | NPASS |